INCB054828 (pemigatinib), a potent and selective inhibitor of fibroblast growth factor receptors 1, 2, and 3, displays activity against genetically defined tumor models
Liu, Phillip C C, Koblish, Holly, Wu, Liangxing, Bowman, Kevin, Diamond, Sharon, DiMatteo, Darlise, Zhang, Yue, Hansbury, Michael, Rupar, Mark, Wen, Xiaoming, Collier, Paul, Feldman, Patricia, Klabe, Ronald, Burke, Krista A, Soloviev, Maxim, Gardiner, Christine, He, Xin, Volgina, Alla, Covington, Maryanne, Ruggeri, Bruce, Wynn, Richard, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Yao, Wenqing, Huber, Reid, Hollis, Gregory
Published in PloS one (21.04.2020)
Published in PloS one (21.04.2020)
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Journal Article
CCR2 modulates inflammatory and metabolic effects of high-fat feeding
Weisberg, Stuart P, Hunter, Deborah, Huber, Reid, Lemieux, Jacob, Slaymaker, Sarah, Vaddi, Kris, Charo, Israel, Leibel, Rudolph L, Ferrante, Jr, Anthony W
Published in The Journal of clinical investigation (01.01.2006)
Published in The Journal of clinical investigation (01.01.2006)
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Journal Article
Preclinical characterization of INCB053914, a novel pan-PIM kinase inhibitor, alone and in combination with anticancer agents, in models of hematologic malignancies
Koblish, Holly, Li, Yun-Long, Shin, Niu, Hall, Leslie, Wang, Qian, Wang, Kathy, Covington, Maryanne, Marando, Cindy, Bowman, Kevin, Boer, Jason, Burke, Krista, Wynn, Richard, Margulis, Alex, Reuther, Gary W, Lambert, Que T, Dostalik Roman, Valerie, Zhang, Ke, Feng, Hao, Xue, Chu-Biao, Diamond, Sharon, Hollis, Greg, Yeleswaram, Swamy, Yao, Wenqing, Huber, Reid, Vaddi, Kris, Scherle, Peggy
Published in PloS one (21.06.2018)
Published in PloS one (21.06.2018)
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Journal Article
Abstract 3819: INCAGN02385 is an antagonist antibody targeting the co-inhibitory receptor LAG-3 for the treatment of human malignancies
Savitsky, David, Ward, Rebecca, Riordan, Christina, Mundt, Cornelia, Jennings, Shawn, Connolly, Joe, Findeis, Mark, Sanicola, Michele, Underwood, Dennis, Nastri, Horacio, Scherle, Peggy, Hollis, Gregory, Huber, Reid, Stein, Robert, Dijk, Marc van, Wilson, Nicholas S.
Published in Cancer research (Chicago, Ill.) (01.07.2018)
Published in Cancer research (Chicago, Ill.) (01.07.2018)
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Journal Article
Discovery and Pharmacological Characterization of a Novel Rodent-Active CCR2 Antagonist, INCB3344
Brodmerkel, Carrie M, Huber, Reid, Covington, Maryanne, Diamond, Sharon, Hall, Leslie, Collins, Robert, Leffet, Lynn, Gallagher, Karen, Feldman, Patricia, Collier, Paul, Stow, Mark, Gu, Xiaomei, Baribaud, Frederic, Shin, Niu, Thomas, Beth, Burn, Tim, Hollis, Greg, Yeleswaram, Swamy, Solomon, Kim, Friedman, Steve, Wang, Anlai, Xue, Chu Biao, Newton, Robert C, Scherle, Peggy, Vaddi, Kris
Published in The Journal of immunology (1950) (15.10.2005)
Published in The Journal of immunology (1950) (15.10.2005)
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Journal Article
Identification of ADAM10 as a major source of HER2 ectodomain sheddase activity in HER2 overexpressing breast cancer cells
Liu, Phillip C.C., Liu, Xiangdong, Li, Yanlong, Covington, Maryanne, Wynn, Richard, Huber, Reid, Hillman, Milton, Yang, Gengjie, Ellis, Dawn, Marando, Cindy, Katiyar, Kamna, Bradley, Jodi, Abremski, Kenneth, Stow, Mark, Rupar, Mark, Zhuo, Jincong, Li, Yun-Long, Lin, Qiyan, Burns, David, Xu, Meizhong, Zhang, Colin, Qian, Ding-Quan, He, Chunhong, Sharief, Vaqar, Weng, Lingkai, Agrios, Costas, Shi, Eric, Metcalf, Brian, Newton, Robert, Friedman, Steven, Yao, Wenqing, Scherle, Peggy A., Hollis, Gregory, Burn, Timothy C.
Published in Cancer biology & therapy (01.06.2006)
Published in Cancer biology & therapy (01.06.2006)
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Journal Article
Generation of multiple farnesoid-X-receptor isoforms through the use of alternative promoters
Huber, Reid M, Murphy, Kathleen, Miao, Bowman, Link, John R, Cunningham, Mark R, Rupar, Mark J, Gunyuzlu, Paul L, Haws, Thomas F, Kassam, Altaf, Powell, Francoise, Hollis, Gregory F, Young, Peter R, Mukherjee, Ranjan, Burn, Timothy C
Published in Gene (15.05.2002)
Published in Gene (15.05.2002)
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Journal Article
Mutations in GPC3 , a glypican gene, cause the Simpson-Golabi-Behmel overgrowth syndrome
Pilia, Giuseppe, Hughes-Benzie, Rhiannon M, MacKenzie, Alex, Baybayan, Primo, Chen, Ellson Y, Huber, Reid, Neri, Giovanni, Cao, Antonio, Forabosco, Antonino, Schlessinger, David
Published in Nature genetics (01.03.1996)
Published in Nature genetics (01.03.1996)
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Journal Article
Dexamethasone and Tumor Necrosis Factor-α Act Together to Induce the Cellular Inhibitor of Apoptosis-2 Gene and Prevent Apoptosis in a Variety of Cell Types
Webster, Jeffrey C, Huber, Reid M, Hanson, Rebecca L, Collier, Paul M, Haws, Thomas F, Mills, Juliane K, Burn, Timothy C, Allegretto, Elizabeth A
Published in Endocrinology (Philadelphia) (01.10.2002)
Published in Endocrinology (Philadelphia) (01.10.2002)
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Journal Article
Absence of Post-translational Aspartyl β-Hydroxylation of Epidermal Growth Factor Domains in Mice Leads to Developmental Defects and an Increased Incidence of Intestinal Neoplasia
Dinchuk, Joseph E., Focht, Richard J., Kelley, Jennifer A., Henderson, Nancy L., Zolotarjova, Nina I., Wynn, Richard, Neff, Nicola T., Link, John, Huber, Reid M., Burn, Timothy C., Rupar, Mark J., Cunningham, Mark R., Selling, Bernard H., Ma, Jianhong, Stern, Andrew A., Hollis, Gregory F., Stein, Robert B., Friedman, Paul A.
Published in The Journal of biological chemistry (12.04.2002)
Published in The Journal of biological chemistry (12.04.2002)
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Journal Article
The effect of long-term ruxolitinib treatment on JAK2p.V617F allele burden in patients with myelofibrosis
Deininger, Michael, Radich, Jerald, Burn, Timothy C., Huber, Reid, Paranagama, Dilan, Verstovsek, Srdan
Published in Blood (24.09.2015)
Published in Blood (24.09.2015)
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Journal Article
PLAC1, a trophoblast-specific gene, is expressed throughout pregnancy in the human placenta and modulated by keratinocyte growth factor
Fant, Michael, Weisoly, David L., Cocchia, Massimo, Huber, Reid, Khan, Shaista, Lunt, Tiffany, Schlessinger, David
Published in Molecular reproduction and development (01.12.2002)
Published in Molecular reproduction and development (01.12.2002)
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Journal Article
Current themes in microarray experimental design and analysis
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Journal Article
Conference Proceeding
Discovery of Pemigatinib: A Potent and Selective Fibroblast Growth Factor Receptor (FGFR) Inhibitor
Wu, Liangxing, Zhang, Colin, He, Chunhong, Qian, Dingquan, Lu, Liang, Sun, Yaping, Xu, Meizhong, Zhuo, Jincong, Liu, Phillip C. C, Klabe, Ronald, Wynn, Richard, Covington, Maryanne, Gallagher, Karen, Leffet, Lynn, Bowman, Kevin, Diamond, Sharon, Koblish, Holly, Zhang, Yue, Soloviev, Maxim, Hollis, Gregory, Burn, Timothy C, Scherle, Peggy, Yeleswaram, Swamy, Huber, Reid, Yao, Wenqing
Published in Journal of medicinal chemistry (12.08.2021)
Published in Journal of medicinal chemistry (12.08.2021)
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Journal Article
DNA Methylation in Transcriptional Repression of Two Differentially Expressed X-Linked Genes, GPC3 and SYBL1
Huber, Reid, Hansen, R. Scott, Strazzullo, Maria, Pengue, Gina, Mazzarella, Richard, D'Urso, Michele, Schlessinger, David, Pilia, Giuseppe, Gartler, Stanley M., D'Esposito, Maurizio
Published in Proceedings of the National Academy of Sciences - PNAS (19.01.1999)
Published in Proceedings of the National Academy of Sciences - PNAS (19.01.1999)
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Journal Article
Characterization of INCB086550: A Potent and Novel Small-Molecule PD-L1 Inhibitor
Koblish, Holly K, Wu, Liangxing, Wang, Liang-Chuan S, Liu, Phillip C C, Wynn, Richard, Rios-Doria, Jonathan, Spitz, Susan, Liu, Hao, Volgina, Alla, Zolotarjova, Nina, Kapilashrami, Kanishk, Behshad, Elham, Covington, Maryanne, Yang, Yan-Ou, Li, Jingwei, Diamond, Sharon, Soloviev, Maxim, O'Hayer, Kevin, Rubin, Stephen, Kanellopoulou, Chrysi, Yang, Gengjie, Rupar, Mark, DiMatteo, Darlise, Lin, Luping, Stevens, Christina, Zhang, Yue, Thekkat, Pramod, Geschwindt, Ryan, Marando, Cindy, Yeleswaram, Swamy, Jackson, Jeff, Scherle, Peggy, Huber, Reid, Yao, Wenqing, Hollis, Gregory
Published in Cancer discovery (02.06.2022)
Published in Cancer discovery (02.06.2022)
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Journal Article
11-β-Hydroxysteroid Dehydrogenase Type 1 Inhibitor INCB13739 Improves Hyperglycemia in Patients With Type 2 Diabetes Inadequately Controlled by Metformin Monotherapy
Rosenstock, Julio, Banarer, Salomon, Fonseca, Vivian A, Inzucchi, Silvio E, Sun, William, Yao, Wenqing, Hollis, Gregory, Flores, Robert, Levy, Richard, Williams, William V, Seckl, Jonathan R, Huber, Reid
Published in Diabetes care (01.07.2010)
Published in Diabetes care (01.07.2010)
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Journal Article
Ruxolitinib, a JAK1/JAK2 Selective Inhibitor Is Highly Efficacious in Corticosteroid Untreated and Refractory MHC-Mismatched Mouse Model of Acute GvHD
Juvekar, Ashish, Ruggeri, Bruce, Condon, Sindy, Borkowski, Andrew, Huber, Reid, Smith, Paul
Published in Blood (29.11.2018)
Published in Blood (29.11.2018)
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Journal Article
Itacitinib, a JAK1 Selective Inhibitor Preserves Graft-Versus-Leukemia (GVL), Enhances Survival and Is Highly Efficacious in a MHC-Mismatched Mouse Model of Acute GvHD
Juvekar, Ashish, Ruggeri, Bruce, Condon, Sindy, Borkowski, Andrew, Huber, Reid, Smith, Paul
Published in Blood (29.11.2018)
Published in Blood (29.11.2018)
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Journal Article