Identification of the first synthetic inhibitors of the type II transmembrane serine protease TMPRSS2 suitable for inhibition of influenza virus activation
Meyer, Daniela, Sielaff, Frank, Hammami, Maya, Böttcher-Friebertshäuser, Eva, Garten, Wolfgang, Steinmetzer, Torsten
Published in Biochemical journal (01.06.2013)
Published in Biochemical journal (01.06.2013)
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Journal Article
Matriptase, HAT, and TMPRSS2 Activate the Hemagglutinin of H9N2 Influenza A Viruses
Baron, Joanna, Tarnow, Carolin, Mayoli-Nüssle, Deborah, Schilling, Eva, Meyer, Daniela, Hammami, Maya, Schwalm, Folker, Steinmetzer, Torsten, Guan, Yi, Garten, Wolfgang, Klenk, Hans-Dieter, Böttcher-Friebertshäuser, Eva
Published in Journal of Virology (01.02.2013)
Published in Journal of Virology (01.02.2013)
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Journal Article
Matriptase Induction of Metalloproteinase‐Dependent Aggrecanolysis In Vitro and In Vivo: Promotion of Osteoarthritic Cartilage Damage by Multiple Mechanisms
Wilkinson, David J., Habgood, Angela, Lamb, Heather K., Thompson, Paul, Hawkins, Alastair R., Désilets, Antoine, Leduc, Richard, Steinmetzer, Torsten, Hammami, Maya, Lee, Melody S., Craik, Charles S., Watson, Sharon, Lin, Hua, Milner, Jennifer M., Rowan, Andrew D.
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2017)
Published in Arthritis & rheumatology (Hoboken, N.J.) (01.08.2017)
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Journal Article
Changing the selectivity profile - from substrate analog inhibitors of thrombin and factor Xa to potent matriptase inhibitors
Maiwald, Alexander, Hammami, Maya, Wagner, Sebastian, Heine, Andreas, Klebe, Gerhard, Steinmetzer, Torsten
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
Published in Journal of enzyme inhibition and medicinal chemistry (01.11.2016)
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Journal Article
New 3-amidinophenylalanine-derived inhibitors of matriptase
Hammami, Maya, Rühmann, Eggert, Maurer, Eva, Heine, Andreas, Gütschow, Michael, Klebe, Gerhard, Steinmetzer, Torsten
Published in MedChemComm (01.07.2012)
Published in MedChemComm (01.07.2012)
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Journal Article
Cover Picture: Development and Characterization of New Peptidomimetic Inhibitors of the West Nile Virus NS2B-NS3 Protease (ChemMedChem 2/2013)
Hammamy, M. Zouhir, Haase, Caroline, Hammami, Maya, Hilgenfeld, Rolf, Steinmetzer, Torsten
Published in ChemMedChem (01.02.2013)
Published in ChemMedChem (01.02.2013)
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Journal Article
New 3-amidinophenylalanine-derived inhibitors of matriptaseElectronic supplementary information (ESI) available: Information regarding the used analytical methods, a table with the analytical data of all new inhibitors, and information regarding the performed enzyme kinetic measurements and the crystallographic data of thrombin in complex with inhibitor 11 (4e7r.pdb). See DOI: 10.1039/c2md20074k
Hammami, Maya, Rühmann, Eggert, Maurer, Eva, Heine, Andreas, Gütschow, Michael, Klebe, Gerhard, Steinmetzer, Torsten
Year of Publication 01.07.2012
Year of Publication 01.07.2012
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Journal Article
USE OF TMPRSS2 INHIBITORS AS MEDICAMENTS
HAMMAMI, MAYA, BÖTTCHER-FRIEBERTSHÄUSER, EVA, GARTEN, WOLFGANG, SIELAFF, FRANK, MEYER, DANIELA, STEINMETZER, TORSTEN
Year of Publication 04.06.2014
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Year of Publication 04.06.2014
Patent
USE OF TMPRSS2 INHIBITORS AS MEDICAMENTS
HAMMAMI, MAYA, GARTEN, WOLFGANG, SIELAFF, FRANK, MEYER, DANIELA, STEINMETZER, TORSTEN, BOETTCHER-FRIEBERTSHAEUSER, EVA
Year of Publication 31.01.2013
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Year of Publication 31.01.2013
Patent
Verwendung von Hemmstoffen der TMPRSS2 als Arzneimittel
FRIEBERTSHAEUSER, EVA, HAMMAMI, MAYA, GARTEN, WOLFGANG, STEINMETZER, TORSTEN, DR, SIELAFF, FRANK, MEYER, DANIELA
Year of Publication 31.01.2013
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Year of Publication 31.01.2013
Patent