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Published in Drug metabolism and disposition (01.12.2004)
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Published in Journal of medicinal chemistry (09.09.2010)
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Published in Journal of medicinal chemistry (21.09.2006)
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Yam, Alice, Hanson, Jeff, Bajjuri, Krishna, Zhou, Sihong, Moreira, Dayson, Smith, Jennifer, Abrahams, Cristina, Li, Xiaofan, Lee, Grace, Armstrong, Stephanie, Gakhal, Amandeep, Calarese, Daniel, Park, Young, Miao Wen, Yin, Gang, Chivers, Simon, Hsieh, Faye, Xu, Guifen, Rubas, Werner, Maderna, Andreas, Bedard, Kristin, Hallam, Trevor
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A Novel Biotransformation of Alkyl Aminopyrrolidine to Aminopiperidine Ring by Human CYP3A
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Published in Drug metabolism and disposition (01.09.2011)
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Simultaneous determination of a p38 MAP kinase inhibitor and its amide hydrolyzed metabolite in Cynomolgus monkey plasma by LC–MS/MS, and its application to a toxicokinetic study
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Published in Journal of pharmaceutical and biomedical analysis (15.07.2011)
Published in Journal of pharmaceutical and biomedical analysis (15.07.2011)
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Structure-Based Design of Novel 2-Amino-6-phenyl-pyrimido[5′,4′:5,6]pyrimido[1,2-a]benzimidazol-5(6H)-ones as Potent and Orally Active Inhibitors of Lymphocyte Specific Kinase (Lck): Synthesis, SAR, and In Vivo Anti-Inflammatory Activity
Martin, Matthew W, Newcomb, John, Nunes, Joseph J, Boucher, Christina, Chai, Lilly, Epstein, Linda F, Faust, Theodore, Flores, Sylvia, Gallant, Paul, Gore, Anu, Gu, Yan, Hsieh, Faye, Huang, Xin, Kim, Joseph L, Middleton, Scot, Morgenstern, Kurt, Oliveira-dos-Santos, Antonio, Patel, Vinod F, Powers, David, Rose, Paul, Tudor, Yanyan, Turci, Susan M, Welcher, Andrew A, Zack, Debra, Zhao, Huilin, Zhu, Li, Zhu, Xiaotian, Ghiron, Chiara, Ermann, Monika, Johnston, David, Saluste, Carl-Gustaf Pierre
Published in Journal of medicinal chemistry (27.03.2008)
Published in Journal of medicinal chemistry (27.03.2008)
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Abstract 711: Small molecule compounds that target cell division cycle 7 (Cdc7) kinase inhibit cell proliferation and tumor growth
Bailis, Julie, Fang, Li, Orf, Jessica, Heller, Scott, Bush, Tammy, Bourbeau, Matthew, Escobar, Sonia, Frohn, Michael, Harrington, Paul, Hsieh, Faye, Pickrell, Alexander, Sham, Kelvin, Siegmund, Aaron, Tan, Helming, Zalameda, Leeanne, Allen, John, Wickramasinghe, Dineli
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Published in Cancer research (Chicago, Ill.) (15.04.2013)
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Oxopyrido[2,3‑d]pyrimidines as Covalent L858R/T790M Mutant Selective Epidermal Growth Factor Receptor (EGFR) Inhibitors
Wurz, Ryan P, Pettus, Liping H, Ashton, Kate, Brown, James, Chen, Jian Jeffrey, Herberich, Brad, Hong, Fang-Tsao, Hu-Harrington, Essa, Nguyen, Tom, St. Jean, David J, Tadesse, Seifu, Bauer, David, Kubryk, Michele, Zhan, Jinghui, Cooke, Keegan, Mitchell, Petia, Andrews, Kristin L, Hsieh, Faye, Hickman, Dean, Kalyanaraman, Nataraj, Wu, Tian, Reid, Darren L, Lobenhofer, Edward K, Andrews, Dina A, Everds, Nancy, Guzman, Roberto, Parsons, Andrew T, Hedley, Simon J, Tedrow, Jason, Thiel, Oliver R, Potter, Matthew, Radinsky, Robert, Beltran, Pedro J, Tasker, Andrew S
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Published in ACS medicinal chemistry letters (10.09.2015)
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Wurz, Ryan P., Pettus, Liping H., Henkle, Bradley, Sherman, Lisa, Plant, Matthew, Miner, Kent, McBride, Helen J., Wong, Lu Min, Saris, Christiaan J.M., Lee, Matthew R., Chmait, Samer, Mohr, Christopher, Hsieh, Faye, Tasker, Andrew S.
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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3-Amino-7-phthalazinylbenzoisoxazoles as a Novel Class of Potent, Selective, and Orally Available Inhibitors of p38α Mitogen-Activated Protein Kinase
Pettus, Liping H, Xu, Shimin, Cao, Guo-Qiang, Chakrabarti, Partha P, Rzasa, Robert M, Sham, Kelvin, Wurz, Ryan P, Zhang, Dawei, Middleton, Scott, Henkle, Bradley, Plant, Matthew H, Saris, Christiaan J. M, Sherman, Lisa, Wong, Lu Min, Powers, David A, Tudor, Yanyan, Yu, Violeta, Lee, Matthew R, Syed, Rashid, Hsieh, Faye, Tasker, Andrew S
Published in Journal of medicinal chemistry (23.10.2008)
Published in Journal of medicinal chemistry (23.10.2008)
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Novel 2-Aminopyrimidine Carbamates as Potent and Orally Active Inhibitors of Lck: Synthesis, SAR, and in Vivo Antiinflammatory Activity
Martin, Matthew W, Newcomb, John, Nunes, Joseph J, McGowan, David C, Armistead, David M, Boucher, Christina, Buchanan, John L, Buckner, William, Chai, Lilly, Elbaum, Daniel, Epstein, Linda F, Faust, Theodore, Flynn, Shaun, Gallant, Paul, Gore, Anu, Gu, Yan, Hsieh, Faye, Huang, Xin, Lee, Josie H, Metz, Daniela, Middleton, Scot, Mohn, Deanna, Morgenstern, Kurt, Morrison, Michael J, Novak, Perry M, Oliveira-dos-Santos, Antonio, Powers, David, Rose, Paul, Schneider, Stephen, Sell, Stephanie, Tudor, Yanyan, Turci, Susan M, Welcher, Andrew A, White, Ryan D, Zack, Debra, Zhao, Huilin, Zhu, Li, Zhu, Xiaotian, Ghiron, Chiara, Amouzegh, Patricia, Ermann, Monika, Jenkins, James, Johnston, David, Napier, Spencer, Power, Eoin
Published in Journal of medicinal chemistry (10.08.2006)
Published in Journal of medicinal chemistry (10.08.2006)
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Discovery of 4-amino-5,6-biaryl-furo[2,3- d]pyrimidines as inhibitors of Lck: Development of an expedient and divergent synthetic route and preliminary SAR
DiMauro, Erin F., Newcomb, John, Nunes, Joseph J., Bemis, Jean E., Boucher, Christina, Buchanan, John L., Buckner, William H., Cheng, Alan, Faust, Theodore, Hsieh, Faye, Huang, Xin, Lee, Josie H., Marshall, Teresa L., Martin, Matthew W., McGowan, David C., Schneider, Stephen, Turci, Susan M., White, Ryan D., Zhu, Xiaotian
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
Published in Bioorganic & medicinal chemistry letters (15.04.2007)
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Part 1: Structure–Activity Relationship (SAR) investigations of fused pyrazoles as potent, selective and orally available inhibitors of p38α mitogen-activated protein kinase
Wurz, Ryan P., Pettus, Liping H., Xu, Shimin, Henkle, Bradley, Sherman, Lisa, Plant, Matthew, Miner, Kent, McBride, Helen, Wong, Lu Min, Saris, Christiaan J.M., Lee, Matthew R., Chmait, Samer, Mohr, Christopher, Hsieh, Faye, Tasker, Andrew S.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Identification of triazolopyridazinones as potent p38α inhibitors
Herberich, Brad, Jackson, Claire, Wurz, Ryan P., Pettus, Liping H., Sherman, Lisa, Liu, Qiurong, Henkle, Bradley, Saris, Christiaan J.M., Wong, Lu Min, Chmait, Samer, Lee, Matthew R., Mohr, Christopher, Hsieh, Faye, Tasker, Andrew S.
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
Published in Bioorganic & medicinal chemistry letters (15.01.2012)
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