Design of thiamine analogues for inhibition of thiamine diphosphate (ThDP)-dependent enzymes: Systematic investigation through Scaffold-Hopping and C2-Functionalisation
Chan, Alex H.Y., Ho, Terence C.S., Irfan, Rimsha, Hamid, Rawia A.A., Rudge, Emma S., Iqbal, Amjid, Turner, Alex, Hirsch, Anna K.H., Leeper, Finian J.
Published in Bioorganic chemistry (01.09.2023)
Published in Bioorganic chemistry (01.09.2023)
Get full text
Journal Article
1-deoxy-D-xylulose-5-phosphate synthase from Pseudomonas aeruginosa and Klebsiella pneumoniae reveals conformational changes upon cofactor binding
Hamid, Rawia, Adam, Sebastian, Lacour, Antoine, Monjas, Leticia, Köhnke, Jesko, Hirsch, Anna K.H.
Published in The Journal of biological chemistry (01.09.2023)
Published in The Journal of biological chemistry (01.09.2023)
Get full text
Journal Article
Not Every Hit‐Identification Technique Works on 1‐Deoxy‐d‐Xylulose 5‐Phosphate Synthase (DXPS): Making the Most of a Virtual Screening Campaign
Johannsen, Sandra, Gierse, Robin M., Olshanova, Aleksandra, Smerznak, Ellie, Laggner, Christian, Eschweiler, Lea, Adeli, Zahra, Hamid, Rawia, Alhayek, Alaa, Reiling, Norbert, Haupenthal, Jörg, Hirsch, Anna K. H.
Published in ChemMedChem (01.06.2023)
Published in ChemMedChem (01.06.2023)
Get full text
Journal Article
Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors
Ropponen, Henni‐Karoliina, Diamanti, Eleonora, Johannsen, Sandra, Illarionov, Boris, Hamid, Rawia, Jaki, Miriam, Sass, Peter, Fischer, Markus, Haupenthal, Jörg, Hirsch, Anna K. H.
Published in ChemMedChem (04.10.2023)
Published in ChemMedChem (04.10.2023)
Get full text
Journal Article
Front Cover: Exploring the Translational Gap of a Novel Class of Escherichia coli IspE Inhibitors (ChemMedChem 19/2023)
Ropponen, Henni‐Karoliina, Diamanti, Eleonora, Johannsen, Sandra, Illarionov, Boris, Hamid, Rawia, Jaki, Miriam, Sass, Peter, Fischer, Markus, Haupenthal, Jörg, Hirsch, Anna K. H.
Published in ChemMedChem (04.10.2023)
Published in ChemMedChem (04.10.2023)
Get full text
Journal Article
Evaluation of ketoclomazone and its analogues as inhibitors of 1-deoxy--xylulose 5-phosphate synthases and other thiamine diphosphate (ThDP)-dependent enzymes
Chan, Alex H. Y, Ho, Terence C. S, Fathoni, Imam, Hamid, Rawia, Hirsch, Anna K. H, Saliba, Kevin J, Leeper, Finian J
Published in RSC medicinal chemistry (22.05.2024)
Published in RSC medicinal chemistry (22.05.2024)
Get full text
Journal Article
Evaluation of ketoclomazone and its analogues as inhibitors of 1-deoxy-d-xylulose 5-phosphate synthases and other thiamine diphosphate (ThDP)-dependent enzymes
Chan, Alex H. Y., Ho, Terence C. S., Fathoni, Imam, Hamid, Rawia, Hirsch, Anna K. H., Saliba, Kevin J., Leeper, Finian J.
Published in MedChemComm (22.05.2024)
Published in MedChemComm (22.05.2024)
Get full text
Journal Article