Discovery of a Parenteral Small Molecule Coagulation Factor XIa Inhibitor Clinical Candidate (BMS-962212)
Pinto, Donald J. P., Orwat, Michael J., Smith, Leon M., Quan, Mimi L., Lam, Patrick Y. S., Rossi, Karen A., Apedo, Atsu, Bozarth, Jeffrey M., Wu, Yiming, Zheng, Joanna J., Xin, Baomin, Toussaint, Nathalie, Stetsko, Paul, Gudmundsson, Olafur, Maxwell, Brad, Crain, Earl J., Wong, Pancras C., Lou, Zhen, Harper, Timothy W., Chacko, Silvi A., Myers, Joseph E., Sheriff, Steven, Zhang, Huiping, Hou, Xiaoping, Mathur, Arvind, Seiffert, Dietmar A., Wexler, Ruth R., Luettgen, Joseph M., Ewing, William R.
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Journal Article
Annotation of 2,507 Saccharomyces cerevisiae genomes
Wang, Meng, Li, Xuan, Liu, Xian, Hou, Xiaoping, He, Yang, Yu, Jun-Hong, Hu, Shumin, Yin, Hua, Xie, Bin-Bin
Published in Microbiology spectrum (02.04.2024)
Published in Microbiology spectrum (02.04.2024)
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Journal Article
Regioselective Epoxide Ring Opening for the Stereospecific Scale-Up Synthesis of BMS-960, A Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
Hou, Xiaoping, Zhang, Huiping, Chen, Bang-Chi, Guo, Zhiwei, Singh, Amarjit, Goswami, Animesh, Gilmore, John L, Sheppeck, James E, Dyckman, Alaric J, Carter, Percy H, Mathur, Arvind
Published in Organic process research & development (17.02.2017)
Published in Organic process research & development (17.02.2017)
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Journal Article
An Efficient Scale-Up Synthesis of BMS-520, a Potent and Selective Isoxazole-Containing S1P1 Receptor Agonist
Hou, Xiaoping, Zhu, Juliang, Chen, Bang-Chi, Watterson, Scott H, Pitts, William J, Dyckman, Alaric J, Carter, Percy H, Mathur, Arvind, Zhang, Huiping
Published in Organic process research & development (20.05.2016)
Published in Organic process research & development (20.05.2016)
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Journal Article
Discovery of novel aminothiadiazole amides as selective EP3 receptor antagonists
Hilfiker, Mark A., Wang, Ning, Hou, Xiaoping, Du, Zhimin, Pullen, Mark A., Nord, Melanie, Nagilla, Rakesh, Fries, Harvey E., Wu, Charlene W., Sulpizio, Anthony C., Jaworski, Jon-Paul, Morrow, Dwight, Edwards, Richard M., Jin, Jian
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Journal Article
The effect of water on the large-scale supercritical fluid chromatography purification of two factor XIa active pharmaceutical ingredients
Li, Peng, Wu, Dauh-Rurng, Yip, Henry, Sun, Dawn, Zhang, Huiping, Hou, Xiaoping, Kempson, James, Mathur, Arvind
Published in Journal of Chromatography A (16.08.2021)
Published in Journal of Chromatography A (16.08.2021)
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Journal Article
Genome-Wide Expression Pattern Analyses of the Arabidopsis Leucine-Rich Repeat Receptor-Like Kinases
Wu, Yunzhe, Xun, Qingqing, Guo, Yi, Zhang, Jinghua, Cheng, Kaili, Shi, Tao, He, Kai, Hou, Suiwen, Gou, Xiaoping, Li, Jia
Published in Molecular plant (01.02.2016)
Published in Molecular plant (01.02.2016)
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Journal Article
Large-scale supercritical fluid chromatography purification of unstable STING agonist intermediates
Sun, Dawn, Wu, Dauh-Rurng, Li, Peng, Yip, Henry, Wang, Bei, Hou, Xiaoping, Zhao, Rulin, Zhang, Huiping, Kempson, James, Mathur, Arvind
Published in Journal of Chromatography A (16.08.2021)
Published in Journal of Chromatography A (16.08.2021)
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Journal Article
Wort composition and its impact on the flavour-active higher alcohol and ester formation of beer - a review
He, Yang, Dong, Jianjun, Yin, Hua, Zhao, Yuxiang, Chen, Rong, Wan, Xiujuan, Chen, Peng, Hou, Xiaoping, Liu, Jia, Chen, Lu
Published in Journal of the Institute of Brewing (01.06.2014)
Published in Journal of the Institute of Brewing (01.06.2014)
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Journal Article
Discovery of Milvexian, a High-Affinity, Orally Bioavailable Inhibitor of Factor XIa in Clinical Studies for Antithrombotic Therapy
Dilger, Andrew K, Pabbisetty, Kumar B, Corte, James R, De Lucca, Indawati, Fang, Tianan, Yang, Wu, Pinto, Donald J. P, Wang, Yufeng, Zhu, Yeheng, Mathur, Arvind, Li, Jianqing, Hou, Xiaoping, Smith, Daniel, Sun, Dawn, Zhang, Huiping, Krishnananthan, Subramaniam, Wu, Dauh-Rurng, Myers, Joseph E, Sheriff, Steven, Rossi, Karen A, Chacko, Silvi, Zheng, Joanna J, Galella, Michael A, Ziemba, Theresa, Dierks, Elizabeth A, Bozarth, Jeffrey M, Wu, Yiming, Crain, Earl, Wong, Pancras C, Luettgen, Joseph M, Wexler, Ruth R, Ewing, William R
Published in Journal of medicinal chemistry (10.02.2022)
Published in Journal of medicinal chemistry (10.02.2022)
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Journal Article
Challenges with the Synthesis of a Macrocyclic Thioether Peptide: From Milligram to Multigram Using Solid Phase Peptide Synthesis (SPPS)
Kempson, James, Zhao, Rulin, Pawluczyk, Joseph, Wang, Bei, Zhang, Huiping, Hou, Xiaoping, Allen, Martin P., Wu, Dauh-Rurng, Li, Peng, Yip, Shiuhang, Smith, Aaron, Traeger, Sarah C., Huang, Stella, Cutrone, Jingfang, Mukherjee, Subha, Sfouggatakis, Chris, Poss, Michael, Scola, Paul M., Meanwell, Nicholas A., Carter, Percy H., Mathur, Arvind
Published in Journal of organic chemistry (17.05.2024)
Published in Journal of organic chemistry (17.05.2024)
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Journal Article
Reduced sensitivity of lager brewing yeast to premature yeast flocculation via adaptive evolution
He, Yang, Yin, Hua, Dong, Jianjun, Yu, Junhong, Zhang, Lei, Yan, Peng, Wan, Xiujuan, Hou, Xiaoping, Zhao, Yuxiang, Chen, Rong, Gibson, Brian, Krogerus, Kristoffer
Published in Food microbiology (01.09.2022)
Published in Food microbiology (01.09.2022)
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Journal Article
Discovery of a Parenteral Small Molecule Coagulation Factor Xla Inhibitor Clinical Candidate (BMS-962212)
Pinto, Donald J. P., Orwat, Michael J., Smith, Leon M., Quan, Mimi L., Lam, Patrick Y. S., Rossi, Karen A., Apedo, Atsu, Bozarth, Jeffrey M., Wu, Yiming, Zheng, Joanna J., Xin, Baomin, Toussaint, Nathalie, Stetsko, Paul, Gudmundsson, Olafur, Maxwell, Brad, Crain, Earl J., Wong, Pancras C., Lou, Zhen, Harper, Timothy W., Chacko, Silvi A., Myers, Joseph E., Sheriff, Steven, Zhang, Huiping, Hou, Xiaoping, Mathur, Arvind, Seiffert, Dietmar A., Wexler, Ruth R., Luettgen, Joseph M., Ewing, William R.
Published in Journal of medicinal chemistry (14.12.2017)
Published in Journal of medicinal chemistry (14.12.2017)
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Journal Article
The Discovery of GSK3640254, a Next-Generation Inhibitor of HIV‑1 Maturation
Regueiro-Ren, Alicia, Sit, Sing-Yuen, Chen, Yan, Chen, Jie, Swidorski, Jacob J., Liu, Zheng, Venables, Brian L., Sin, Ny, Hartz, Richard A., Protack, Tricia, Lin, Zeyu, Zhang, Sharon, Li, Zhufang, Wu, Dauh-Rurng, Li, Peng, Kempson, James, Hou, Xiaoping, Gupta, Anuradha, Rampulla, Richard, Mathur, Arvind, Park, Hyunsoo, Sarjeant, Amy, Benitex, Yulia, Rahematpura, Sandhya, Parker, Dawn, Phillips, Thomas, Haskell, Roy, Jenkins, Susan, Santone, Kenneth S., Cockett, Mark, Hanumegowda, Umesh, Dicker, Ira, Meanwell, Nicholas A., Krystal, Mark
Published in Journal of medicinal chemistry (22.09.2022)
Published in Journal of medicinal chemistry (22.09.2022)
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Journal Article
Evolution of the Synthetic Process to an Advanced GPR40 Agonist
Hou, Xiaoping, Hernandez, Lucas W., Jurica, Elizabeth A., Zhao, Rulin, Wang, Bei, Wong, Michael, Sun, Jung-Hui, Sun, Dawn, Wu, Dauh-Rurng, Yuan, Changxia, Hay, Michael, Yu, Miao, Wu, Ximao, Huang, Yanting, Ellsworth, Bruce A., Bobes, Francisco Gonzalez, Mathur, Arvind, Kempson, James
Published in Organic process research & development (19.01.2024)
Published in Organic process research & development (19.01.2024)
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Journal Article
Regioselective Epoxide Ring Opening for the Stereospecific Scale-Up Synthesis of BMS-960, A Potent and Selective Isoxazole-Containing S1P(1) Receptor Agonist
Hou, Xiaoping, Zhang, Huiping, Chen, Bang-Chi, Guo, Zhiwei, Singh, Amarjit, Goswami, Animesh, Gilmore, John L., Sheppeck, James E., Dyckman, Alaric J., Carter, Percy H., Mathur, Arvind
Published in Organic process research & development (01.02.2017)
Published in Organic process research & development (01.02.2017)
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Journal Article
Discovery of novel pyridinones as MGAT2 inhibitors for the treatment of metabolic disorders
Moore, Fang, Wang, Wei, Zhao, Guohua, Mignone, James, Meng, Wei, Chu, Ching-Hsuen, Ma, Zhengping, Azzara, Anthony, Cullen, Mary Jane, Pelleymounter, Mary Ann, Appiah, Kingsley, Cvijic, Mary Ellen, Dierks, Elizabeth, Chang, Shu, Foster, Kimberly, Kopcho, Lisa, O'Malley, Kevin, Li, Yi-Xin, Khandelwal, Purnima, Whaley, Jean M., Mathur, Arvind, Hou, Xiaoping, Wu, Dauh-Rurng, Robl, Jeffrey A., Cheng, Dong, Devasthale, Pratik
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
Published in Bioorganic & medicinal chemistry letters (15.07.2023)
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Journal Article
Development of a Rapid Scale-Up Synthesis of ( S )- N -(8-((2-Amino-2,4-dimethylpentyl)oxy)-5 H -chromeno[3,4- c ]pyridin-2-yl)acetamide, a Potent Adaptor-Associated Kinase 1 Inhibitor
Li, Jianqing, Smith, Daniel, Pawluczyk, Joseph, Krishnananthan, Subramaniam, Wang, Bei, Hou, Xiaoping, Zhao, Rulin, Kempson, James, Sun, Dawn, Yip, Shiuhang, Wu, Dauh-Rurng, Maddala, Nageswararao, Vetrichelvan, Muthalagu, Gupta, Anuradha, Macor, John E., Dzierba, Carolyn D., Mathur, Arvind
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
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