High‐Throughput Reaction Optimisation and Activity Screening of Ferrocene‐Based Lewis Acid–Catalyst Complexes by Using Continuous‐Flow Reaction Detection Mass Spectrometry
Martha, Cornelius T., Heemskerk, Anton, Hoogendoorn, Jan‐Carel, Elders, Niels, Niessen, Wilfried M. A., Orru, Romano V. A., Irth, Hubertus
Published in Chemistry : a European journal (27.07.2009)
Published in Chemistry : a European journal (27.07.2009)
Get full text
Journal Article
Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel 3,4-Diarylpyrazolines as Potent and Selective CB1 Cannabinoid Receptor Antagonists
Lange, Jos H. M, Coolen, Hein K. A. C, van Stuivenberg, Herman H, Dijksman, Jessica A. R, Herremans, Arnoud H. J, Ronken, Eric, Keizer, Hiskias G, Tipker, Koos, McCreary, Andrew C, Veerman, Willem, Wals, Henri C, Stork, Bob, Verveer, Peter C, den Hartog, Arnold P, de Jong, Natasja M. J, Adolfs, Tiny J. P, Hoogendoorn, Jan, Kruse, Chris G
Published in Journal of medicinal chemistry (29.01.2004)
Published in Journal of medicinal chemistry (29.01.2004)
Get full text
Journal Article
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB1 receptor antagonists
LANGE, Jos H. M, VAN DER NEUT, Martina A. W, DEN HARTOG, Arnold P, WALS, Henri C, HOOGENDOORN, Jan, VAN STUIVENBERG, Herman H, VAN VLIET, Bernard J, KRUSE, Chris G
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Get full text
Journal Article
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB 1 receptor antagonists
Lange, Jos H.M., van der Neut, Martina A.W., den Hartog, Arnold P., Wals, Henri C., Hoogendoorn, Jan, van Stuivenberg, Herman H., van Vliet, Bernard J., Kruse, Chris G.
Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
Get full text
Journal Article
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB sub(1) receptor antagonists
Lange, Jos HM, Van der Neut, Martina AW, Hartog, Arnold Pden, Wals, Henri C, Hoogendoorn, Jan, Van Stuivenberg, Herman H, Van Vliet, Bernard J, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Get full text
Journal Article
Desalination of brackish groundwater: the concentrate dilemma
Get full text
Journal Article
Conference Proceeding
Synthesis, SAR and intramolecular hydrogen bonding pattern of 1,3,5-trisubstituted 4,5-dihydropyrazoles as potent cannabinoid CB(1) receptor antagonists
Lange, Jos H M, van der Neut, Martina A W, den Hartog, Arnold P, Wals, Henri C, Hoogendoorn, Jan, van Stuivenberg, Herman H, van Vliet, Bernard J, Kruse, Chris G
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Get full text
Journal Article
Synthesis, biological properties, and molecular modeling investigations of novel 3,4-diarylpyrazolines as potent and selective CB(1) cannabinoid receptor antagonists
Lange, Jos H M, Coolen, Hein K A C, van Stuivenberg, Herman H, Dijksman, Jessica A R, Herremans, Arnoud H J, Ronken, Eric, Keizer, Hiskias G, Tipker, Koos, McCreary, Andrew C, Veerman, Willem, Wals, Henri C, Stork, Bob, Verveer, Peter C, den Hartog, Arnold P, de Jong, Natasja M J, Adolfs, Tiny J P, Hoogendoorn, Jan, Kruse, Chris G
Published in Journal of medicinal chemistry (29.01.2004)
Get full text
Published in Journal of medicinal chemistry (29.01.2004)
Journal Article
Synthesis, Biological Properties, and Molecular Modeling Investigations of Novel 3,4-Diarylpyrazolines as Potent and Selective CB 1 Cannabinoid Receptor Antagonists
Lange, Jos H. M., Coolen, Hein K. A. C., van Stuivenberg, Herman H., Dijksman, Jessica A. R., Herremans, Arnoud H. J., Ronken, Eric, Keizer, Hiskias G., Tipker, Koos, McCreary, Andrew C., Veerman, Willem, Wals, Henri C., Stork, Bob, Verveer, Peter C., den Hartog, Arnold P., de Jong, Natasja M. J., Adolfs, Tiny J. P., Hoogendoorn, Jan, Kruse, Chris G.
Published in Journal of medicinal chemistry (01.01.2004)
Published in Journal of medicinal chemistry (01.01.2004)
Get full text
Journal Article
4,5-DIHYDRO-1H-PYRAZOLE DERIVATIVES HAVING CB1-ANTAGONISTIC ACTIVITY
LANGE, JOSEPHUS H.M, HOOGENDOORN, JAN, TIPKER, JACOBUS, KRUSE, CORNELIS G
Year of Publication 26.10.2010
Get full text
Year of Publication 26.10.2010
Patent