Searching for New Leads for Tuberculosis: Design, Synthesis, and Biological Evaluation of Novel 2‑Quinolin-4-yloxyacetamides
Pitta, Eleni, Rogacki, Maciej K, Balabon, Olga, Huss, Sophie, Cunningham, Fraser, Lopez-Roman, Eva Maria, Joossens, Jurgen, Augustyns, Koen, Ballell, Lluis, Bates, Robert H, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.07.2016)
Published in Journal of medicinal chemistry (28.07.2016)
Get full text
Journal Article
Optimization of Hydantoins as Potent Antimycobacterial Decaprenylphosphoryl-β‑d‑Ribose Oxidase (DprE1) Inhibitors
Balabon, Olga, Pitta, Eleni, Rogacki, Maciej K, Meiler, Eugenia, Casanueva, Ruth, Guijarro, Laura, Huss, Sophie, Lopez-Roman, Eva Maria, Santos-Villarejo, Ángel, Augustyns, Koen, Ballell, Lluis, Aguirre, David Barros, Bates, Robert H, Cunningham, Fraser, Cacho, Monica, Van der Veken, Pieter
Published in Journal of medicinal chemistry (28.05.2020)
Published in Journal of medicinal chemistry (28.05.2020)
Get full text
Journal Article
Identification and Profiling of HydantoinsA Novel Class of Potent Antimycobacterial DprE1 Inhibitors
Rogacki, Maciej K, Pitta, Eleni, Balabon, Olga, Huss, Sophie, Lopez-Roman, Eva Maria, Argyrou, Argyrides, Blanco-Ruano, Delia, Cacho, Monica, Vande Velde, Christophe M. L, Augustyns, Koen, Ballell, Lluis, Barros, David, Bates, Robert H, Cunningham, Fraser, Van der Veken, Pieter
Published in Journal of medicinal chemistry (27.12.2018)
Published in Journal of medicinal chemistry (27.12.2018)
Get full text
Journal Article
Fueling Open-Source Drug Discovery: 177 Small-Molecule Leads against Tuberculosis
Ballell, Lluís, Bates, Robert H., Young, Rob J., Alvarez-Gomez, Daniel, Alvarez-Ruiz, Emilio, Barroso, Vanessa, Blanco, Delia, Crespo, Benigno, Escribano, Jaime, González, Rubén, Lozano, Sonia, Huss, Sophie, Santos-Villarejo, Angel, Martín-Plaza, José Julio, Mendoza, Alfonso, Rebollo-Lopez, María José, Remuiñan-Blanco, Modesto, Lavandera, José Luis, Pérez-Herran, Esther, Gamo-Benito, Francisco Javier, García-Bustos, José Francisco, Barros, David, Castro, Julia P., Cammack, Nicholas
Published in ChemMedChem (01.02.2013)
Published in ChemMedChem (01.02.2013)
Get full text
Journal Article
Stereospecific Synthesis and NMR Conformational Studies of .gamma.-Butyrolactones of Nucleosides as Chiral Synthons for the Preparation of 2'-C- and 3'-C-Branched-Chain Nucleosides
Velazquez, Sonsoles, Jimeno, Maria Luisa, Huss, Sophie, Balzarini, Jan, Camarasa, Maria-Jose
Published in Journal of organic chemistry (01.12.1994)
Published in Journal of organic chemistry (01.12.1994)
Get full text
Journal Article
Antitubercular drugs for an old target: GSK693 as a promising InhA direct inhibitor
Martínez-Hoyos, María, Perez-Herran, Esther, Gulten, Gulcin, Encinas, Lourdes, Álvarez-Gómez, Daniel, Alvarez, Emilio, Ferrer-Bazaga, Santiago, García-Pérez, Adolfo, Ortega, Fátima, Angulo-Barturen, Iñigo, Rullas-Trincado, Joaquin, Blanco Ruano, Delia, Torres, Pedro, Castañeda, Pablo, Huss, Sophie, Fernández Menéndez, Raquel, González del Valle, Silvia, Ballell, Lluis, Barros, David, Modha, Sundip, Dhar, Neeraj, Signorino-Gelo, François, McKinney, John D., García-Bustos, Jose Francisco, Lavandera, Jose Luis, Sacchettini, James C., Jimenez, M. Soledad, Martín-Casabona, Nuria, Castro-Pichel, Julia, Mendoza-Losana, Alfonso
Published in EBioMedicine (01.06.2016)
Published in EBioMedicine (01.06.2016)
Get full text
Journal Article
Antifungal sordarins. Part 4: synthesis and structure–activity relationships of 3′,4′-fused alkyl-tetrahydrofuran derivatives
Bueno, José M, Chicharro, Jesús, Fiandor, José M, Gómez de las Heras, Federico, Huss, Sophie
Published in Bioorganic & medicinal chemistry letters (08.07.2002)
Published in Bioorganic & medicinal chemistry letters (08.07.2002)
Get full text
Journal Article