Role of the autotaxin-lysophosphatidic acid axis in glaucoma, aqueous humor drainage and fibrogenic activity
Ho, Leona T.Y., Osterwald, Anja, Ruf, Iris, Hunziker, Daniel, Mattei, Patrizio, Challa, Pratap, Vann, Robin, Ullmer, Christoph, Rao, Ponugoti Vasanth
Published in Biochimica et biophysica acta. Molecular basis of disease (01.01.2020)
Published in Biochimica et biophysica acta. Molecular basis of disease (01.01.2020)
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Synthesis, Characterization, and in vivo Evaluation of a Novel Potent Autotaxin-Inhibitor
Hunziker, Daniel, Reinehr, Sabrina, Palmhof, Marina, Wagner, Natalie, Biniasch, Thomas, Stute, Gesa, Mattei, Patrizio, Schmitz, Petra, DiGiorgio, Patrick, Hert, Jérôme, Rudolph, Markus G, Benz, Joerg, Stihle, Martine, Gsell, Bernard, Müller, Stephan, Gasser, Rodolfo, Schonhoven, Nina, Ullmer, Christoph, Joachim, Stephanie C
Published in Frontiers in pharmacology (18.01.2022)
Published in Frontiers in pharmacology (18.01.2022)
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Journal Article
Challenges and Rewards in Medicinal Chemistry Targeting Cardiovascular and Metabolic Diseases
Neidhart, Werner, Ackermann, Jean, Amrein, Kurt, Conte, Aurelia, Hunziker, Daniel, Kuhn, Bernd, Märki, Hans Peter, Nettekoven, Matthias, Ruf, Armin, Schulz-Gasch, Tanja, Mayweg, Alexander V
Published in Chimia (01.01.2015)
Published in Chimia (01.01.2015)
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Inhibitors of dipeptidyl peptidase IV--recent advances and structural views
Hunziker, Daniel, Hennig, Michael, Peters, Jens-Uwe
Published in Current topics in medicinal chemistry (01.12.2005)
Published in Current topics in medicinal chemistry (01.12.2005)
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Precursor directed biosynthesis of novel 6-deoxyerythronolide B analogs containing non-natural oxygen substituents and reactive functionalities
Hunziker, Daniel, Wu, Nicholas, Kenoshita, Kenji, Cane, David E., Khosla, Chaitan
Published in Tetrahedron letters (01.01.1999)
Published in Tetrahedron letters (01.01.1999)
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Preclinical Characterization of a Next-Generation Brain Permeable, Paradox Breaker BRAF Inhibitor
Wichmann, Jürgen, Rynn, Caroline, Friess, Thomas, Petrig-Schaffland, Jeannine, Kornacker, Martin, Handl, Cornelia, Emmenegger, Jasmin, Eckmann, Jan, Herting, Frank, Frances, Nicolas, Hunziker, Daniel, Krummenacher, Daniela, Rüttinger, Dominik, Ribeiro, Alison, Bacac, Marina, Brigo, Alessandro, Hewings, David S, Dummer, Reinhard, Levesque, Mitchell P, Schnetzler, Gabriel, Martoglio, Bruno, Bischoff, James R, Pettazzoni, Piergiorgio
Published in Clinical cancer research (15.02.2022)
Published in Clinical cancer research (15.02.2022)
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Enhancing Drug Discovery and Development through the Integration of Medicinal Chemistry, Chemical Biology, and Academia-Industry Partnerships: Insights from Roche's Endocannabinoid System Projects
Aebi, Johannes, Atz, Kenneth, Ametamey, Simon M, Benz, Jörg, Blaising, Julie, Butini, Stefania, Campiani, Giuseppe, Carreira, Erick M, Collin, Ludovic, De Lago, Eva, Gazzi, Thais, Gertsch, Jürg, Gobbi, Luca, Guba, Wolfgang, Fernández-Ruiz, Javier, Fingerle, Jürgen, Haider, Ahmed, He, Yingfang, Heitman, Laura H, Honer, Michael, Hunziker, Daniel, Kuhn, Bernd, Maccarrone, Mauro, Märki, Hans Peter, Martin, Rainer E, Mohr, Peter, Mu, Linjing, Nazaré, Marc, Nippa, David F, Oddi, Sergio, O'Hara, Fionn, Pacher, Pal, Romero, Julian, Röver, Stephan, Rufer, Arne C, Schibli, Roger, Schneider, Gisbert, Stepan, Antonia F, Sykes, David A, Ullmer, Christoph, Van der Stelt, Mario, Veprintsev, Dmitry B, Wittwer, Matthias B, Grether, Uwe
Published in Chimia (21.08.2024)
Published in Chimia (21.08.2024)
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Journal Article
패러독스 파괴제로서의 새로운 BRAF 억제제
PETTAZZONI PIERGIORGIO FRANCESCO TOMMASO, KRUMMENACHER DANIELA, HUNZIKER DANIEL, DOLENTE COSIMO, HEWINGS DAVID STEPHEN, WICHMANN JUERGEN
Year of Publication 11.08.2022
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Year of Publication 11.08.2022
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신규 메틸퀴나졸리논 유도체
PETTAZZONI PIERGIORGIO FRANCESCO TOMMASO, KRUMMENACHER DANIELA, HUNZIKER DANIEL, DOLENTE COSIMO, HEWINGS DAVID STEPHEN, WICHMANN JUERGEN
Year of Publication 08.08.2022
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Year of Publication 08.08.2022
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Identification of an antimalarial synthetic trioxolane drug development candidate
Vennerstrom, Jonathan L, Arbe-Barnes, Sarah, Brun, Reto, Charman, Susan A, Chiu, Francis C. K, Chollet, Jacques, Dong, Yuxiang, Dorn, Arnulf, Hunziker, Daniel, Matile, Hugues, McIntosh, Kylie, Padmanilayam, Maniyan, Santo Tomas, Josefina, Scheurer, Christian, Scorneaux, Bernard, Tang, Yuanqing, Urwyler, Heinrich, Wittlin, Sergio, Charman, William N
Published in Nature (19.08.2004)
Published in Nature (19.08.2004)
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돌연변이 BRAF의 분해를 위한 요법
JACKSON KATRINA L, VEITS GESINE KERSTIN, PETTAZZONI PIERGIORGIO FRANCESO TOMMASO, FITZGERALD MARK E, HEWING DAVID STEPHEN, HUNZIKER DANIEL, DOLENTE COSIMO, GARZA VICTORIA, WICHMANN JUERGEN, YU ROBERT T, DUPLESSIS MARTIN, O'SHEA MORGAN WELZEL, NASVESCHUK CHRISTOPHER G, KRUMMENACHER DANIELA, LIANG YANKE, GOOD ANDREW CHARLES
Year of Publication 13.02.2024
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Year of Publication 13.02.2024
Patent
Cytochrome P450-Mediated Metabolism and CYP Inhibition for the Synthetic Peroxide Antimalarial OZ439
Shackleford, David M, Chiu, Francis C. K, Katneni, Kasiram, Blundell, Scott, McLaren, Jenna, Wang, Xiaofang, Zhou, Lin, Sriraghavan, Kamaraj, Alker, André M, Hunziker, Daniel, Scheurer, Christian, Zhao, Qingjie, Dong, Yuxiang, Möhrle, Jörg J, Abla, Nada, Matile, Hugues, Wittlin, Sergio, Vennerstrom, Jonathan L, Charman, Susan A
Published in ACS infectious diseases (09.07.2021)
Published in ACS infectious diseases (09.07.2021)
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Journal Article
BRAF 분해제
JACKSON KATRINA L, PETTAZZONI PIERGIORGIO FRANCESCO TOMMASO, VEITS GESINE KERSTIN, MOUSTAKIM MOSES, FITZGERALD MARK E, KUHN BERND, HUNZIKER DANIEL, DOLENTE COSIMO, GARZA VICTORIA, HEWINGS DAVID STEPHEN, WICHMANN JUERGEN, DUPLESSIS MARTIN, O'SHEA MORGAN WELZEL, YU ROBERT T, NASVESCHUK CHRISTOPHER G, RIEMER CLAUS, YAP JEREMY L, RICKLIN FABIENNE, LIANG YANKE, GOOD ANDREW CHARLES
Year of Publication 23.03.2023
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Year of Publication 23.03.2023
Patent
Aryl- and heteroaryl-substituted aminobenzo[ a]quinolizines as dipeptidyl peptidase IV inhibitors
Boehringer, Markus, Fischer, Holger, Hennig, Michael, Hunziker, Daniel, Huwyler, Joerg, Kuhn, Bernd, Loeffler, Bernd M., Luebbers, Thomas, Mattei, Patrizio, Narquizian, Robert, Sebokova, Elena, Sprecher, Urs, Wessel, Hans Peter
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
Published in Bioorganic & medicinal chemistry letters (01.02.2010)
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이중 오토탁신(ATX)/탄산 무수화효소(CA) 억제제로서 유용한 헤테로환형 화합물
RUDOLPH MARKUS, SCHMITZ PETRA, MATTEI PATRIZIO, HUNZIKER DANIEL, DI GIORGIO PATRICK, HERT JEROME, GOMME JUSTIN
Year of Publication 20.11.2019
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Year of Publication 20.11.2019
Patent