Initial SAR studies on apamin-displacing 2-aminothiazole blockers of calcium-activated small conductance potassium channels
Gentles, Robert G., Grant-Young, Katherine, Hu, Shuanghua, Huang, Yazhong, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine KCa channel blockers
GENTLES, Robert G, SHUANGHUA HU, HARDEN, David G, YAZHONG HUANG, GRANT-YOUNG, Katherine, POSS, Michael A, ANDRES, Charles, FIEDLER, Tracey, KNOX, Ronald, LODGE, Nicholas, WEAVER, C. David
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Identification of a Potent and Selective 5-HT6 Antagonist: One-Step Synthesis of (E)-3-(Benzenesulfonyl)-2- (methylsulfanyl)pyrido[1,2-a]pyrimidin- 4-ylidenamine from 2-(Benzenesulfonyl)-3,3- bis(methylsulfanyl)acrylonitrile
Wu, Yong-Jin, He, Huan, Hu, Shuanghua, Huang, Yazhong, Scola, Paul M, Grant-Young, Katharine, Bertekap, Robert L, Wu, Dedong, Gao, Qi, Li, Yi, Klakouski, Cheryl, Westphal, Ryan S
Published in Journal of medicinal chemistry (06.11.2003)
Published in Journal of medicinal chemistry (06.11.2003)
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Novel Dihydropyrazine Analogues as NPY Antagonists
Sit, Sing-Yuen, Huang, Yazhong, Antal-Zimanyi, Ildiko, Ward, Sally, Poindexter, Graham S
Published in Bioorganic & medicinal chemistry letters (11.02.2002)
Published in Bioorganic & medicinal chemistry letters (11.02.2002)
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Journal Article
Discovery of D1 Dopamine Receptor Positive Allosteric Modulators: Characterization of Pharmacology and Identification of Residues that Regulate Species Selectivity
Lewis, Martin A, Hunihan, Lisa, Watson, John, Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Bronson, Joanne, Macor, John E, Beno, Brett R, Ferrante, Meredith, Hendricson, Adam, Knox, Ronald J, Molski, Thaddeus F, Kong, Yan, Cvijic, Mary Ellen, Rockwell, Kristin L, Weed, Michael R, Cacace, Angela M, Westphal, Ryan S, Alt, Andrew, Brown, Jeffrey M
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
Published in The Journal of pharmacology and experimental therapeutics (01.09.2015)
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Structure activity relationship studies on chemically non-reactive glycine sulfonamide inhibitors of diacylglycerol lipase
Chupak, Louis S., Zheng, Xiaofan, Hu, Shuanghua, Huang, Yazhong, Ding, Min, Lewis, Martin A., Westphal, Ryan S., Blat, Yuval, McClure, Andrea, Gentles, Robert G.
Published in Bioorganic & medicinal chemistry (01.04.2016)
Published in Bioorganic & medicinal chemistry (01.04.2016)
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Structure activity relationship studies of 3-arylsulfonyl-pyrido[1,2-a]pyrimidin-4-imines as potent 5-HT6 antagonists
Hu, Shuanghua, Huang, Yazhong, Wu, Yong-Jin, He, Huan, Grant-Young, Katherine A., Bertekap, Robert L., Whiterock, Valerie, Brassil, Patrick, Lentz, Kimberley, Sivaprakasam, Prasanna, Langley, David R., Westphal, Ryan S., Scola, Paul M.
Published in Bioorganic & medicinal chemistry (01.03.2014)
Published in Bioorganic & medicinal chemistry (01.03.2014)
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T 세포 활성화제로서 유용한 나프티리디논 화합물
DING MIN, CHUPAK LOUIS S, MARTIN SCOTT W, MERCER STEPHEN E, MCDONALD IVAR M, ZHENG XIAOFAN, GENTLES ROBERT G, OLSON RICHARD E, HUANG YAZHONG, VELAPARTHI UPENDER, WICHROSKI MICHAEL
Year of Publication 05.03.2021
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Year of Publication 05.03.2021
Patent
DGK 억제제 및 체크포인트 길항제의 조합물
DING MIN, TOKARSKI JOHN S, ROY SAUMYA, KAMBLE MANJUNATHA NARAYANA RAO, VELAPARTHI UPENDER, GRUNENFELDER DENISE, ZHENG XIAOFAN, RAJA THIRUVENKADAM, JALAGAM PRASADA RAO, BENCI JOSEPH L, OLSON RICHARD E, CHUPAK LOUIS S, REDDY KOTHA RATHNAKAR, WEE SUSAN, DARNE CHETAN P, WANG XINYU, TONUKUNURU GOPIKISHAN, WARRIER JAYAKUMAR SANKARA, MARTIN SCOTT W, WICHROSKI MICHAEL J, MCDONALD IVAR M, DASGUPTA BIRESHWAR, MANNOORI RAJU, RAHAMAN HASIBUR, VELAIAH SIVASUDAR, GENTLES ROBERT G, HUANG YAZHONG
Year of Publication 25.08.2022
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Year of Publication 25.08.2022
Patent
T 세포 활성화제로서 유용한 치환된 나프티리디논 화합물
DING MIN, CHUPAK LOUIS S, TOKARSKI JOHN S, REDDY KOTHA RATHNAKAR, ROY SAUMYA, TONUKUNURU GOPIKISHAN, KAMBLE MANJUNATHA NARAYANA RAO, VELAPARTHI UPENDER, WARRIER JAYAKUMAR SANKARA, DARNE CHETAN PADMAKAR, MARTIN SCOTT W, MCDONALD IVAR M, ZHENG XIAOFAN, DASGUPTA BIRESHWAR, MANNOORI RAJU, RAJA THIRUVENKADAM, JALAGAM PRASADA RAO, RAHAMAN HASIBUR, VELAIAH SIVASUDAR, GENTLES ROBERT G, OLSON RICHARD E, HUANG YAZHONG
Year of Publication 05.03.2021
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Year of Publication 05.03.2021
Patent
Heterocyclic modification of a novel bicyclo[3.1.0]hexane NPY1 receptor antagonist
Luo, Guanglin, Chen, Ling, Hu, Shuanghua, Huang, Yazhong, Mattson, Gail, Iben, Lawrence G., Russell, John W., Clarke, Wendy J., Hogan, John B., Antal-Zimanyi, Ildiko, Poindexter, Graham S.
Published in Bioorganic & medicinal chemistry letters (01.07.2013)
Published in Bioorganic & medicinal chemistry letters (01.07.2013)
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Journal Article
Preliminary SAR studies on non-apamin-displacing 4-(aminomethylaryl)pyrrazolopyrimidine K Ca channel blockers
Gentles, Robert G., Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A., Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, C. David, Harden, David G.
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
Published in Bioorganic & medicinal chemistry letters (15.10.2008)
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Journal Article
Preliminary SAR studies on non-apamin-displacing 4- (aminomethylaryl)pyrrazolopyrimidine K sub(Ca) channel blockers
Gentles, Robert G, Hu, Shuanghua, Huang, Yazhong, Grant-Young, Katherine, Poss, Michael A, Andres, Charles, Fiedler, Tracey, Knox, Ronald, Lodge, Nicholas, Weaver, CDavid, Harden, David G
Published in Bioorganic & medicinal chemistry (01.10.2008)
Published in Bioorganic & medicinal chemistry (01.10.2008)
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Journal Article
Discovery of a Novel Class of Bicyclo[3.1.0]hexanylpiperazines as Noncompetitive Neuropeptide Y Y1 Antagonists
Hu, Shuanghua, Huang, Yazhong, Deshpande, Milind, Luo, Guanglin, Bruce, Marc A, Chen, Ling, Mattson, Gail, Iben, Lawrence G, Zhang, Jie, Russell, John W, Clarke, Wendy J, Hogan, John B, Ortiz, Astrid, Flint, Oliver, Henwood, Andrew, Gao, Qi, Antal-Zimanyi, Ildiko, Poindexter, Graham S
Published in ACS medicinal chemistry letters (08.03.2012)
Published in ACS medicinal chemistry letters (08.03.2012)
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