The SERM/SERD bazedoxifene disrupts ESR1 helix 12 to overcome acquired hormone resistance in breast cancer cells
Fanning, Sean W, Jeselsohn, Rinath, Dharmarajan, Venkatasubramanian, Mayne, Christopher G, Karimi, Mostafa, Buchwalter, Gilles, Houtman, René, Toy, Weiyi, Fowler, Colin E, Han, Ross, Lainé, Muriel, Carlson, Kathryn E, Martin, Teresa A, Nowak, Jason, Nwachukwu, Jerome C, Hosfield, David J, Chandarlapaty, Sarat, Tajkhorshid, Emad, Nettles, Kendall W, Griffin, Patrick R, Shen, Yang, Katzenellenbogen, John A, Brown, Myles, Greene, Geoffrey L
Published in eLife (29.11.2018)
Published in eLife (29.11.2018)
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Journal Article
Stereospecific lasofoxifene derivatives reveal the interplay between estrogen receptor alpha stability and antagonistic activity in ESR1 mutant breast cancer cells
Hosfield, David J, Weber, Sandra, Li, Nan-Sheng, Suavage, Madline, Joiner, Carstyn F, Hancock, Govinda R, Sullivan, Emily A, Ndukwe, Estelle, Han, Ross, Cush, Sydney, Lainé, Muriel, Mader, Sylvie C, Greene, Geoffrey L, Fanning, Sean W
Published in eLife (16.05.2022)
Published in eLife (16.05.2022)
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High-risk human papillomavirus genotype distribution and attribution to cervical cancer and precancerous lesions in a rural Chinese population
Zhao, Xue Lian, Hu, Shang Ying, Zhang, Qian, Dong, Li, Feng, Rui Mei, Han, Ross, Zhao, Fang Hui
Published in Journal of gynecologic oncology (01.07.2017)
Published in Journal of gynecologic oncology (01.07.2017)
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Abstract 2472: Effective ER antagonists resist conformational restrictions imposed by somatic mutation but do not correlate with effects on receptor stability in live cells
Hosfield, David, Li, Nan-Sheng, Han, Ross, Laine, Muriel, Weber, Sandra, Sauvage, Madaline, Madar, Sylvie, Greene, Geoffrey, Fanning, Sean
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Safety and efficacy of repeat Y90 radioembolization to the same hepatic arterial territory
Badar, Wali, Van Ha, Thuong, Zangan, Steven, Navuluri, Rakesh, Pillai, Anjana, Baker, Talia, Dalag, Leonard, Han, Ross, Ahmed, Osman
Published in British journal of radiology (01.03.2021)
Published in British journal of radiology (01.03.2021)
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Endovascular Arteriovenous Fistula Creation
Tyagi, Ravi, Han, Ross, Ahmed, Osman, Navuluri, Rakesh
Published in Advances in clinical radiology (Online) (01.09.2021)
Published in Advances in clinical radiology (Online) (01.09.2021)
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SUN-006 Lasofoxifene Achieves Potent Anti-Tumor Activity in Hormone-Resistant Breast Tumors by Maintaining High Affinity Binding for Y537S ERα
Fanning, Sean, Laine, Muriel, Greene, Marianne, Chang, Ya-Fang, Phung, Linda, Green, Bradley, Hiipakka, Richard, Han, Ross, Komm, Barry, Greene, Geoffrey
Published in Journal of the Endocrine Society (30.04.2019)
Published in Journal of the Endocrine Society (30.04.2019)
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Journal Article
Stereo-specific Lasofoxifene Derivatives Reveal the Interplay between Estrogen Receptor Alpha Stability and Antagonistic Activity in ESR1 Mutant Breast Cancer Cells
Hosfield, David J, Weber, Sandra, Nan-Sheng, Li, Suavage, Madline, Sullivan, Emily, Nduwke, Estelle, Han, Ross, Cush, Sydney, Laine, Muriel, Mader, Sylvie C, Greene, Geoffrey L, Fanning, Sean W
Published in bioRxiv (28.08.2021)
Published in bioRxiv (28.08.2021)
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