New Strategic Reactions for Organic Synthesis: Catalytic Asymmetric C−H Activation α to Nitrogen as a Surrogate for the Mannich Reaction
Davies, Huw M. L, Venkataramani, Chandrasekar, Hansen, Tore, Hopper, Darrin W
Published in Journal of the American Chemical Society (28.05.2003)
Published in Journal of the American Chemical Society (28.05.2003)
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Journal Article
Highly Regio-, Diastereo-, and Enantioselective C−H Insertions of Methyl Aryldiazoacetates into Cyclic N-Boc-Protected Amines. Asymmetric Synthesis of Novel C 2-Symmetric Amines and threo-Methylphenidate
Davies, Huw M. L, Hansen, Tore, Hopper, Darrin W, Panaro, Stephen A
Published in Journal of the American Chemical Society (14.07.1999)
Published in Journal of the American Chemical Society (14.07.1999)
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Novel pyrazolopyrimidines as highly potent B-Raf inhibitors
Di Grandi, Martin J., Berger, Dan M., Hopper, Darrin W., Zhang, Chunchun, Dutia, Minu, Dunnick, Alejandro L., Torres, Nancy, Levin, Jeremy I., Diamantidis, George, Zapf, Christoph W., Bloom, Jonathan D., Hu, YongBo, Powell, Dennis, Wojciechowicz, Donald, Collins, Karen, Frommer, Eileen
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
Published in Bioorganic & medicinal chemistry letters (15.12.2009)
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Journal Article
Synthesis and biological evaluation of tricyclic anilinopyrimidines as IKKβ inhibitors
Crombie, Aimee L., Sum, Fuk-Wah, Powell, Dennis W., Hopper, Darrin W., Torres, Nancy, Berger, Dan M., Zhang, Yixian, Gavriil, Maria, Sadler, Tammy M., Arndt, Kim
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Journal Article
Synthesis and biological evaluation of ((4-keto)-phenoxy)methyl biphenyl-4-sulfonamides: A class of potent aggrecanase-1 inhibitors
Hopper, Darrin W., Vera, Matthew D., How, David, Sabatini, Joshua, Xiang, Jason S., Ipek, Manus, Thomason, Jennifer, Hu, Yonghan, Feyfant, Eric, Wang, Qin, Georgiadis, Katy E., Reifenberg, Erica, Sheldon, Richard T., Keohan, Cristin C., Majumdar, Manas K., Morris, Elisabeth A., Skotnicki, Jerauld, Sum, Phaik-Eng
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
Published in Bioorganic & medicinal chemistry letters (01.05.2009)
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Journal Article
Quantification in Patient Urine Samples of Felbamate and Three Metabolites: Acid Carbamate and Two Mercapturic Acids
Thompson, Charles D., Barthen, Mary T., Hopper, Darrin W., Miller, Thomas A., Quigg, Mark, Hudspeth, Candice, Montouris, Georgia, Marsh, LaDonna, Perhach, James L., Sofia, R. Duane, Macdonald, Timothy L.
Published in Epilepsia (Copenhagen) (01.06.1999)
Published in Epilepsia (Copenhagen) (01.06.1999)
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Journal Article
Characterization of a Receptor Subtype-Selective Lysophosphatidic Acid Mimetic
Hooks, S B, Ragan, S P, Hopper, D W, Hönemann, C W, Durieux, M E, Macdonald, T L, Lynch, K R
Published in Molecular pharmacology (01.02.1998)
Published in Molecular pharmacology (01.02.1998)
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Structure/Activity Relationships in Lysophosphatidic Acid: The 2-Hydroxyl Moiety
Lynch, K R, Hopper, D W, Carlisle, S J, Catalano, J G, Zhang, M, MacDonald, T L
Published in Molecular pharmacology (01.07.1997)
Published in Molecular pharmacology (01.07.1997)
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Journal Article
Facile synthesis of lysophospholipids containing unsaturated fatty acid chains
Hopper, Darrin W., Catalano, John G., Macdonald, Timothy L.
Published in Tetrahedron letters (28.10.1996)
Published in Tetrahedron letters (28.10.1996)
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Journal Article
Highly Regio-, Diastereo-, and Enantioselective C−H Insertions of Methyl Aryldiazoacetates into Cyclic N-Boc-Protected Amines. Asymmetric Synthesis of Novel C2-Symmetric Amines and threo-Methylphenidate
DAVIES, Huw M. L., HANSEN, Tore, HOPPER, Darrin W., PANARO, Stephen A.
Published in Journal of the American Chemical Society (14.07.1999)
Published in Journal of the American Chemical Society (14.07.1999)
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Journal Article
Observation of differential reactivity of cyclic amines in SN2 and SNAr displacement reactions in the course of synthesizing C-6, C-7 substituted quinolinecarbonitrile MEK1 kinase inhibitors
Hopper, Darrin W., Dutia, Minu, Berger, Dan M., Powell, Dennis W.
Published in Tetrahedron letters (01.01.2008)
Published in Tetrahedron letters (01.01.2008)
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Journal Article
Observation of differential reactivity of cyclic amines in S(N)2 and SNAr displacement reactions in the course of synthesizing C-6, C-7 substituted quinolinecarbonitrile MEK1 kinase inhibitors
Hopper, Darrin W., Dutia, Minu, Berger, Dan M., Powell, Dennis W.
Published in Tetrahedron letters (01.01.2008)
Published in Tetrahedron letters (01.01.2008)
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Journal Article
Observation of differential reactivity of cyclic amines in S N2 and S NAr displacement reactions in the course of synthesizing C-6, C-7 substituted quinolinecarbonitrile MEK1 kinase inhibitors
Hopper, Darrin W., Dutia, Minu, Berger, Dan M., Powell, Dennis W.
Published in Tetrahedron letters (2008)
Published in Tetrahedron letters (2008)
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Journal Article
New strategic reactions for organic synthesis: Catalytic asymmetric C-H activation a to nitrogen as a surrogate for the mannich reaction
DAVIES, Huw M. L, VENKATARAMANI, Chandrasekar, HANSEN, Tore, HOPPER, Darrin W
Published in Journal of the American Chemical Society (2003)
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Published in Journal of the American Chemical Society (2003)
Journal Article
Synthesis and biological evaluation of tricyclic anilinopyrimidines as IKKbeta inhibitors
Crombie, Aimee L, Sum, Fuk-Wah, Powell, Dennis W, Hopper, Darrin W, Torres, Nancy, Berger, Dan M, Zhang, Yixian, Gavriil, Maria, Sadler, Tammy M, Arndt, Kim
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
Published in Bioorganic & medicinal chemistry letters (15.06.2010)
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Journal Article
ChemInform Abstract: Six-Membered Ring Systems: Pyridine and Benzo Derivatives
Hopper, Darrin W., Crombie, Aimee L., Clemens, Jeremy J., Kwon, Soojin
Published in ChemInform (11.05.2010)
Published in ChemInform (11.05.2010)
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Journal Article
ChemInform Abstract: Six-Membered Ring Systems - Pyridine and Benzo Derivatives
Hopper, Darrin W., Kutterer, Kristina M. K., Crombie, Aimee L., Clemens, Jeremy J.
Published in ChemInform (03.11.2009)
Published in ChemInform (03.11.2009)
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