Optimization of 1,3,4-Benzotriazepine-Based CCK2 Antagonists to Obtain Potent, Orally Active Inhibitors of Gastrin-Mediated Gastric Acid Secretion
McDonald, Iain M, Black, James W, Buck, Ildiko M, Dunstone, David J, Griffin, Eric P, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Lilley, Elliot J, Linney, Ian D, Pether, Michael J, Roberts, Sonia P, Shaxted, Mark E, Spencer, John, Steel, Katherine I. M, Sykes, David A, Walker, Martin K, Watt, Gillian F, Wright, Laurence, Wright, Paul T, Xun, Wei
Published in Journal of medicinal chemistry (28.06.2007)
Published in Journal of medicinal chemistry (28.06.2007)
Get full text
Journal Article
Design, Synthesis, and Structure−Activity Relationships of Novel Non-Imidazole Histamine H3 Receptor Antagonists
Linney, Ian D, Buck, Ildiko M, Harper, Elaine A, Kalindjian, S. Barret, Pether, Michael J, Shankley, Nigel P, Watt, Gillian F, Wright, Paul T
Published in Journal of medicinal chemistry (15.06.2000)
Published in Journal of medicinal chemistry (15.06.2000)
Get full text
Journal Article
Characterization of SNARE Proteins in Human Pituitary Adenomas: Targeted Secretion Inhibitors as a New Strategy for the Treatment of Acromegaly?
Garcia, Edwin A, Trivellin, Giampaolo, Aflorei, Elena D, Powell, Michael, Grieve, Joana, Alusi, Ghassan, Pobereskin, Luis, Shariati, Babak, Cudlip, Simon, Roncaroli, Federico, Mendoza, Nigel, Grossman, Ashley B, Harper, Elaine A, Korbonits, Márta
Published in The journal of clinical endocrinology and metabolism (01.12.2013)
Published in The journal of clinical endocrinology and metabolism (01.12.2013)
Get full text
Journal Article
Discovery and Characterization of Novel, Potent, Non-Peptide Parathyroid Hormone-1 Receptor Antagonists
McDonald, Iain M, Austin, Carol, Buck, Ildiko M, Dunstone, David J, Gaffen, John, Griffin, Eric, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Patel, Dipa, Pether, Michael J, Raynor, Michelle, Roberts, Sonia P, Shaxted, Mark E, Spencer, John, Steel, Katherine I. M, Sykes, David A, Wright, Paul T, Xun, Wei
Published in Journal of medicinal chemistry (04.10.2007)
Published in Journal of medicinal chemistry (04.10.2007)
Get full text
Journal Article
Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template
SPENCER, John, GAFFEN, John, GRIFFIN, Eric, HARPER, Elaine A, LINNEY, Ian D, MCDONALD, Iain M, ROBERTS, Sonia P, SHAXTED, Mark E, ADATIA, Trushar, BASHALL, Alan
Published in Bioorganic & medicinal chemistry (15.03.2008)
Published in Bioorganic & medicinal chemistry (15.03.2008)
Get full text
Journal Article
Novel, Achiral 1,3,4-Benzotriazepine Analogues of 1,4-Benzodiazepine-Based CCK2 Antagonists That Display High Selectivity over CCK1 Receptors
McDonald, Iain M, Austin, Carol, Buck, Ildiko M, Dunstone, David J, Griffin, Eric, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Linney, Ian D, Low, Caroline M. R, Pether, Michael J, Spencer, John, Wright, Paul T, Adatia, Trushar, Bashall, Alan
Published in Journal of medicinal chemistry (06.04.2006)
Published in Journal of medicinal chemistry (06.04.2006)
Get full text
Journal Article
Optimization of the in Vitro and in Vivo Properties of a Novel Series of 2,4,5-Trisubstituted Imidazoles as Potent Cholecystokinin-2 (CCK2) Antagonists
Buck, Ildiko M, Black, James W, Cooke, Tracey, Dunstone, David J, Gaffen, John D, Griffin, Eric P, Harper, Elaine A, Hull, Robert A. D, Kalindjian, S. Barret, Lilley, Elliot J, Linney, Ian D, Low, Caroline M. R, McDonald, Iain M, Pether, Michael J, Roberts, Sonia P, Shankley, Nigel P, Shaxted, Mark E, Steel, Katherine I. M, Sykes, David A, Tozer, Matthew J, Watt, Gillian F, Walker, Martin K, Wright, Laurence, Wright, Paul T
Published in Journal of medicinal chemistry (03.11.2005)
Published in Journal of medicinal chemistry (03.11.2005)
Get full text
Journal Article
Erratum to “Achiral, selective CCK2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template” [Bioorg. Med. Chem. 16 (2008) 2974–2983]
Spencer, John, Gaffen, John, Griffin, Eric, Harper, Elaine A., Linney, Ian D., McDonald, Iain M., Roberts, Sonia P., Shaxted, Mark E., Adatia, Trushar, Bashall, Alan
Published in Bioorganic & medicinal chemistry (15.08.2008)
Published in Bioorganic & medicinal chemistry (15.08.2008)
Get full text
Journal Article
Achiral, selective CCK 2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template
Spencer, John, Gaffen, John, Griffin, Eric, Harper, Elaine A., Linney, Ian D., McDonald, Iain M., Roberts, Sonia P., Shaxted, Mark E., Adatia, Trushar, Bashall, Alan
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
Get full text
Journal Article
Erratum to “Achiral, selective CCK 2 receptor antagonists based on a 1,3,5-benzotriazepine-2,4-dione template” [Bioorg. Med. Chem. 16 (2008) 2974–2983]
Spencer, John, Gaffen, John, Griffin, Eric, Harper, Elaine A., Linney, Ian D., McDonald, Iain M., Roberts, Sonia P., Shaxted, Mark E., Adatia, Trushar, Bashall, Alan
Published in Bioorganic & medicinal chemistry (2008)
Published in Bioorganic & medicinal chemistry (2008)
Get full text
Journal Article
Optimization of 1,3,4-benzotriazepine-based CCK(2) antagonists to obtain potent, orally active inhibitors of gastrin-mediated gastric acid secretion
McDonald, Iain M, Black, James W, Buck, Ildiko M, Dunstone, David J, Griffin, Eric P, Harper, Elaine A, Hull, Robert A D, Kalindjian, S Barret, Lilley, Elliot J, Linney, Ian D, Pether, Michael J, Roberts, Sonia P, Shaxted, Mark E, Spencer, John, Steel, Katherine I M, Sykes, David A, Walker, Martin K, Watt, Gillian F, Wright, Laurence, Wright, Paul T, Xun, Wei
Published in Journal of medicinal chemistry (28.06.2007)
Get full text
Published in Journal of medicinal chemistry (28.06.2007)
Journal Article
Optimization of 1,3,4-Benzotriazepine-Based CCK 2 Antagonists to Obtain Potent, Orally Active Inhibitors of Gastrin-Mediated Gastric Acid Secretion
McDonald, Iain M., Black, James W., Buck, Ildiko M., Dunstone, David J., Griffin, Eric P., Harper, Elaine A., Hull, Robert A. D., Kalindjian, S. Barret, Lilley, Elliot J., Linney, Ian D., Pether, Michael J., Roberts, Sonia P., Shaxted, Mark E., Spencer, John, Steel, Katherine I. M., Sykes, David A., Walker, Martin K., Watt, Gillian F., Wright, Laurence, Wright, Paul T., Xun, Wei
Published in Journal of medicinal chemistry (01.06.2007)
Published in Journal of medicinal chemistry (01.06.2007)
Get full text
Journal Article
Novel, achiral 1,3,4-benzotriazepine analogues of 1,4-benzodiazepine-based CCK(2) antagonists that display high selectivity over CCK(1) receptors
McDonald, Iain M, Austin, Carol, Buck, Ildiko M, Dunstone, David J, Griffin, Eric, Harper, Elaine A, Hull, Robert A D, Kalindjian, S Barret, Linney, Ian D, Low, Caroline M R, Pether, Michael J, Spencer, John, Wright, Paul T, Adatia, Trushar, Bashall, Alan
Published in Journal of medicinal chemistry (06.04.2006)
Get full text
Published in Journal of medicinal chemistry (06.04.2006)
Journal Article
Novel, Achiral 1,3,4-Benzotriazepine Analogues of 1,4-Benzodiazepine-Based CCK 2 Antagonists That Display High Selectivity over CCK 1 Receptors
McDonald, Iain M., Austin, Carol, Buck, Ildiko M., Dunstone, David J., Griffin, Eric, Harper, Elaine A., Hull, Robert A. D., Kalindjian, S. Barret, Linney, Ian D., Low, Caroline M. R., Pether, Michael J., Spencer, John, Wright, Paul T., Adatia, Trushar, Bashall, Alan
Published in Journal of medicinal chemistry (01.04.2006)
Published in Journal of medicinal chemistry (01.04.2006)
Get full text
Journal Article
From histamine to imidazolylalkyl-sulfonamides: The design of a novel series of histamine H 3-receptor antagonists
Tozer, Matthew J., Harper, Elaine A., Kalindjian, S.Barret, Pether, Michael J., Shankley, Nigel P., Watt, Gillian F.
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
Published in Bioorganic & medicinal chemistry letters (05.07.1999)
Get full text
Journal Article