An insight on synthetic and medicinal aspects of pyrazolo[1,5-a]pyrimidine scaffold
Cherukupalli, Srinivasulu, Karpoormath, Rajshekhar, Chandrasekaran, Balakumar, Hampannavar, Girish. A., Thapliyal, Neeta, Palakollu, Venkata Narayana
Published in European journal of medicinal chemistry (27.01.2017)
Published in European journal of medicinal chemistry (27.01.2017)
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Current perspective of natural alkaloid carbazole and its derivatives as antitumor agents
Shaikh, Mahamadhanif S, Karpoormath, Rajshekhar, Thapliyal, Neeta, Rane, Rajesh A, Palkar, Mahesh B, Faya, A M, Patel, Harun M, Alwan, Wesam S, Jain, Kavita, Hampannavar, Girish A
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
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Novel series of coumarinyl substituted-thiazolidin-2,4-dione analogs as anticancer agents: design, synthesis, spectral studies and cytotoxicity evaluation
Palkar, Mahesh B, Jalalpure, Sunil S, Rane, Rajesh A, Patel, Harun M, Shaikh, Mahamadhanif S, Hampannavar, Girish A, Alwan, Wesam S, Bolakatti, Girish S, Karpoormath, Rajshekhar
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
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An insight into purine, tyrosine and tryptophan derived marine antineoplastic alkaloids
Palkar, Mahesh B, Rane, Rajesh A, Thapliyal, Neeta, Shaikh, Mahamadhanif S, Alwan, Wesam S, Jain, Kavita S, Karunanidhi, Sivanandhan, Patel, Harun M, Hampannavar, Girish A, Karpoormath, Rajshekhar
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
Published in Anti-cancer agents in medicinal chemistry (01.01.2015)
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An appraisal on synthetic and pharmaceutical perspectives of pyrazolo[4,3-d]pyrimidine scaffold
Cherukupalli, Srinivasulu, Hampannavar, Girish A., Chinnam, Sampath, Chandrasekaran, Balakumar, Sayyad, Nisar, Kayamba, Francis, Reddy Aleti, Rajeshwar, Karpoormath, Rajshekhar
Published in Bioorganic & medicinal chemistry (15.01.2018)
Published in Bioorganic & medicinal chemistry (15.01.2018)
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Discovery of novel N-methyl carbazole tethered rhodanine derivatives as direct inhibitors of Mycobacterium tuberculosis InhA
Shaikh, Mahamadhanif S., Kanhed, Ashish M., Chandrasekaran, Balakumar, Palkar, Mahesh B., Agrawal, Nikhil, Lherbet, Christian, Hampannavar, Girish A., Karpoormath, Rajshekhar
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
Published in Bioorganic & medicinal chemistry letters (15.08.2019)
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Dehydrozingerone Inspired Styryl Hydrazine Thiazole Hybrids as Promising Class of Antimycobacterial Agents
Hampannavar, Girish A, Karpoormath, Rajshekhar, Palkar, Mahesh B, Shaikh, Mahamadhanif S, Chandrasekaran, Balakumar
Published in ACS medicinal chemistry letters (14.07.2016)
Published in ACS medicinal chemistry letters (14.07.2016)
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Ligand- and structure-based in silico studies to identify kinesin spindle protein (KSP) inhibitors as potential anticancer agents
Balakumar, Chandrasekaran, Ramesh, Muthusamy, Tham, Chuin Lean, Khathi, Samukelisiwe Pretty, Kozielski, Frank, Srinivasulu, Cherukupalli, Hampannavar, Girish A., Sayyad, Nisar, Soliman, Mahmoud E., Karpoormath, Rajshekhar
Published in Journal of biomolecular structure & dynamics (26.10.2018)
Published in Journal of biomolecular structure & dynamics (26.10.2018)
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Journal Article
Design, synthesis and QSAR studies of 2-amino benzo[d]thiazolyl substituted pyrazol-5-ones: novel class of promising antibacterial agents
Palkar, Mahesh B., Patil, Aniket, Hampannavar, Girish A., Shaikh, Mahamadhanif S., Patel, Harun M., Kanhed, Ashish M., Yadav, Mange Ram, Karpoormath, Rajshekhar V.
Published in Medicinal chemistry research (01.09.2017)
Published in Medicinal chemistry research (01.09.2017)
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Synthesis of 4,6-disubstituted pyrazolo[3,4-d]pyrimidine analogues: Cyclin-dependent kinase 2 (CDK2) inhibition, molecular docking and anticancer evaluation
Cherukupalli, Srinivasulu, Chandrasekaran, Balakumar, Aleti, Rajeshwar Reddy, Sayyad, Nisar, Hampannavar, Girish A., Merugu, Srinivas Reddy, Rachamalla, Harikrishna Reddy, Banerjee, Rajkumar, Karpoormath, Rajshekhar
Published in Journal of molecular structure (15.01.2019)
Published in Journal of molecular structure (15.01.2019)
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DEHYDROZINGERONE INSPIRED STYRYL HYDRAZINE THIAZOLE HYBRIDS AS PROMISING CLASS OF ANTI-MYCOBACTERIAL AGENTS
Aleti, Rajeshwar Reddy, Hampannavar, Girish A, Karpoormath, Rajshekhar V, Shaikh, Mahamadhanif B, Chandrasekaran, Balakumar
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
Published in Proceedings for Annual Meeting of The Japanese Pharmacological Society (2018)
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Journal Article
Design and synthesis of novel carbazolo–thiazoles as potential anti-mycobacterial agents using a molecular hybridization approach
Shaikh, Mahamadhanif S., Palkar, Mahesh B., Patel, Harun M., Rane, Rajesh A., Alwan, Wesam S., Shaikh, Mahidansha M., Shaikh, Iqbal M., Hampannavar, Girish A., Karpoormath, Rajshekhar
Published in RSC advances (2014)
Published in RSC advances (2014)
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Recent Advances on the s‐Triazine Scaffold with Emphasis on Synthesis, Structure‐Activity and Pharmacological Aspects: A Concise Review
Majeed Ganai, Ab, Khan Pathan, Tabasum, Hampannavar, Girish A., Pawar, Chandrakant, Obakachi, Vincent A., Kushwaha, Babita, Deshwar Kushwaha, Narva, Karpoormath, Rajshekhar
Published in ChemistrySelect (Weinheim) (17.02.2021)
Published in ChemistrySelect (Weinheim) (17.02.2021)
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Novel series of phenylalanine analogs endowed with promising anti-inflammatory activity: synthesis, pharmacological evaluation, and computational insights
Palkar, Mahesh B., Praveen, D. M., Ronad, Pradeepkumar M., Viswanathswamy, A. H. M., Rane, Rajesh A., Patel, Harun M., Shaikh, Mahamadhanif S., Hampannavar, Girish A., Jain, Kavita S., Karpoormath, Rajshekhar
Published in Medicinal chemistry research (01.05.2015)
Published in Medicinal chemistry research (01.05.2015)
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Design and synthesis of novel carbazolo-thiazoles as potential anti-mycobacterial agents using a molecular hybridization approachElectronic supplementary information (ESI) available. See DOI: 10.1039/c4ra11752b
Shaikh, Mahamadhanif S, Palkar, Mahesh B, Patel, Harun M, Rane, Rajesh A, Alwan, Wesam S, Shaikh, Mahidansha M, Shaikh, Iqbal M, Hampannavar, Girish A, Karpoormath, Rajshekhar
Year of Publication 19.11.2014
Year of Publication 19.11.2014
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