TSPO Ligands Boost Mitochondrial Function and Pregnenolone Synthesis
Lejri, Imane, Grimm, Amandine, Hallé, François, Abarghaz, Mustapha, Klein, Christian, Maitre, Michel, Schmitt, Martine, Bourguignon, Jean-Jacques, Mensah-Nyagan, Ayikoe Guy, Bihel, Frederic, Eckert, Anne
Published in Journal of Alzheimer's disease (01.01.2019)
Published in Journal of Alzheimer's disease (01.01.2019)
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Human erythrocytes release ATP by a novel pathway involving VDAC oligomerization independent of pannexin-1
Marginedas-Freixa, Irene, Alvarez, Cora Lilia, Moras, Martina, Leal Denis, María Florencia, Hattab, Claude, Halle, François, Bihel, Frédéric, Mouro-Chanteloup, Isabelle, Lefevre, Sophie Denise, Le Van Kim, Caroline, Schwarzbaum, Pablo Julio, Ostuni, Mariano Anibal
Published in Scientific reports (30.07.2018)
Published in Scientific reports (30.07.2018)
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Pharmacomodulation of a ligand targeting the HBV capsid hydrophobic pocket
Briday, Mathilde, Hallé, François, Lecoq, Lauriane, Radix, Sylvie, Martin, Juliette, Montserret, Roland, Dujardin, Marie, Fogeron, Marie-Laure, Nassal, Michael, Meier, Beat H, Lomberget, Thierry, Böckmann, Anja
Published in Chemical science (Cambridge) (04.08.2022)
Published in Chemical science (Cambridge) (04.08.2022)
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The translocator protein ligand XBD173 improves clinical symptoms and neuropathological markers in the SJL/J mouse model of multiple sclerosis
Leva, Géraldine, Klein, Christian, Benyounes, Jérémie, Hallé, François, Bihel, Frédéric, Collongues, Nicolas, De Seze, Jérôme, Mensah-Nyagan, Ayikoe-Guy, Patte-Mensah, Christine
Published in Biochimica et biophysica acta. Molecular basis of disease (01.12.2017)
Published in Biochimica et biophysica acta. Molecular basis of disease (01.12.2017)
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χ‑Space Screening of Dermorphin-Based Tetrapeptides through Use of Constrained Arylazepinone and Quinolinone Scaffolds
Van der Poorten, Olivier, Van Den Hauwe, Robin, Eiselt, Emilie, Betti, Cecilia, Guillemyn, Karel, Chung, Nga N, Hallé, François, Bihel, Frédéric, Schiller, Peter W, Tourwé, Dirk, Sarret, Philippe, Gendron, Louis, Ballet, Steven
Published in ACS medicinal chemistry letters (09.11.2017)
Published in ACS medicinal chemistry letters (09.11.2017)
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Synthesis of 3-amino-3,4-dihydro-1H-quinolin-2-ones through regioselective palladium-catalyzed intramolecular cyclization
Hallé, François, Van der Poorten, Olivier, Doebelin, Christelle, Niederst, Marie, Schneider, Séverine, Schmitt, Martine, Ballet, Steven, Bihel, Frédéric
Published in Tetrahedron letters (06.04.2016)
Published in Tetrahedron letters (06.04.2016)
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Emissive Synthetic Cofactors: Enzymatic Interconversions of tzA Analogues of ATP, NAD+, NADH, NADP+, and NADPH
Hallé, François, Fin, Andrea, Rovira, Alexander R., Tor, Yitzhak
Published in Angewandte Chemie (22.01.2018)
Published in Angewandte Chemie (22.01.2018)
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Design, synthesis, and structure-activity relationship studies of 6 H -benzo[ b ]indeno[1,2- d ]thiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors
Faouzi, Abdelfattah, Arnaud, Alexandre, Hallé, François, Roussel, Jean, Aymard, Mandy, Denavit, Vincent, Do, Cong Viet, Mularoni, Angélique, Salah, Mohamed, ElHady, Ahmed, Pham, Thanh-Nhat, Bancet, Alexandre, Le Borgne, Marc, Terreux, Raphaël, Barret, Roland, Engel, Matthias, Lomberget, Thierry
Published in RSC medicinal chemistry (17.10.2024)
Published in RSC medicinal chemistry (17.10.2024)
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Journal Article
Design, synthesis, and structure-activity relationship studies of 6H-benzobindeno1,2-dthiophen-6-one derivatives as DYRK1A/CLK1/CLK4/haspin inhibitors
Faouzi, Abdelfattah, Arnaud, Alexandre, Hallé, François, Roussel, Jean, Aymard, Mandy, Denavit, Vincent, Do, Cong Viet, Mularoni, Angélique, Salah, Mohamed, ElHady, Ahmed, Pham, Thanh-Nhat, Bancet, Alexandre, Le Borgne, Marc, Terreux, Raphaël, Barret, Roland, Engel, Matthias, Lomberget, Thierry
Published in RSC medicinal chemistry (17.10.2024)
Published in RSC medicinal chemistry (17.10.2024)
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A Journey through Hemetsberger–Knittel, Leimgruber–Batcho and Bartoli Reactions: Access to Several Hydroxy 5‐ and 6‐Azaindoles
Radix, Sylvie, Hallé, François, Mahiout, Zahia, Teissonnière, Amélie, Bouchez, Grégoire, Auberger, Ludovic, Barret, Roland, Lomberget, Thierry
Published in Helvetica chimica acta (01.03.2022)
Published in Helvetica chimica acta (01.03.2022)
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Journal Article
Improved methods for mutacin detection and production
Nicolas, Guillaume, Auger, Isabelle, Beaudoin, Martine, Hallé, Francois, Morency, Hélène, LaPointe, Gisèle, Lavoie, Marc C.
Published in Journal of microbiological methods (01.12.2004)
Published in Journal of microbiological methods (01.12.2004)
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Crystal structure and identification of a pyrimido[6,1-b][1,3]oxazin-6-one derivative from the reaction of acrolein with 5-(phenoxymethyl)-2-amino-2-oxazoline
Guillon, Jean, Rubio, Sandra, Savrimoutou, Solène, Hallé, François, Moreau, Stéphane, Sonnet, Pascal, Marchivie, Mathieu
Published in Comptes rendus. Chimie (01.11.2018)
Published in Comptes rendus. Chimie (01.11.2018)
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New 6-Formyl-oxazolo[3,2-a]Pyrimidine Derivatives: Synthesis and Evaluation as Potential Src Kinase Inhibitors
Guillon, Jean, Halle, François, Savrimoutou, Solène, Moreau, Stéphane, Henri Caignard, Daniel, Sonnet, Pascal
Published in Acta Scientific Pharmaceutical Sciences (19.11.2019)
Published in Acta Scientific Pharmaceutical Sciences (19.11.2019)
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ChemInform Abstract: Synthesis of 3‐Amino‐3,4‐dihydro‐1H‐quinolin‐2‐ones Through Regioselective Palladium‐Catalyzed Intramolecular Cyclization
Halle, Francois, Van der Poorten, Olivier, Doebelin, Christelle, Niederst, Marie, Schneider, Severine, Schmitt, Martine, Ballet, Steven, Bihel, Frederic
Published in ChemInform (01.07.2016)
Published in ChemInform (01.07.2016)
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