Discovery of Aryl Aminoquinazoline Pyridones as Potent, Selective, and Orally Efficacious Inhibitors of Receptor Tyrosine Kinase c-Kit
Hu, Essa, Tasker, Andrew, White, Ryan D, Kunz, Roxanne K, Human, Jason, Chen, Ning, Bürli, Roland, Hungate, Randall, Novak, Perry, Itano, Andrea, Zhang, Xuxia, Yu, Violeta, Nguyen, Yen, Tudor, Yanyan, Plant, Matthew, Flynn, Shaun, Xu, Yang, Meagher, Kristin L, Whittington, Douglas A, Ng, Gordon Y
Published in Journal of medicinal chemistry (12.06.2008)
Published in Journal of medicinal chemistry (12.06.2008)
Get full text
Journal Article
Allosteric inhibitors of Aktl and Akt2 : Discovery of [1,2,4]triazolo[3,4-f][1,6]naphthyridines with potent and balanced activity
YIWEI LI, JUN LIANG, HUBER, Hans E, MITTAL, Sachin, COSFORD, Nicholas, PRASIT, Peppi, SIU, Tony, HU, Essa, ROSSI, Michael A, BARNETT, Stanley F, DEFEO-JONES, Deborah, JONES, Raymond E, ROBINSON, Ronald G, LEANDER, Karen
Published in Bioorganic & medicinal chemistry letters (2009)
Get full text
Published in Bioorganic & medicinal chemistry letters (2009)
Journal Article
PEPTIDE PAC1 ANTAGONISTS
CHEN, IRWIN, LONG, JASON C, CHONG, SU, HARRINGTON, ESSA HU, MIRANDA, LESLIE P, HONG, FANG-TSAO
Year of Publication 06.12.2018
Get full text
Year of Publication 06.12.2018
Patent
Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors
HARRINGTON ESSA HU, RZASA ROBERT M, MONENSCHEIN HOLGER, REICHELT ANDREAS, ALLEN JENNIFER R, NGUYEN THOMAS T, HORNE DANIEL B, KALLER MATTHEW R
Year of Publication 28.06.2016
Get full text
Year of Publication 28.06.2016
Patent
UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS
HARRINGTON ESSA HU, CHEN JIAN J, LIU QINGYIAN, RUMFELT SHANNON, FROHN MICHAEL J, ZHONG WENGE, RZASA ROBERT M, PICKRELL ALEXANDER J, ALLEN JENNIFER R
Year of Publication 14.04.2016
Get full text
Year of Publication 14.04.2016
Patent
ANTAGONISTAS DE PÉPTIDO PAC1
CHEN, IRWIN, LONG, JASON, MIRANDA, LESLIE, CHONG, SU, HONG, FANG, TSAO - HARRINGTON, ESSA HU
Year of Publication 21.08.2019
Get full text
Year of Publication 21.08.2019
Patent
PYRAZINE COMPOUNDS AS PHOSPHODIESTERASE 10 INHIBITORS
JENNIFER R. ALLEN, ESSA HU, MATTHEW P. BOURBEAU, SHANNON RUMFELT, ROXANNE KUNZ, NING CHEN
Year of Publication 08.01.2013
Get full text
Year of Publication 08.01.2013
Patent
Nitrogen heterocyclic compounds useful as pde10 inhibitors
HARRINGTON ESSA HU, CHEN JIAN J, LIU QINGYIAN, RUMFELT SHANNON, ZHONG WENGE, FROHN MICHAEL J, RZASA ROBERT M, PICKRELL ALEXANDER J, ALLEN JENNIFER R
Year of Publication 27.02.2015
Get full text
Year of Publication 27.02.2015
Patent
Peptide PAC1 antagonists
CHEN, IRWIN, LONG, JASON C, CHONG, SU, HARRINGTON, ESSA HU, MIRANDA, LESLIE P, HONG, FANG-TSAO
Year of Publication 01.06.2019
Get full text
Year of Publication 01.06.2019
Patent
Heterobicyclic compounds
AMEGADZIE ALBERT, YUAN CHESTER CHENGUANG, ALLEN JENNIFER R, ANDREWS KRISTIN L, HARRINGTON ESSA HU, CHEN JIAN J, QIAN WENYUAN, LIU QINGYIAN, RUMFELT SHANNON, ZHONG WENGE, BROWN JAMES, CHEN NING, RZASA ROBERT M, PICKRELL ALEXANDER J, NGUYEN THOMAS T
Year of Publication 03.11.2015
Get full text
Year of Publication 03.11.2015
Patent
UNSATURATED NITROGEN HETEROCYCLIC COMPOUNDS USEFUL AS PDE10 INHIBITORS
HARRINGTON ESSA HU, CHEN JIAN J, LIU QINGYIAN, RUMFELT SHANNON, FROHN MICHAEL J, ZHONG WENGE, RZASA ROBERT M, PICKRELL ALEXANDER J, ALLEN JENNIFER R
Year of Publication 31.07.2014
Get full text
Year of Publication 31.07.2014
Patent
HETEROARYLOXYCARBOCYCLYL COMPOUNDS AS PDE10 INHIBITORS
SHAM, KELVIN, PICKRELL, ALEXANDER, RZASA, ROBERT, FROHN, MICHAEL, HARRINGTON, PAUL, HARRINGTON, ESSA HU, ALLEN, JENNIFER
Year of Publication 20.03.2013
Get full text
Year of Publication 20.03.2013
Patent
Heteroaryloxyheterocyclyl compounds as PDE10 inhibitors
MONENSCHEIN, HOLGER, HARRINGTON, ESSA HU, ALLEN, JENNIFER, HORNE, DANIEL B, REICHELT, ANDREAS, RZASA, ROBERT M, NGUYEN, THOMAS T, KALLER, MATTHEW R
Year of Publication 01.05.2014
Get full text
Year of Publication 01.05.2014
Patent
Amides as pim inhibitors
CEE VICTOR, WU BIN, TASKER ANDREW, SMITH ADRIAN L, WURZ RYAN, TAMAYO NURIA A, HARRINGTON ESSA HU, HERBERICH BRADLEY, CHEN JIAN J, LANMAN BRIAN A, CHAVEZ, JR. FRANK, PETTUS LIPING H, JACKSON CLAIRE L. M, NORMAN MARK H, NGUYEN THOMAS T, REED ANTHONY B, WANG HUI-LING
Year of Publication 19.07.2016
Get full text
Year of Publication 19.07.2016
Patent
HETEROBICYCLIC COMPOUNDS AND THEIR USE AS PHOSPHODIESTERASE INHIBITORS
ZHONG, WENGE, RUMFELT, SHANNON, CHEN, NING, LIU, QINGYIAN, ALLEN, JENNIFER R, QIAN, WENYUAN, RZASA, ROBERT M, ANDREWS, KRISTIN L, NGUYEN, THOMAS T, YUAN, CHESTER CHENGUANG, CHEN, JIAN J, BROWN, JAMES, HARRINGTON, ESSA HU, AMEGADZIE, ALBERT, PICKRELL, ALEXANDER J
Year of Publication 07.01.2015
Get full text
Year of Publication 07.01.2015
Patent