A Review of HER4 (ErbB4) Kinase, Its Impact on Cancer, and Its Inhibitors
El-Gamal, Mohammed I, Mewafi, Nada H, Abdelmotteleb, Nada E, Emara, Minnatullah A, Tarazi, Hamadeh, Sbenati, Rawan M, Madkour, Moustafa M, Zaraei, Seyed-Omar, Shahin, Afnan I, Anbar, Hanan S
Published in Molecules (Basel, Switzerland) (05.12.2021)
Published in Molecules (Basel, Switzerland) (05.12.2021)
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Journal Article
Design and synthesis of novel anti-urease imidazothiazole derivatives with promising antibacterial activity against Helicobacter pylori
Shahin, Afnan I, Zaib, Sumera, Zaraei, Seyed-Omar, Kedia, Reena A, Anbar, Hanan S, Younas, Muhammad Tayyab, Al-Tel, Taleb H, Khoder, Ghalia, El-Gamal, Mohammed I
Published in PloS one (02.06.2023)
Published in PloS one (02.06.2023)
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Journal Article
Anti-proliferative activity of RIHMS-Qi-23 against MCF-7 breast cancer cell line is through inhibition of cell proliferation and senescence but not inhibition of targeted kinases
El-Gamal, Randa, Elfarrash, Sara, EL-Nablaway, Mohammad, Salem, Asmaa Ahmed, Zaraei, Seyed-Omar, Anbar, Hanan S, Shoma, Ashraf, El-Gamal, Mohammed I
Published in BMC cancer (02.11.2023)
Published in BMC cancer (02.11.2023)
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Journal Article
Comparison of the effects of levocetirizine and losartan on diabetic nephropathy and vascular dysfunction in streptozotocin-induced diabetic rats
Anbar, Hanan S., Shehatou, George S.G., Suddek, Ghada M., Gameil, Nariman M.
Published in European journal of pharmacology (05.06.2016)
Published in European journal of pharmacology (05.06.2016)
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Journal Article
Imidazothiazole-based potent inhibitors of V600E-B-RAF kinase with promising anti-melanoma activity: biological and computational studies
Anbar, Hanan S., El-Gamal, Mohammed I., Tarazi, Hamadeh, Lee, Bong S., Jeon, Hong R., Kwon, Dow, Oh, Chang-Hyun
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
Published in Journal of enzyme inhibition and medicinal chemistry (01.01.2020)
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Journal Article
FMS Kinase Inhibitors: Current Status and Future Prospects
El-Gamal, Mohammed I., Anbar, Hanan S., Yoo, Kyung Ho, Oh, Chang-Hyun
Published in Medicinal research reviews (01.05.2013)
Published in Medicinal research reviews (01.05.2013)
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Journal Article
Novel Anti-Acanthamoebic Activities of Irosustat and STX140 and Their Nanoformulations
Siddiqui, Ruqaiyyah, Rawas-Qalaji, Mutasem, El-Gamal, Mohammed I, Sajeev, Sreedevi, Jagal, Jayalakshmi, Zaraei, Seyed-Omar, Sbenati, Rawan M, Anbar, Hanan S, Dohle, Wolfgang, Potter, Barry V L, Khan, Naveed Ahmed
Published in Antibiotics (Basel) (01.03.2023)
Published in Antibiotics (Basel) (01.03.2023)
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Journal Article
Current status and future prospects of p38α/MAPK14 kinase and its inhibitors
Madkour, Moustafa M., Anbar, Hanan S., El-Gamal, Mohammed I.
Published in European journal of medicinal chemistry (05.03.2021)
Published in European journal of medicinal chemistry (05.03.2021)
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Journal Article
Synthesis, biological evaluation, and docking studies of novel pyrrolo[2,3-b]pyridine derivatives as both ectonucleotide pyrophosphatase/phosphodiesterase inhibitors and antiproliferative agents
Ullah, Saif, El-Gamal, Mohammed I., El-Gamal, Randa, Pelletier, Julie, Sévigny, Jean, Shehata, Mahmoud K., Anbar, Hanan S., Iqbal, Jamshed
Published in European journal of medicinal chemistry (05.05.2021)
Published in European journal of medicinal chemistry (05.05.2021)
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Journal Article
The wound healing and hypoglycemic activates of date palm (Phoenix dactylifera) leaf extract and saponins in diabetic and normal rats
Anbar, Hanan S, Shehab, Naglaa Gamil, Yasin, Ayah, Shaar, Lana Mazen, Ashraf, Ruba, Rahi, Zahraa, Alamir, Raneem, Alsabbagh, Deema, Thabet, Aya, Altaas, Israa, Lozon, Yosra A, El Rouby, Nadia M M, Shahiwala, Aliasgar
Published in PloS one (23.09.2024)
Published in PloS one (23.09.2024)
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Journal Article
Design and discovery of urease and Helicobacter pylori inhibitors based on benzofuran/benzothiophene-sulfonate and sulfamate scaffolds for the treatment of ureolytic bacterial infections
Hashem, Omar, Zaib, Sumera, Zaraei, Seyed-Omar, Javed, Hira, Kedia, Reena A., Anbar, Hanan S., Khan, Imtiaz, Ravi, Anil, El-Gamal, Mohammed I., Khoder, Ghalia
Published in International journal of biological macromolecules (01.06.2024)
Published in International journal of biological macromolecules (01.06.2024)
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Journal Article
Sulfamates in drug design and discovery: Pre-clinical and clinical investigations
Zaraei, Seyed-Omar, Abduelkarem, Abduelmula R., Anbar, Hanan S., Kobeissi, Sara, Mohammad, Miami, Ossama, Aya, El-Gamal, Mohammed I.
Published in European journal of medicinal chemistry (01.10.2019)
Published in European journal of medicinal chemistry (01.10.2019)
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Journal Article
Promising drug candidates for the treatment of polycystic ovary syndrome (PCOS) as alternatives to the classical medication metformin
Anbar, Hanan S., Vahora, Nisha Yarifbhai, Shah, Hajra laghman, Azam, Mariyam Mohammed, Islam, Tamanna, Hersi, Fatima, Omar, Hany A., Dohle, Wolfgang, Potter, Barry V.L., El-Gamal, Mohammed I.
Published in European journal of pharmacology (05.12.2023)
Published in European journal of pharmacology (05.12.2023)
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Journal Article
Eicosapentaenoic and docosahexaenoic acids attenuate methotrexate-induced apoptosis and suppression of splenic T, B-Lymphocytes and macrophages with modulation of expression of CD3, CD20 and CD68
Elsayed, Hassan Reda Hassan, Anbar, Hanan S., Rabei, Mohammed R., Adel, Mohamed, El-Gamal, Randa
Published in Tissue & cell (01.10.2021)
Published in Tissue & cell (01.10.2021)
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Journal Article
Synthesis, biological evaluation, and stability studies of raloxifene mono- and bis-sulfamates as dual-targeting agents
Zaraei, Seyed-Omar, Dohle, Wolfgang, Anbar, Hanan S., El-Gamal, Randa, Leblond, Bertrand, Foster, Paul A., Al-Tel, Taleb H., Potter, Barry V.L., El-Gamal, Mohammed I.
Published in Bioorganic & medicinal chemistry (01.03.2024)
Published in Bioorganic & medicinal chemistry (01.03.2024)
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Journal Article
Discovery of first-in-class imidazothiazole-based potent and selective ErbB4 (HER4) kinase inhibitors
Zaraei, Seyed-Omar, Sbenati, Rawan M., Alach, Nour N., Anbar, Hanan S., El-Gamal, Randa, Tarazi, Hamadeh, Shehata, Mahmoud K., Abdel-Maksoud, Mohammed S., Oh, Chang-Hyun, El-Gamal, Mohammed I.
Published in European journal of medicinal chemistry (15.11.2021)
Published in European journal of medicinal chemistry (15.11.2021)
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Journal Article