Designing heterocyclic selective kinase inhibitors: from concept to new drug candidates
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Design and Synthesis of the First Generation of Novel Potent, Selective, and in Vivo Active (Benzothiazol-2-yl)acetonitrile Inhibitors of the c-Jun N-Terminal Kinase
Gaillard, Pascale, Jeanclaude-Etter, Isabelle, Ardissone, Vittoria, Arkinstall, Steve, Cambet, Yves, Camps, Montserrat, Chabert, Christian, Church, Dennis, Cirillo, Rocco, Gretener, Denise, Halazy, Serge, Nichols, Anthony, Szyndralewiez, Cedric, Vitte, Pierre-Alain, Gotteland, Jean-Pierre
Published in Journal of medicinal chemistry (14.07.2005)
Published in Journal of medicinal chemistry (14.07.2005)
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In vitro and in vivo pharmacological profile of AS057278, a selective d -amino acid oxidase inhibitor with potential anti-psychotic properties
Adage, Tiziana, Trillat, Anne-Cécile, Quattropani, Anna, Perrin, Dominique, Cavarec, Laurent, Shaw, Jeffrey, Guerassimenko, Oxana, Giachetti, Claudio, Gréco, Béatrice, Chumakov, Ilya, Halazy, Serge, Roach, Arthur, Zaratin, Paola
Published in European neuropsychopharmacology (01.03.2008)
Published in European neuropsychopharmacology (01.03.2008)
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(Aryloxy)methylsilane Derivatives as New Cholesterol Biosynthesis Inhibitors: Synthesis and Hypocholesterolemic Activity of a New Class of Squalene Epoxidase Inhibitors
Gotteland, Jean-Pierre, Brunel, Isabelle, Gendre, Fabrice, Desire, Jerome, Delhon, Andre, Junquero, Didier, Oms, Philippe, Halazy, Serge
Published in Journal of medicinal chemistry (01.08.1995)
Published in Journal of medicinal chemistry (01.08.1995)
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Synthesis and serotonergic activity of arylpiperazide derivatives of serotonin: potent agonists for 5-HT1D receptors
Perez, Michel, Fourrier, Catherine, Sigogneau, Isabelle, Pauwels, Petrus J, Palmier, Christiane, John, Gareth W, Valentin, Jean-Pierre, Halazy, Serge
Published in Journal of medicinal chemistry (01.09.1995)
Published in Journal of medicinal chemistry (01.09.1995)
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Studies on the synthesis of the antitumor agent CC-1065. Synthesis of PDE I and PDE II, inhibitors of cyclic adenosine-3',5'-monophosphate phosphodiesterase using the 3,3'-bipyrrole strategy
Carter, Paul, Fitzjohn, Steven, Halazy, Serge, Magnus, Philip
Published in Journal of the American Chemical Society (01.04.1987)
Published in Journal of the American Chemical Society (01.04.1987)
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3,6-Dibromocarbazole Piperazine Derivatives of 2-Propanol as First Inhibitors of Cytochrome c Release via Bax Channel Modulation
Bombrun, Agnes, Gerber, Patrick, Casi, Giulio, Terradillos, Olivier, Antonsson, Bruno, Halazy, Serge
Published in Journal of medicinal chemistry (09.10.2003)
Published in Journal of medicinal chemistry (09.10.2003)
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GLEPP1/Protein-tyrosine Phosphatase ϕ Inhibitors Block Chemotaxis in Vitro and in Vivo and Improve Murine Ulcerative Colitis
Gobert, Rosanna Pescini, van den Eijnden, Monique, Szyndralewiez, Cedric, Jorand-Lebrun, Catherine, Swinnen, Dominique, Chen, Linfeng, Gillieron, Corine, Pixley, Fiona, Juillard, Pierre, Gerber, Patrick, Johnson-Léger, Caroline, Halazy, Serge, Camps, Montserrat, Bombrun, Agnes, Shipp, Margaret, Vitte, Pierre-Alain, Ardissone, Vittoria, Ferrandi, Chiara, Perrin, Dominique, Rommel, Christian, van Huijsduijnen, Rob Hooft
Published in The Journal of biological chemistry (24.04.2009)
Published in The Journal of biological chemistry (24.04.2009)
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Design, Synthesis, and Biological Activity of Novel, Potent, and Selective (Benzoylaminomethyl)thiophene Sulfonamide Inhibitors of c-Jun-N-Terminal Kinase
Rückle, Thomas, Biamonte, Marco, Grippi-Vallotton, Tania, Arkinstall, Steve, Cambet, Yves, Camps, Montserrat, Chabert, Christian, Church, Dennis J, Halazy, Serge, Jiang, Xuliang, Martinou, Isabelle, Nichols, Anthony, Sauer, Wolfgang, Gotteland, Jean-Pierre
Published in Journal of medicinal chemistry (30.12.2004)
Published in Journal of medicinal chemistry (30.12.2004)
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GLEPP1/Protein-tyrosine Phosphatase φ Inhibitors Block Chemotaxis in Vitro and in Vivo and Improve Murine Ulcerative ColitisS
Gobert, Rosanna Pescini, van den Eijnden, Monique, Szyndralewiez, Cedric, Jorand-Lebrun, Catherine, Swinnen, Dominique, Chen, Linfeng, Gillieron, Corine, Pixley, Fiona, Juillard, Pierre, Gerber, Patrick, Johnson-Léger, Caroline, Halazy, Serge, Camps, Montserrat, Bombrun, Agnes, Shipp, Margaret, Vitte, Pierre-Alain, Ardissone, Vittoria, Ferrandi, Chiara, Perrin, Dominique, Rommel, Christian, van Huijsduijnen, Rob Hooft
Published in The Journal of biological chemistry (24.04.2009)
Published in The Journal of biological chemistry (24.04.2009)
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GLEPP1/Protein-tyrosine Phosphatase Ï Inhibitors Block Chemotaxis in Vitro and in Vivo and Improve Murine Ulcerative Colitis
Rosanna Pescini Gobert, Monique van den Eijnden, Cedric Szyndralewiez, Catherine Jorand-Lebrun, Dominique Swinnen, Linfeng Chen, Corine Gillieron, Fiona Pixley, Pierre Juillard, Patrick Gerber, Caroline Johnson-Léger, Serge Halazy, Montserrat Camps, Agnes Bombrun, Margaret Shipp, Pierre-Alain Vitte, Vittoria Ardissone, Chiara Ferrandi, Dominique Perrin, Christian Rommel, Rob Hooft van Huijsduijnen
Published in The Journal of biological chemistry (24.04.2009)
Published in The Journal of biological chemistry (24.04.2009)
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GLEPP1/Protein-tyrosine Phosphatase {phi} Inhibitors Block Chemotaxis in Vitro and in Vivo and Improve Murine Ulcerative Colitis
Gobert, Rosanna Pescini, van den Eijnden, Monique, Szyndralewiez, Cedric, Jorand-Lebrun, Catherine, Swinnen, Dominique, Chen, Linfeng, Gillieron, Corine, Pixley, Fiona, Juillard, Pierre, Gerber, Patrick, Johnson-Léger, Caroline, Halazy, Serge, Camps, Montserrat, Bombrun, Agnes, Shipp, Margaret, Vitte, Pierre-Alain, Ardissone, Vittoria, Ferrandi, Chiara, Perrin, Dominique, Rommel, Christian, van Huijsduijnen, Rob Hooft
Published in The Journal of biological chemistry (2009)
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Published in The Journal of biological chemistry (2009)
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