Discovery of the Selective CYP17A1 Lyase Inhibitor BMS-351 for the Treatment of Prostate Cancer
Huang, Audris, Jayaraman, Lata, Fura, Aberra, Vite, Gregory D, Trainor, George L, Gottardis, Marco M, Spires, Thomas E, Spires, Vanessa M, Rizzo, Cheryl A, Obermeier, Mary T, Elzinga, Paul A, Todderud, Gordon, Fan, Yi, Newitt, John A, Beyer, Sophie M, Zhu, Yongxin, Warrack, Bethanne M, Goodenough, Angela K, Tebben, Andrew J, Doweyko, Arthur M, Gold, David L, Balog, Aaron
Published in ACS medicinal chemistry letters (14.01.2016)
Published in ACS medicinal chemistry letters (14.01.2016)
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Journal Article
Broad-Spectrum Antiherpes Activities of 4-Hydroxyquinoline Carboxamides, a Novel Class of Herpesvirus Polymerase Inhibitors
OIEN, Nancee L, BRIDEAU, Roger J, VAILLANCOURT, Vallerie A, CLAYTON, Terrance L, TUCKER, John A, WATHEN, Michael W, HOPKINS, Todd A, WIEBER, Janet L, KNECHTEL, Mary L, SHELLY, John A, ANSTADT, Robert A, WELLS, Peter A, POORMAN, Roger A, HUANG, Audris
Published in Antimicrobial Agents and Chemotherapy (01.03.2002)
Published in Antimicrobial Agents and Chemotherapy (01.03.2002)
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Journal Article
Broad-spectrum antiviral activity of PNU-183792, a 4-oxo-dihydroquinoline, against human and animal herpesviruses
Brideau, Roger J., Knechtel, Mary L., Huang, Audris, Vaillancourt, Valerie A., Vera, Ellen E., Oien, Nancee L., Hopkins, Todd A., Wieber, Janet L., Wilkinson, Karen F., Rush, Bob D., Schwende, Francis J., Wathen, Michael W.
Published in Antiviral research (01.04.2002)
Published in Antiviral research (01.04.2002)
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Journal Article
The discovery of BMS-737 as a potent, CYP17 lyase-selective inhibitor for the treatment of castration-resistant prostate cancer
Padmakar Darne, Chetan, Velaparthi, Upender, Saulnier, Mark, Frennesson, David, Liu, Peiying, Huang, Audris, Tokarski, John, Fura, Aberra, Spires, Thomas, Newitt, John, Spires, Vanessa M., Obermeier, Mary T., Elzinga, Paul A., Gottardis, Marco M., Jayaraman, Lata, Vite, Gregory D., Balog, Aaron
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
Published in Bioorganic & medicinal chemistry letters (01.11.2022)
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Journal Article
Total Synthesis of (−)-Lasonolide A
Trost, Barry M, Stivala, Craig E, Fandrick, Daniel R, Hull, Kami L, Huang, Audris, Poock, Caroline, Kalkofen, Rainer
Published in Journal of the American Chemical Society (14.09.2016)
Published in Journal of the American Chemical Society (14.09.2016)
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Journal Article
A Concise Synthesis of (−)-Lasonolide A
Trost, Barry M, Stivala, Craig E, Hull, Kami L, Huang, Audris, Fandrick, Daniel R
Published in Journal of the American Chemical Society (08.01.2014)
Published in Journal of the American Chemical Society (08.01.2014)
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Journal Article
Radiochemistry challenges and progression for incorporation of 18F into a complex substituted 6-18F-fluoroquinoline BMS-986205 for IDO imaging
Cole, Erin, Donnelly, David, Wallace, Michael, Tran, Tritin, Burrell, Richard, Turley, Wesley, Allentoff, Alban, Huang, Audris, Balog, Aaron, Bonacorsi, Samuel
Published in The Journal of nuclear medicine (1978) (01.05.2018)
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Published in The Journal of nuclear medicine (1978) (01.05.2018)
Journal Article
Radiochemistry challenges and progression for incorporation of ^sup 18^F into a complex substituted 6-^sup 18^F-fluoroquinoline BMS-986205 for IDO imaging
Cole, Erin, Donnelly, David, Wallace, Michael, Tran, Tritin, Burrell, Richard, Turley, Wesley, Allentoff, Alban, Huang, Audris, Balog, Aaron, Bonacorsi, Samuel
Published in The Journal of nuclear medicine (1978) (01.05.2018)
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Published in The Journal of nuclear medicine (1978) (01.05.2018)
Journal Article
Long-Acting Tumor-Activated Prodrug of a TGFβR Inhibitor
Zhang, Yong, Parrish, Karen E, Tortolani, David R, Poss, Michael A, Huang, Audris, Wan, Honghe, Purandare, Ashok V, Donnell, Andrew F, Kempson, James, Hou, Xiaoping, Pawluczyk, Joseph, Yip, Shiuhang, Luk, Emily, Raghavan, Nimmi, Swanson, Jesse, Smalley, James, Murtaza, Anwar, Yang, Zheng, Augustine-Rauch, Karen, Lombardo, Louis J, Borzilleri, Robert
Published in Journal of medicinal chemistry (11.11.2021)
Published in Journal of medicinal chemistry (11.11.2021)
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Journal Article
피리디닐 치환된 옥소이소인돌린 화합물
PENMETSA SURESH BABU VISHWA KRISHNA, CHEN YAN, BALOG JAMES AARON, HUANG AUDRIS, KUMI GODWIN KWAME, NAIR SATHEESH KESAVAN, SHIMPUKADE BHARAT DINKAR
Year of Publication 05.12.2023
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Year of Publication 05.12.2023
Patent
헬리오스 단백질의 억제제로서 유용한 화합물
PURANDARE ASHOK VINAYAK, DEGNAN ANDREW P, SHAN WEIFANG, GUO LI, BALOG JAMES AARON, HUANG AUDRIS, KUMI GODWIN KWAME
Year of Publication 22.07.2022
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Year of Publication 22.07.2022
Patent
암의 치료를 위한 치환된 옥소이소인돌린 화합물
DEGNAN ANDREW P, PARK PETER KINAM, HUANG AUDRIS, KUMI GODWIN KWAME, PURANDARE ASHOK V, BILDER DONNA M, CHERNEY EMILY, TEBBEN ANDREW J
Year of Publication 30.11.2022
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Year of Publication 30.11.2022
Patent
Conformational-Analysis-Guided Discovery of 2,3-Disubstituted Pyridine IDO1 Inhibitors
Cherney, Emily C, Zhang, Liping, Guo, Weiwei, Huang, Audris, Williams, David, Seitz, Steven, Shan, Weifang, Zhu, Xiao, Gullo-Brown, Johnni, Maley, Derrick, Lin, Tai-an, Hunt, John T, Huang, Christine, Yang, Zheng, D’Arienzo, Celia J, Discenza, Lorell N, Ranasinghe, Asoka, Grubb, Mary F, Traeger, Sarah C, Li, Xin, Johnston, Kathy A, Kopcho, Lisa, Fereshteh, Mark, Foster, Kimberly A, Stefanski, Kevin, Delpy, Diane, Dhar, Gopal, Anandam, Aravind, Mahankali, Sandeep, Padmanabhan, Shweta, Rajanna, Prabhakar, Murali, Venkata, Mariappan, T. Thanga, Pattasseri, Shabeerali, Nimje, Roshan Y, Hong, Zhenqiu, Kempson, James, Rampulla, Richard, Mathur, Arvind, Gupta, Anuradha, Borzilleri, Robert, Vite, Gregory, Balog, Aaron
Published in ACS medicinal chemistry letters (08.07.2021)
Published in ACS medicinal chemistry letters (08.07.2021)
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Journal Article
인돌아민 2,3-디옥시게나제의 억제제 및 그의 사용 방법
SHAN WEIFANG, BALOG JAMES AARON, NARA SUSHEEL JETHANAND, HUANG AUDRIS, CHERNEY EMILY CHARLOTTE, ZHANG LIPING
Year of Publication 18.04.2019
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Year of Publication 18.04.2019
Patent
인돌아민 2,3-디옥시게나제의 억제제 및 그의 사용 방법
SHAN WEIFANG, GUO WEIWEI, BALOG JAMES AARON, HUANG AUDRIS, CHERNEY EMILY CHARLOTTE, ZHANG LIPING, WILLIAMS DAVID K
Year of Publication 09.01.2019
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Year of Publication 09.01.2019
Patent
IDO1 효소를 영상화하기 위한 방사성리간드
BALOG JAMES AARON, BURRELL RICHARD CHARLES, DONNELLY DAVID J, HUANG AUDRIS, TURLEY WESLEY A, ALLENTOFF ALBAN J, SKINBJERG METTE, WALLACE MICHAEL ARTHUR, COLE ERIN LEE
Year of Publication 22.03.2019
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Year of Publication 22.03.2019
Patent
암의 치료를 위한 인돌아민-2,3-디옥시게나제의 억제제
SHAN WEIFANG, GUO WEIWEI, BALOG JAMES AARON, MARKWALDER JAY A, ROY SAUMYA, HUANG AUDRIS, NARA SUSHEEL JETHANAND, WILLIAMS DAVID K
Year of Publication 07.12.2017
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Year of Publication 07.12.2017
Patent