Antiplasmodial and Cytotoxic Flavonoids from Pappea capensis (Eckl. & Zeyh.) Leaves
Tajuddeen, Nasir, Swart, Tarryn, Hoppe, Heinrich C., van Heerden, Fanie R.
Published in Molecules (Basel, Switzerland) (25.06.2021)
Published in Molecules (Basel, Switzerland) (25.06.2021)
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Journal Article
Potential repurposing of four FDA approved compounds with antiplasmodial activity identified through proteome scale computational drug discovery and in vitro assay
Diallo, Bakary N’tji, Swart, Tarryn, Hoppe, Heinrich C., Tastan Bishop, Özlem, Lobb, Kevin
Published in Scientific reports (14.01.2021)
Published in Scientific reports (14.01.2021)
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Identification of Novel Potential Inhibitors of Pteridine Reductase 1 in Trypanosoma brucei via Computational Structure-Based Approaches and in Vitro Inhibition Assays
Kimuda, Magambo Phillip, Laming, Dustin, Hoppe, Heinrich C, Tastan Bishop, Özlem
Published in Molecules (Basel, Switzerland) (01.01.2019)
Published in Molecules (Basel, Switzerland) (01.01.2019)
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Coumarin-Annulated Ferrocenyl 1,3-Oxazine Derivatives Possessing In Vitro Antimalarial and Antitrypanosomal Potency
Mbaba, Mziyanda, Dingle, Laura M K, Zulu, Ayanda I, Laming, Dustin, Swart, Tarryn, de la Mare, Jo-Anne, Hoppe, Heinrich C, Edkins, Adrienne L, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (02.03.2021)
Published in Molecules (Basel, Switzerland) (02.03.2021)
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Hydrazone‐Tethered 5‐(Pyridin‐4‐yl)‐4H‐1,2,4‐triazole‐3‐thiol Hybrids: Synthesis, Characterisation, in silico ADME Studies, and in vitro Antimycobacterial Evaluation and Cytotoxicity
Oderinlo, Ogunyemi O., Jordaan, Audrey, Seldon, Ronnett, Isaacs, Michelle, Hoppe, Heinrich C., Warner, Digby F., Tukulula, Matshawandile, Khanye, Setshaba D.
Published in ChemMedChem (14.03.2023)
Published in ChemMedChem (14.03.2023)
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Journal Article
Easy-To-Access Quinolone Derivatives Exhibiting Antibacterial and Anti-Parasitic Activities
Beteck, Richard M, Jordaan, Audrey, Seldon, Ronnett, Laming, Dustin, Hoppe, Heinrich C, Warner, Digby F, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (20.02.2021)
Published in Molecules (Basel, Switzerland) (20.02.2021)
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Journal Article
New Quinolone-Based Thiosemicarbazones Showing Activity Against Plasmodium falciparum and Mycobacterium tuberculosis
Beteck, Richard M, Seldon, Ronnett, Jordaan, Audrey, Warner, Digby F, Hoppe, Heinrich C, Laming, Dustin, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (04.05.2019)
Published in Molecules (Basel, Switzerland) (04.05.2019)
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Journal Article
Synthesis, Structure and In Vitro Anti-Trypanosomal Activity of Non-Toxic Arylpyrrole-Based Chalcone Derivatives
Zulu, Ayanda I, Oderinlo, Ogunyemi O, Kruger, Cuan, Isaacs, Michelle, Hoppe, Heinrich C, Smith, Vincent J, Veale, Clinton G L, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (04.04.2020)
Published in Molecules (Basel, Switzerland) (04.04.2020)
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Journal Article
Isolation, Chemical Profile and Antimalarial Activities of Bioactive Compounds from Rauvolfia caffra Sond
Tlhapi, Dorcas B, Ramaite, Isaiah D I, Van Ree, Teunis, Anokwuru, Chinedu P, Orazio, Taglialatela-Scafati, Hoppe, Heinrich C
Published in Molecules (Basel, Switzerland) (21.12.2018)
Published in Molecules (Basel, Switzerland) (21.12.2018)
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Journal Article
Cinnamoyl-Oxaborole Amides: Synthesis and Their in Vitro Biological Activity
Gumbo, Maureen, Beteck, Richard M, Mandizvo, Tawanda, Seldon, Ronnett, Warner, Digby F, Hoppe, Heinrich C, Isaacs, Michelle, Laming, Dustin, Tam, Christina C, Cheng, Luisa W, Liu, Nicole, Land, Kirkwood M, Khanye, Setshaba D
Published in Molecules (Basel, Switzerland) (15.08.2018)
Published in Molecules (Basel, Switzerland) (15.08.2018)
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Journal Article
Wherever I may roam: Protein and membrane trafficking in P. falciparum-infected red blood cells
Deponte, Marcel, Hoppe, Heinrich C., Lee, Marcus C.S., Maier, Alexander G., Richard, Dave, Rug, Melanie, Spielmann, Tobias, Przyborski, Jude M.
Published in Molecular and biochemical parasitology (01.12.2012)
Published in Molecular and biochemical parasitology (01.12.2012)
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In vitro antiplasmodium and antitrypanosomal activities, β-haematin formation inhibition, molecular docking and DFT computational studies of quinoline-urea-benzothiazole hybrids
Oyeneyin, Oluwatoba E., Moodley, Rashmika, Mashaba, Chakes, Garnie, Larnelle F., Omoboyowa, Damilola A., Rakodi, Goitsemodimo H., Maphoru, Mabuatsela V., Balogun, Mohamed O., Hoppe, Heinrich C., Egan, Timothy J., Tukulula, Matshawandile
Published in Heliyon (15.10.2024)
Published in Heliyon (15.10.2024)
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Journal Article
Anti-Trypanosomal and Antimalarial Properties of Tetralone Derivatives and Structurally Related Benzocycloalkanones
Beteck, Richard M, Legoabe, Lesetja J, Isaacs, Michelle, Khanye, Setshaba D, Laming, Dustin, Hoppe, Heinrich C
Published in Medicina (Kaunas, Lithuania) (24.05.2019)
Published in Medicina (Kaunas, Lithuania) (24.05.2019)
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Journal Article
Biological activities of plant extracts from Ficus elastica and Selaginella vogelli: An antimalarial, antitrypanosomal and cytotoxity evaluation
Mbosso Teinkela, Jean Emmanuel, Siwe Noundou, Xavier, Nguemfo, Edwige Laure, Meyer, Franck, Wintjens, Rene, Isaacs, Michelle, Mpondo Mpondo, Albert Emmanuel, Hoppe, Heinrich C., Krause, Rui Werner Maçedo, Azebaze, Anatole Guy Blaise
Published in Saudi journal of biological sciences (01.01.2018)
Published in Saudi journal of biological sciences (01.01.2018)
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Heterologous expression of plasmodial proteins for structural studies and functional annotation
Birkholtz, Lyn-Marie, Blatch, Gregory, Coetzer, Theresa L, Hoppe, Heinrich C, Human, Esmaré, Morris, Elizabeth J, Ngcete, Zoleka, Oldfield, Lyndon, Roth, Robyn, Shonhai, Addmore, Stephens, Linda, Louw, Abraham I
Published in Malaria journal (01.10.2008)
Published in Malaria journal (01.10.2008)
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Journal Article
Differential Effects of Quinoline Antimalarials on Endocytosis in Plasmodium falciparum
Roberts, Lindi, Egan, Timothy J, Joiner, Keith A, Hoppe, Heinrich C
Published in Antimicrobial Agents and Chemotherapy (01.05.2008)
Published in Antimicrobial Agents and Chemotherapy (01.05.2008)
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Journal Article
Antiplasmodial Activity of the n -Hexane Extract from Pleurotus ostreatus (Jacq. ex. Fr) P. Kumm
Afieroho, Ozadheoghene Eriarie, Noundou, Xavier Siwe, Onyia, Chiazor P, Festus, Osamuyi H, Chukwu, Elizabeth C, Adedokun, Olutayo M, Isaacs, Michelle, Hoppe, Heinrich C, Krause, Rui Wm, Abo, Kio A
Published in Turkish journal of pharmaceutical sciences (01.03.2019)
Published in Turkish journal of pharmaceutical sciences (01.03.2019)
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