Phospholipidosis as a Function of Basicity, Lipophilicity, and Volume of Distribution of Compounds
Hanumegowda, Umesh M, Wenke, Gottfried, Regueiro-Ren, Alicia, Yordanova, Roumyana, Corradi, John P, Adams, Stephen P
Published in Chemical research in toxicology (19.04.2010)
Published in Chemical research in toxicology (19.04.2010)
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Synthesis, Structure–Activity Relationships, and In Vivo Evaluation of Novel C‑17 Amine Derivatives Based on GSK3640254 as HIV‑1 Maturation Inhibitors with Broad Spectrum Activity
Hartz, Richard A., Xu, Li, Sit, Sing-Yuen, Chen, Jie, Venables, Brian L., Lin, Zeyu, Zhang, Sharon, Li, Zhufang, Parker, Dawn, Simmons, Tara S., Jenkins, Susan, Hanumegowda, Umesh M., Dicker, Ira, Krystal, Mark, Meanwell, Nicholas A., Regueiro-Ren, Alicia
Published in Journal of medicinal chemistry (08.12.2022)
Published in Journal of medicinal chemistry (08.12.2022)
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Thrombin and Protease-Activated Receptor-1 Agonists Promote Lipopolysaccharide-Induced Hepatocellular Injury in Perfused Livers
Copple, Bryan L, Moulin, Frederic, Hanumegowda, Umesh M, Ganey, Patricia E, Roth, Robert A
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
Published in The Journal of pharmacology and experimental therapeutics (01.05.2003)
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Multiplexed assay panel of cytotoxicity in HK-2 cells for detection of renal proximal tubule injury potential of compounds
Wu, Yang, Connors, David, Barber, Lauren, Jayachandra, Sukhanya, Hanumegowda, Umesh M., Adams, Stephen P.
Published in Toxicology in vitro (01.09.2009)
Published in Toxicology in vitro (01.09.2009)
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Discovery and Preclinical Evaluation of BMS-955829, a Potent Positive Allosteric Modulator of mGluR5
Yang, Fukang, Snyder, Lawrence B, Balakrishnan, Anand, Brown, Jeffrey M, Sivarao, Digavalli V, Easton, Amy, Fernandes, Alda, Gulianello, Michael, Hanumegowda, Umesh M, Huang, Hong, Huang, Yanling, Jones, Kelli M, Li, Yu-Wen, Matchett, Michele, Mattson, Gail, Miller, Regina, Santone, Kenneth S, Senapati, Arun, Shields, Eric E, Simutis, Frank J, Westphal, Ryan, Whiterock, Valerie J, Bronson, Joanne J, Macor, John E, Degnan, Andrew P
Published in ACS medicinal chemistry letters (10.03.2016)
Published in ACS medicinal chemistry letters (10.03.2016)
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Discovery of Indazoles as Potent, Orally Active Dual Neurokinin 1 Receptor Antagonists and Serotonin Transporter Inhibitors for the Treatment of Depression
Degnan, Andrew P, Tora, George O, Huang, Hong, Conlon, David A, Davis, Carl D, Hanumegowda, Umesh M, Hou, Xiaoping, Hsiao, Yi, Hu, Joanna, Krause, Rudolph, Li, Yu-Wen, Newton, Amy E, Pieschl, Rick L, Raybon, Joseph, Rosner, Thorsten, Sun, Jung-Hui, Taber, Matthew T, Taylor, Sarah J, Wong, Michael K, Zhang, Huiping, Lodge, Nicholas J, Bronson, Joanne J, Macor, John E, Gillman, Kevin W
Published in ACS chemical neuroscience (21.12.2016)
Published in ACS chemical neuroscience (21.12.2016)
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Endothelial Cell Injury and Coagulation System Activation during Synergistic Hepatotoxicity from Monocrotaline and Bacterial Lipopolysaccharide Coexposure
Yee, Steven B., Hanumegowda, Umesh M., Copple, Bryan L., Shibuya, Masabumi, Ganey, Patricia E., Roth, Robert A.
Published in Toxicological sciences (01.07.2003)
Published in Toxicological sciences (01.07.2003)
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