Direct Quantitative Analysis of a 20 kDa PEGylated Human Calcitonin Gene Peptide Antagonist in Cynomolgus Monkey Serum Using In-Source CID and UPLC-MS/MS
Li, Hongyan, Rose, Mark J., Holder, Jerry Ryan, Wright, Marie, Miranda, Les P., James, Christopher A.
Published in Journal of the American Society for Mass Spectrometry (01.09.2011)
Published in Journal of the American Society for Mass Spectrometry (01.09.2011)
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Journal Article
Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the Mouse Melanocortin Receptors: Part 2 Modifications at the Phe Position
Holder, Jerry Ryan, Bauzo, Rayna M, Xiang, Zhimin, Haskell-Luevano, Carrie
Published in Journal of medicinal chemistry (04.07.2002)
Published in Journal of medicinal chemistry (04.07.2002)
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Journal Article
Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the Mouse Melanocortin Receptors. 1. Modifications at the His Position
Holder, Jerry Ryan, Bauzo, Rayna M, Xiang, Zhimin, Haskell-Luevano, Carrie
Published in Journal of medicinal chemistry (20.06.2002)
Published in Journal of medicinal chemistry (20.06.2002)
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Journal Article
Structure−Activity Relationships of the Melanocortin Tetrapeptide Ac-His-d-Phe-Arg-Trp-NH2 at the Mouse Melanocortin Receptors. 4. Modifications at the Trp Position
Holder, Jerry Ryan, Xiang, Zhimin, Bauzo, Rayna M, Haskell-Luevano, Carrie
Published in Journal of medicinal chemistry (19.12.2002)
Published in Journal of medicinal chemistry (19.12.2002)
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Journal Article
GIPR GLP-1 METHOD OF TREATING OR AMELIORATING METABOLIC DISORDERS USING GLP-1 RECEPTOR AGONISTS CONJUGATED TO ANTAGONISTS FOR GASTRIC INHIBITORY PEPTIDE RECEPTORGIPR
YIE JUNMING, NETIROJJANAKUL CHAWITA, VENIANT ELLISON MURIELLE M, STANISLAUS SHANAKA, WU BIN, FALSEY JAMES R, XU JING, HOLDER JERRY RYAN, SHAM KELVIN, MIRANDA LESLIE P, CHENG YUAN, HERBERICH BRADLEY J, LU SHU CHEN
Year of Publication 30.08.2024
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Year of Publication 30.08.2024
Patent
Design and pharmacology of peptoids and peptide-peptoid hybrids based on the melanocortin agonists core tetrapeptide sequence
HOLDER, Jerry Ryan, BAUZO, Rayna M, ZHIMIN XIANG, SCOTT, Joseph, HASKELL-LUEVANO, Carrie
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
Published in Bioorganic & medicinal chemistry letters (15.12.2003)
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Journal Article
Characterization of aliphatic, cyclic, and aromatic N-terminally capped His-D-Phe-Arg-Trp-NH2 tetrapeptides at the melanocortin receptors
HOLDER, Jerry Ryan, MARQUES, Fernanda F, ZHIMIN XIANG, BAUZO, Rayna M, HASKELL-LUEVANO, Carrie
Published in European journal of pharmacology (21.02.2003)
Published in European journal of pharmacology (21.02.2003)
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Journal Article
위 저해 펩타이드 수용체(GIPR)에 대한 길항제에 접합된 GLP-1 수용체 작용제를 사용하여 대사 장애를 치료 또는 개선하는 방법
YIE JUNMING, NETIROJJANAKUL CHAWITA, VENIANT ELLISON MURIELLE M, STANISLAUS SHANAKA, WU BIN, FALSEY JAMES R, XU JING, HOLDER JERRY RYAN, SHAM KELVIN, MIRANDA LESLIE P, CHENG YUAN, HERBERICH BRADLEY J, LU SHU CHEN
Year of Publication 06.09.2019
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Year of Publication 06.09.2019
Patent
Half-life extension of peptidic APJ agonists by N-terminal lipid conjugation
Reed, Anthony B., Lanman, Brian A., Holder, Jerry Ryan, Yang, Bryant H., Ma, Ji, Humphreys, Sara C., Wang, Zhican, Chan, Joyce C.Y., Miranda, Les P., Swaminath, Gayathri, Allen, John G.
Published in Bioorganic & medicinal chemistry letters (01.11.2020)
Published in Bioorganic & medicinal chemistry letters (01.11.2020)
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Journal Article
Identification and Optimization of a Minor Allele-Specific siRNA to Prevent PNPLA3 I148M-Driven Nonalcoholic Fatty Liver Disease
Murray, Justin K, Long, Jason, Liu, Lei, Singh, Shivani, Pruitt, Danielle, Ollmann, Michael, Swearingen, Elissa, Hardy, Miki, Homann, Oliver, Wu, Bin, Holder, Jerry Ryan, Sham, Kelvin, Herberich, Brad, Lo, Mei-Chu, Dou, Hui, Shkumatov, Artem, Florio, Monica, Rulifson, Ingrid C
Published in Nucleic acid therapeutics (01.10.2021)
Published in Nucleic acid therapeutics (01.10.2021)
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Journal Article
Engineering Antibody Reactivity for Efficient Derivatization to Generate NaV1.7 Inhibitory GpTx‑1 Peptide–Antibody Conjugates
Biswas, Kaustav, Nixey, Thomas E, Murray, Justin K, Falsey, James R, Yin, Li, Liu, Hantao, Gingras, Jacinthe, Hall, Brian E, Herberich, Brad, Holder, Jerry Ryan, Li, Hongyan, Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, Soriano, Brian D, Soto, Marcus, Tran, Linh, Tegley, Christopher M, Zou, Anrou, Gunasekaran, Kannan, Moyer, Bryan D, Doherty, Liz, Miranda, Les P
Published in ACS chemical biology (15.09.2017)
Published in ACS chemical biology (15.09.2017)
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Journal Article
Discovery of Melanocortin Ligands via a Double Simultaneous Substitution Strategy Based on the Ac-His- d Phe-Arg-Trp-NH 2 Template
Todorovic, Aleksandar, Lensing, Cody J., Holder, Jerry Ryan, Scott, Joseph W., Sorensen, Nicholas B., Haskell-Luevano, Carrie
Published in ACS chemical neuroscience (21.11.2018)
Published in ACS chemical neuroscience (21.11.2018)
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Journal Article
Discovery of Melanocortin Ligands via a Double Simultaneous Substitution Strategy Based on the Ac-His‑dPhe-Arg-Trp-NH2 Template
Todorovic, Aleksandar, Lensing, Cody J, Holder, Jerry Ryan, Scott, Joseph W, Sorensen, Nicholas B, Haskell-Luevano, Carrie
Published in ACS chemical neuroscience (21.11.2018)
Published in ACS chemical neuroscience (21.11.2018)
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Journal Article
Discovery of Melanocortin Ligands via a Double Simultaneous Substitution Strategy Based on the Ac-His-dPhe-Arg-Trp-NH 2 Template
Todorovic, Aleksandar, Lensing, Cody J, Holder, Jerry Ryan, Scott, Joseph W, Sorensen, Nicholas B, Haskell-Luevano, Carrie
Published in ACS chemical neuroscience (21.11.2018)
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Published in ACS chemical neuroscience (21.11.2018)
Journal Article
Engineering Antibody Reactivity for Efficient Derivatization to Generate Na V 1.7 Inhibitory GpTx-1 Peptide-Antibody Conjugates
Biswas, Kaustav, Nixey, Thomas E, Murray, Justin K, Falsey, James R, Yin, Li, Liu, Hantao, Gingras, Jacinthe, Hall, Brian E, Herberich, Brad, Holder, Jerry Ryan, Li, Hongyan, Ligutti, Joseph, Lin, Min-Hwa Jasmine, Liu, Dong, Soriano, Brian D, Soto, Marcus, Tran, Linh, Tegley, Christopher M, Zou, Anrou, Gunasekaran, Kannan, Moyer, Bryan D, Doherty, Liz, Miranda, Les P
Published in ACS chemical biology (15.09.2017)
Published in ACS chemical biology (15.09.2017)
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Journal Article
Identification of Potent, Selective, and Metabolically Stable Peptide Antagonists to the Calcitonin Gene-Related Peptide (CGRP) Receptor
Miranda, Les P, Holder, Jerry Ryan, Shi, Licheng, Bennett, Brian, Aral, Jennifer, Gegg, Colin V, Wright, Marie, Walker, Kenneth, Doellgast, George, Rogers, Rick, Li, Hongyan, Valladares, Violeta, Salyers, Kevin, Johnson, Eileen, Wild, Kenneth
Published in Journal of medicinal chemistry (25.12.2008)
Published in Journal of medicinal chemistry (25.12.2008)
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Journal Article
Peptide and Small Molecules Rescue the Functional Activity and Agonist Potency of Dysfunctional Human Melanocortin-4 Receptor Polymorphisms
Xiang, Zhimin, Pogozheva, Irina D, Sorenson, Nicholas B, Wilczynski, Andrzej M, Holder, Jerry Ryan, Litherland, Sally A, Millard, William J, Mosberg, Henry I, Haskell-Luevano, Carrie
Published in Biochemistry (Easton) (17.07.2007)
Published in Biochemistry (Easton) (17.07.2007)
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Journal Article
Structure-activity relationships of the melanocortin tetrapeptide Ac-His-DPhe-Arg-Trp-NH2 at the mouse melanocortin receptors. Part 3: modifications at the Arg position
HOLDER, Jerry Ryan, ZHIMIN XIANG, BAUZO, Rayna M, HASKELL-LUEVANO, Carrie
Published in Peptides (New York, N.Y. : 1980) (2003)
Published in Peptides (New York, N.Y. : 1980) (2003)
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Journal Article