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Published in Bioorganic & medicinal chemistry letters (2010)
Published in Bioorganic & medicinal chemistry letters (2010)
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Discovery of pyrimidyl-5-hydroxamic acids as new potent histone deacetylase inhibitors
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Published in European journal of medicinal chemistry (01.06.2005)
Published in European journal of medicinal chemistry (01.06.2005)
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Synthesis of 3-Amino-4-fluoropyrazoles
Surmont, Riccardo, Verniest, Guido, De Schrijver, Mathias, Thuring, Jan Willem, ten Holte, Peter, Deroose, Frederik, De Kimpe, Norbert
Published in Journal of organic chemistry (20.05.2011)
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Library Enhancement through the Wisdom of Crowds
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Published in Journal of chemical information and modeling (27.12.2011)
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Synthesis of gem-difluorinated 1,6-naphthyridine-5,7-diones
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Published in Tetrahedron (26.08.2012)
Published in Tetrahedron (26.08.2012)
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Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidines
Surmont, Riccardo, Verniest, Guido, Thuring, Jan Willem, ten Holte, Peter, Deroose, Frederik, De Kimpe, Norbert
Published in Organic & biomolecular chemistry (21.10.2010)
Published in Organic & biomolecular chemistry (21.10.2010)
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Synthesis of 2-aryl-3-hydroxymethyl-5,5-difluoropiperidines
Moens, Matthias, Verniest, Guido, De Schrijver, Matthias, ten Holte, Peter, Thuring, Jan-Willem, Deroose, Frederik, De Kimpe, Norbert
Published in Tetrahedron (11.11.2012)
Published in Tetrahedron (11.11.2012)
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Synthesis of 5-amino- and 5-hydroxy-3,3-difluoropiperidinesElectronic supplementary information (ESI) available: Experimental procedures and spectroscopic data for compounds 5a, 6b-d, 8-11 and 13-16 are available. See DOI: 10.1039/c0ob00231c
Surmont, Riccardo, Verniest, Guido, Thuring, Jan Willem, ten Holte, Peter, Deroose, Frederik, De Kimpe, Norbert
Year of Publication 29.09.2010
Year of Publication 29.09.2010
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ChemInform Abstract: Synthesis of gem-Difluorinated 1,6-Naphthyridine-5,7-diones
Piron, Karel, Kenis, Sara, Verniest, Guido, Surmont, Riccardo, Thuring, Jan Willem, ten Holte, Peter, Deroose, Frederik, De Kimpe, Norbert
Published in ChemInform (01.01.2013)
Published in ChemInform (01.01.2013)
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MTP INHIBITING TETRAHYDRO-NAPHTHALENE-1-CARBOXYLIC ACID DERIVATIVES
BACKX, LEO JACOBUS JOZEF, BUSSCHER, GUUSKE FREDERIKE, MEERPOEL, LIEVEN, TEN HOLTE, PETER
Year of Publication 01.12.2015
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Year of Publication 01.12.2015
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