Neuropharmacokinetic visualization of regional and subregional unbound antipsychotic drug transport across the blood-brain barrier
Luptáková, Dominika, Vallianatou, Theodosia, Nilsson, Anna, Shariatgorji, Reza, Hammarlund-Udenaes, Margareta, Loryan, Irena, Andrén, Per E
Published in Molecular psychiatry (01.12.2021)
Published in Molecular psychiatry (01.12.2021)
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Journal Article
Rate and extent of mitragynine and 7‐hydroxymitragynine blood–brain barrier transport and their intra‐brain distribution: the missing link in pharmacodynamic studies
Yusof, Siti R., Mohd Uzid, Mahathir, Teh, Eng‐Huat, Hanapi, Nur Aziah, Mohideen, Mazlin, Mohamad Arshad, Ahmad Saifuddin, Mordi, Mohd Nizam, Loryan, Irena, Hammarlund‐Udenaes, Margareta
Published in Addiction biology (01.09.2019)
Published in Addiction biology (01.09.2019)
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Journal Article
Oxymorphone Active Uptake at the Blood–Brain Barrier and Population Modeling of its Pharmacokinetic–Pharmacodynamic Relationship
Sadiq, Muhammad Waqas, Boström, Emma, Keizer, Ron, Bjorkman, Sven, Hammarlund-Udenaes, Margareta
Published in Journal of pharmaceutical sciences (01.09.2013)
Published in Journal of pharmaceutical sciences (01.09.2013)
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Journal Article
Active‐Site Concentrations of Chemicals – Are They a Better Predictor of Effect than Plasma/Organ/Tissue Concentrations?
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Journal Article
Conference Proceeding
Pharmacokinetics of P‐glycoprotein inhibition in the rat blood‐brain barrier
Syvänen, Stina, Hooker, Andrew, Rahman, Obaidur, Wilking, Helena, Blomquist, Gunnar, Långström, Bengt, Bergström, Mats, Hammarlund‐Udenaes, Margareta
Published in Journal of pharmaceutical sciences (01.12.2008)
Published in Journal of pharmaceutical sciences (01.12.2008)
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Journal Article
On-line desalting and determination of morphine, morphine-3-glucuronide and morphine-6-glucuronide in microdialysis and plasma samples using column switching and liquid chromatography/tandem mass spectrometry
Bengtsson, Jörgen, Jansson, Britt, Hammarlund-Udenaes, Margareta
Published in Rapid communications in mass spectrometry (01.01.2005)
Published in Rapid communications in mass spectrometry (01.01.2005)
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Journal Article
On The Rate and Extent of Drug Delivery to the Brain
Hammarlund-Udenaes, Margareta, Fridén, Markus, Syvänen, Stina, Gupta, Anubha
Published in Pharmaceutical research (01.08.2008)
Published in Pharmaceutical research (01.08.2008)
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Journal Article
The role of P‐glycoprotein in blood‐brain barrier transport of morphine: transcortical microdialysis studies in mdr1a (−/−) and mdr1a (+/+) mice
Xie, Rujia, Hammarlund‐Udenaes, Margareta, De Boer, Albertus G, De Lange, Elizabeth C M
Published in British journal of pharmacology (01.10.1999)
Published in British journal of pharmacology (01.10.1999)
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Journal Article
Effects of pharmacists' interventions on appropriateness of prescribing and evaluation of the instruments' (MAI, STOPP and STARTs') ability to predict hospitalization--analyses from a randomized controlled trial
Gillespie, Ulrika, Alassaad, Anna, Hammarlund-Udenaes, Margareta, Mörlin, Claes, Henrohn, Dan, Bertilsson, Maria, Melhus, Håkan
Published in PloS one (17.05.2013)
Published in PloS one (17.05.2013)
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Journal Article
Structure−Brain Exposure Relationships in Rat and Human Using a Novel Data Set of Unbound Drug Concentrations in Brain Interstitial and Cerebrospinal Fluids
Fridén, Markus, Winiwarter, Susanne, Jerndal, Gunilla, Bengtsson, Ola, Wan, Hong, Bredberg, Ulf, Hammarlund-Udenaes, Margareta, Antonsson, Madeleine
Published in Journal of medicinal chemistry (22.10.2009)
Published in Journal of medicinal chemistry (22.10.2009)
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Journal Article
Species Differences in Blood-Brain Barrier Transport of Three Positron Emission Tomography Radioligands with Emphasis on P-Glycoprotein Transport
Syvänen, Stina, Lindhe, Orjan, Palner, Mikael, Kornum, Birgitte R, Rahman, Obaidur, Långström, Bengt, Knudsen, Gitte M, Hammarlund-Udenaes, Margareta
Published in Drug metabolism and disposition (01.03.2009)
Published in Drug metabolism and disposition (01.03.2009)
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Journal Article
Measurement of Unbound Drug Exposure in Brain: Modeling of pH Partitioning Explains Diverging Results between the Brain Slice and Brain Homogenate Methods
FRIDEN, Markus, BERGSTROM, Fredrik, HONG WAN, REHNGREN, Mikael, AHLIN, Gustav, HAMMARLUND-UDENAES, Margareta, BREDBERG, Ulf
Published in Drug metabolism and disposition (01.03.2011)
Published in Drug metabolism and disposition (01.03.2011)
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Journal Article
Improved measurement of drug exposure in the brain using drug-specific correction for residual blood
Fridén, Markus, Ljungqvist, Helena, Middleton, Brian, Bredberg, Ulf, Hammarlund-Udenaes, Margareta
Published in Journal of cerebral blood flow and metabolism (01.01.2010)
Published in Journal of cerebral blood flow and metabolism (01.01.2010)
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Journal Article
Mechanistic Study on the Use of the l‑Type Amino Acid Transporter 1 for Brain Intracellular Delivery of Ketoprofen via Prodrug: A Novel Approach Supporting the Development of Prodrugs for Intracellular Targets
Puris, Elena, Gynther, Mikko, de Lange, Elizabeth C.M, Auriola, Seppo, Hammarlund-Udenaes, Margareta, Huttunen, Kristiina M, Loryan, Irena
Published in Molecular pharmaceutics (01.07.2019)
Published in Molecular pharmaceutics (01.07.2019)
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Journal Article