Biology of the Major Facilitative Folate Transporters SLC19A1 and SLC46A1
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Book Chapter
Journal Article
Human reduced folate carrier: translation of basic biology to cancer etiology and therapy
Matherly, Larry H, Hou, Zhanjun, Deng, Yijun
Published in Cancer and metastasis reviews (01.03.2007)
Published in Cancer and metastasis reviews (01.03.2007)
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Journal Article
Targeted therapy of pyrrolo[2,3-d]pyrimidine antifolates in a syngeneic mouse model of high grade serous ovarian cancer and the impact on the tumor microenvironment
Wallace-Povirk, Adrianne, Rubinsak, Lisa, Malysa, Agnes, Dzinic, Sijana H, Ravindra, Manasa, Schneider, Mathew, Glassbrook, James, O'Connor, Carrie, Hou, Zhanjun, Kim, Seongho, Back, Jessica, Polin, Lisa, Morris, Robert T, Gangjee, Aleem, Gibson, Heather, Matherly, Larry H
Published in Scientific reports (05.07.2022)
Published in Scientific reports (05.07.2022)
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Journal Article
Dual Targeting of Epithelial Ovarian Cancer Via Folate Receptor α and the Proton-Coupled Folate Transporter with 6-Substituted Pyrrolo[2,3- d ]pyrimidine Antifolates
Hou, Zhanjun, Gattoc, Leda, O'Connor, Carrie, Yang, Si, Wallace-Povirk, Adrianne, George, Christina, Orr, Steve, Polin, Lisa, White, Kathryn, Kushner, Juiwanna, Morris, Robert T, Gangjee, Aleem, Matherly, Larry H
Published in Molecular cancer therapeutics (01.05.2017)
Published in Molecular cancer therapeutics (01.05.2017)
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Journal Article
Folate Transport and One-Carbon Metabolism in Targeted Therapies of Epithelial Ovarian Cancer
Wallace-Povirk, Adrianne, Hou, Zhanjun, Nayeen, Md Junayed, Gangjee, Aleem, Matherly, Larry H
Published in Cancers (31.12.2021)
Published in Cancers (31.12.2021)
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Journal Article
Synthesis and Discovery of High Affinity Folate Receptor-Specific Glycinamide Ribonucleotide Formyltransferase Inhibitors with Antitumor Activity
Deng, Yijun, Wang, Yiqiang, Cherian, Christina, Hou, Zhanjun, Buck, Steven A, Matherly, Larry H, Gangjee, Aleem
Published in Journal of medicinal chemistry (28.08.2008)
Published in Journal of medicinal chemistry (28.08.2008)
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Journal Article
Synthesis and Biological Activity of a Novel Series of 6-Substituted Thieno[2,3-d]pyrimidine Antifolate Inhibitors of Purine Biosynthesis with Selectivity for High Affinity Folate Receptors over the Reduced Folate Carrier and Proton-Coupled Folate Transporter for Cellular Entry
Deng, Yijun, Zhou, Xilin, Kugel Desmoulin, Sita, Wu, Jianmei, Cherian, Christina, Hou, Zhanjun, Matherly, Larry H, Gangjee, Aleem
Published in Journal of medicinal chemistry (14.05.2009)
Published in Journal of medicinal chemistry (14.05.2009)
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Journal Article
Synthesis and Antitumor Activity of a Novel Series of 6-Substituted Pyrrolo[2,3-d]pyrimidine Thienoyl Antifolate Inhibitors of Purine Biosynthesis with Selectivity for High Affinity Folate Receptors and the Proton-Coupled Folate Transporter over the Reduced Folate Carrier for Cellular Entry
Wang, Lei, Cherian, Christina, Kugel Desmoulin, Sita, Polin, Lisa, Deng, Yijun, Wu, Jianmei, Hou, Zhanjun, White, Kathryn, Kushner, Juiwanna, Matherly, Larry H, Gangjee, Aleem
Published in Journal of medicinal chemistry (11.02.2010)
Published in Journal of medicinal chemistry (11.02.2010)
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Journal Article
Therapeutic targeting of a novel 6-substituted pyrrolo [2,3-d]pyrimidine thienoyl antifolate to human solid tumors based on selective uptake by the proton-coupled folate transporter
Kugel Desmoulin, Sita, Wang, Lei, Hales, Eric, Polin, Lisa, White, Kathryn, Kushner, Juiwanna, Stout, Mark, Hou, Zhanjun, Cherian, Christina, Gangjee, Aleem, Matherly, Larry H
Published in Molecular pharmacology (01.12.2011)
Published in Molecular pharmacology (01.12.2011)
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Journal Article
Pattern Analysis of Organellar Maps for Interpretation of Proteomic Data
Burton, Jordan B, Carruthers, Nicholas J, Hou, Zhanjun, Matherly, Larry H, Stemmer, Paul M
Published in Proteomes (23.05.2022)
Published in Proteomes (23.05.2022)
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Journal Article
Discovery of 5‑Substituted Pyrrolo[2,3‑d]pyrimidine Antifolates as Dual-Acting Inhibitors of Glycinamide Ribonucleotide Formyltransferase and 5‑Aminoimidazole-4-carboxamide Ribonucleotide Formyltransferase in De Novo Purine Nucleotide Biosynthesis: Implications of Inhibiting 5‑Aminoimidazole-4-carboxamide Ribonucleotide Formyltransferase to AMPK Activation and Antitumor Activity
Mitchell-Ryan, Shermaine, Wang, Yiqiang, Raghavan, Sudhir, Ravindra, Manasa Punaha, Hales, Eric, Orr, Steven, Cherian, Christina, Hou, Zhanjun, Matherly, Larry H, Gangjee, Aleem
Published in Journal of medicinal chemistry (27.12.2013)
Published in Journal of medicinal chemistry (27.12.2013)
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Journal Article
Structural determinants of human proton-coupled folate transporter oligomerization: role of GXXXG motifs and identification of oligomeric interfaces at transmembrane domains 3 and 6
Wilson, Mike R, Kugel, Sita, Huang, Jenny, Wilson, Lucas J, Wloszczynski, Patrick A, Ye, Jun, Matherly, Larry H, Hou, Zhanjun
Published in Biochemical journal (01.07.2015)
Published in Biochemical journal (01.07.2015)
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Journal Article
Identification and Functional Impact of Homo-oligomers of the Human Proton-coupled Folate Transporter
Hou, Zhanjun, Kugel Desmoulin, Sita, Etnyre, Erika, Olive, Mary, Hsiung, Benjamin, Cherian, Christina, Wloszczynski, Patrick A., Moin, Kamiar, Matherly, Larry H.
Published in The Journal of biological chemistry (10.02.2012)
Published in The Journal of biological chemistry (10.02.2012)
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Journal Article
Therapeutic targeting malignant mesothelioma with a novel 6-substituted pyrrolo[2,3-d]pyrimidine thienoyl antifolate via its selective uptake by the proton-coupled folate transporter
Cherian, Christina, Kugel Desmoulin, Sita, Wang, Lei, Polin, Lisa, White, Kathryn, Kushner, Juiwanna, Stout, Mark, Hou, Zhanjun, Gangjee, Aleem, Matherly, Larry H.
Published in Cancer chemotherapy and pharmacology (01.04.2013)
Published in Cancer chemotherapy and pharmacology (01.04.2013)
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Journal Article