Synthesis of targeted dibenzo[b,f]thiepines and dibenzo[b,f]oxepines as potential lead molecules with promising anti-breast cancer activity
Ansari, Mohd. Imran, Hussain, Mohd. Kamil, Arun, Ashutosh, Chakravarti, Bandana, Konwar, Rituraj, Hajela, K.
Published in European journal of medicinal chemistry (24.06.2015)
Published in European journal of medicinal chemistry (24.06.2015)
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Silica supported perchloric acid catalyzed rapid N-formylation under solvent-free conditions
Ansari, Mohd. Imran, Hussain, Mohd. Kamil, Yadav, Nisha, Gupta, Puneet K., Hajela, K.
Published in Tetrahedron letters (18.04.2012)
Published in Tetrahedron letters (18.04.2012)
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New piperidine derivative DTPEP acts as dual‐acting anti‐breast cancer agent by targeting ERα and downregulating PI3K/Akt‐PKCα leading to caspase‐dependent apoptosis
Arun, A., Ansari, M.I., Popli, P., Jaiswal, S., Mishra, A.K., Dwivedi, A., Hajela, K., Konwar, R.
Published in Cell proliferation (01.12.2018)
Published in Cell proliferation (01.12.2018)
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Design and synthesis of ERα/ERβ selective coumarin and chromene derivatives as potential anti-breast cancer and anti-osteoporotic agents
Hussain, M. Kamil, Ansari, M. Imran, Yadav, N., Gupta, Puneet K., Gupta, A. K., Saxena, R., Fatima, I., Manohar, M., Kushwaha, P., Khedgikar, V., Gautam, J., Kant, Ruchir, Maulik, P. R., Trivedi, R., Dwivedi, A., Kumar, K. Ravi, Saxena, A. K., Hajela, K.
Published in RSC advances (2014)
Published in RSC advances (2014)
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Inhibitory effect of 2-(piperidinoethoxyphenyl)-3-(4-hydroxyphenyl)-2H-benzo(b)pyran (K-1) on human primary endometrial hyperplasial cells mediated via combined suppression of Wnt/β-catenin signaling and PI3K/Akt survival pathway
Chandra, V, Fatima, I, Manohar, M, Popli, P, Sirohi, V K, Hussain, M K, Hajela, K, Sankhwar, P, Dwivedi, A
Published in Cell death & disease (21.08.2014)
Published in Cell death & disease (21.08.2014)
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Exposure to an environmental neurotoxicant hastens the onset of amyotrophic lateral sclerosis-like phenotype in human Cu2+/Zn2+ superoxide dismutase 1 G93A mice: glutamate-mediated excitotoxicity
Johnson, Frank O, Yuan, Yukun, Hajela, Ravindra K, Chitrakar, Alisha, Parsell, Dawn M, Atchison, William D
Published in The Journal of pharmacology and experimental therapeutics (01.08.2011)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2011)
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The anti-proliferative effect of 2-[piperidinoethoxyphenyl]-3-[4-hydroxyphenyl]-2H-benzo(b) pyran is potentiated via induction of estrogen receptor beta and p21 in human endometrial adenocarcinoma cells
Fatima, I., Saxena, R., Kharkwal, G., Hussain, M.K., Yadav, N., Hajela, K., Sankhwar, P.L., Dwivedi, A.
Published in The Journal of steroid biochemistry and molecular biology (01.11.2013)
Published in The Journal of steroid biochemistry and molecular biology (01.11.2013)
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Synthesis and biological evaluation of indolyl bisphosphonates as anti-bone resorptive and anti-leishmanial agents
Singh, Uma Sharan, Shankar, Ravi, Kumar, Avinash, Trivedi, Ritu, Chattopadhyay, Naibedya, Shakya, Nishi, Palne, Shraddha, Gupta, Suman, Hajela, K.
Published in Bioorganic & medicinal chemistry (15.09.2008)
Published in Bioorganic & medicinal chemistry (15.09.2008)
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Synthesis and biological evaluation of 3,4,6-triaryl-2-pyranones as a potential new class of anti-breast cancer agents
Shankar, Ravi, Chakravarti, Bandana, Singh, Uma Sharan, Ansari, Mohd. Imran, Deshpande, Shreekant, Dwivedi, Shailendra Kumar Dhar, Bid, Hemant Kumar, Konwar, Rituraj, Kharkwal, Geetika, Chandra, Vishal, Dwivedi, Anila, Hajela, K.
Published in Bioorganic & medicinal chemistry (01.06.2009)
Published in Bioorganic & medicinal chemistry (01.06.2009)
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Anti-tumorigenic action of 2-[piperidinoethoxyphenyl]-3-[4-hydroxyphenyl]-2H-benzo(b)pyran: Evidence for involvement of GPR30/EGFR signaling pathway
Chandra, V, Fatima, I, Saxena, R, Hussain, M.K, Hajela, K, Sankhwar, P, Roy, B.G, Chandna, S, Dwivedi, A
Published in Gynecologic oncology (01.05.2013)
Published in Gynecologic oncology (01.05.2013)
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2,3-Diaryl-2H-1-benzopyran derivatives interfere with classical and non-classical estrogen receptor signaling pathways, inhibit Akt activation and induce apoptosis in human endometrial cancer cells
Fatima, I., Chandra, V., Saxena, R., Manohar, M., Sanghani, Y., Hajela, K., Negi, M.P.S., Sankhwar, P.L., Jain, S.K., Dwivedi, A.
Published in Molecular and cellular endocrinology (02.01.2012)
Published in Molecular and cellular endocrinology (02.01.2012)
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The Biological Functions of MBL-Associated Serine Proteases (MASPs)
Hajela, Krishnan, Kojima, Mayumi, Ambrus, Geza, Nicky Wong, K.H., Moffatt, Beryl E., Ferluga, Janez, Hajela, Sumati, Gál, Peter, Sim, Robert B.
Published in Immunobiology (1979) (01.09.2002)
Published in Immunobiology (1979) (01.09.2002)
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Leishmania donovani: Identification of stimulatory soluble antigenic proteins using cured human and hamster lymphocytes for their prophylactic potential against visceral leishmaniasis
Garg, Ravendra, Gupta, Shraddha K., Tripathi, Parul, Hajela, K., Sundar, S., Naik, S., Dube, Anuradha
Published in Vaccine (05.04.2006)
Published in Vaccine (05.04.2006)
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Synthesis and structure guided evaluation of estrogen agonist and antagonist activities of some new tetrazolyl indole derivatives
Singh, Uma Sharan, Shankar, Ravi, Yadav, Gaya P., Kharkwal, Geetika, Dwivedi, Anila, Keshri, Govind, Singh, M.M., Moulik, P.R., Hajela, K.
Published in European journal of medicinal chemistry (01.10.2008)
Published in European journal of medicinal chemistry (01.10.2008)
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Lack of genetic association of promoter and structural variants of mannan-binding lectin (MBL2) gene with susceptibility to generalized vitiligo
Dwivedi, M., Gupta, K., Gulla, K.C., Laddha, N.C., Hajela, K., Begum, R.
Published in British journal of dermatology (1951) (01.07.2009)
Published in British journal of dermatology (1951) (01.07.2009)
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Effects of Methylmercury on Human Neuronal L-Type Calcium Channels Transiently Expressed in Human Embryonic Kidney Cells (HEK-293)
Peng, Shuangqing, Hajela, Ravindra K, Atchison, William D
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2002)
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