Melanocortin receptor agonists, penile erection, and sexual motivation: human studies with Melanotan II
Wessells, H, Levine, N, Hadley, M E, Dorr, R, Hruby, V
Published in International journal of impotence research (01.10.2000)
Published in International journal of impotence research (01.10.2000)
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Discovery of Prototype Peptidomimetic Agonists at the Human Melanocortin Receptors MC1R and MC4R
Haskell-Luevano, Carrie, Hendrata, Siska, North, Cheryl, Sawyer, Tomi K, Hadley, Mac E, Hruby, Victor J, Dickinson, Chris, Gantz, Ira
Published in Journal of medicinal chemistry (04.07.1997)
Published in Journal of medicinal chemistry (04.07.1997)
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Characterizations of the Unusual Dissociation Properties of Melanotropin Peptides from the Melanocortin Receptor, hMC1R
Haskell-Luevano, Carrie, Miwa, Hiroto, Dickinson, Chris, Hadley, Mac E, Hruby, Victor J, Yamada, Tadataka, Gantz, Ira
Published in Journal of medicinal chemistry (19.01.1996)
Published in Journal of medicinal chemistry (19.01.1996)
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Topographical modification of melanotropin peptide analogs with .beta.-methyltryptophan isomers at position 9 leads to differential potencies and prolonged biological activities
Haskell-Luevano, Carrie, Boteju, Lakmal W, Miwa, Hiroto, Dickinson, Chris, Gantz, Ira, Yamada, Tadataka, Hadley, Mac E, Hruby, Victor J
Published in Journal of medicinal chemistry (01.11.1995)
Published in Journal of medicinal chemistry (01.11.1995)
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4 - Norleucine, 7-D-phenylalanine-α -melanocyte-stimulating Hormone: A Highly Potent α -melanotropin with Ultralong Biological Activity
Sawyer, Tomi K., Sanfilippo, Pauline J., Hruby, Victor J., Engel, Michael H., Heward, Christopher B., Burnett, Jean B., Hadley, Mac E.
Published in Proceedings of the National Academy of Sciences - PNAS (01.10.1980)
Published in Proceedings of the National Academy of Sciences - PNAS (01.10.1980)
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α-melanotropin: The minimal active sequence in the lizard skin bioassay
Castrucci, A.M.L., Hadley, M.E., Sawyer, T.K., Wilkes, B.C., Al-Obeidi, F., Staples, D.J., de Vaux, A.E., Dym, O., Hintz, M.F., Riehm, J.P., Rao, K.R., Hruby, V.J.
Published in General and comparative endocrinology (1989)
Published in General and comparative endocrinology (1989)
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The Proopiomelanocortin System
HADLEY, MAC E., HASKELL-LUEVANO, CARRIE
Published in Annals of the New York Academy of Sciences (01.10.1999)
Published in Annals of the New York Academy of Sciences (01.10.1999)
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alpha.-Melanotropin: the minimal active sequence in the frog skin bioassay
Hruby, Victor J, Wilkes, Brian C, Hadley, Mac E, Al-Obeidi, Fahad, Sawyer, Tomi K, Staples, Douglas J, DeVaux, Ann E, Dym, Orin, Castrucci, Ana Maria de L
Published in Journal of medicinal chemistry (01.11.1987)
Published in Journal of medicinal chemistry (01.11.1987)
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Synthetic melanotropic peptide initiates erections in men with psychogenic erectile dysfunction: double-blind, placebo controlled crossover study
Wessells, H, Fuciarelli, K, Hansen, J, Hadley, M E, Hruby, V J, Dorr, R, Levine, N
Published in The Journal of urology (01.08.1998)
Published in The Journal of urology (01.08.1998)
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Effect of an alpha-melanocyte stimulating hormone analog on penile erection and sexual desire in men with organic erectile dysfunction
WESSELLS, Hunter, GRALNEK, D. A. N, DORR, Robert, HRUBY, Victor J, HADLEY, Mac. E, LEVINE, Norman
Published in Urology (Ridgewood, N.J.) (01.10.2000)
Published in Urology (Ridgewood, N.J.) (01.10.2000)
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New Mustard Prodrugs for Antibody-Directed Enzyme Prodrug Therapy: Alternatives to the Amide Link
Dowell, Robert I, Springer, Caroline J, Davies, David H, Hadley, Elizabeth M, Burke, Philip J, Boyle, F. Thomas, Melton, Roger G, Connors, Thomas A, Blakey, David C, Mauger, Anthony B
Published in Journal of medicinal chemistry (01.03.1996)
Published in Journal of medicinal chemistry (01.03.1996)
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[half-Cys4,half-Cys10]-α -Melanocyte-Stimulating Hormone: A Cyclic α -melanotropin Exhibiting Superagonist Biological Activity
Sawyer, Tomi K., Hruby, Victor J., Darman, Paul S., Hadley, Mac E.
Published in Proceedings of the National Academy of Sciences - PNAS (01.03.1982)
Published in Proceedings of the National Academy of Sciences - PNAS (01.03.1982)
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Skin Pigmentation and Pharmacokinetics of Melanotan-I in Humans
UGWU, SYDNEY O., BLANCHARD, JAMES, DORR, ROBERT T., LEVINE, NORMAN, BROOKS, CHRISTINE, HADLEY, MAC E., AICKIN, MIKEL, HRUBY, VICTOR J.
Published in Biopharmaceutics & drug disposition (01.04.1997)
Published in Biopharmaceutics & drug disposition (01.04.1997)
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