Rational design of novel, potent piperazinone and imidazolidinone BACE1 inhibitors
Cumming, J.N., Le, T.X., Babu, S., Carroll, C., Chen, X., Favreau, L., Gaspari, P., Guo, T., Hobbs, D.W., Huang, Y., Iserloh, U., Kennedy, M.E., Kuvelkar, R., Li, G., Lowrie, J., McHugh, N.A., Ozgur, L., Pan, J., Parker, E.M., Saionz, K., Stamford, A.W., Strickland, C., Tadesse, D., Voigt, J., Wang, L., Wu, Y., Zhang, L., Zhang, Q.
Published in Bioorganic & medicinal chemistry (01.06.2008)
Published in Bioorganic & medicinal chemistry (01.06.2008)
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The different strategies for designing GPCR and kinase targeted libraries
Lowrie, J F, Delisle, R K, Hobbs, D W, Diller, D J
Published in Combinatorial chemistry & high throughput screening (01.08.2004)
Published in Combinatorial chemistry & high throughput screening (01.08.2004)
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Synthesis and anti-herpes virus activity of acyclic 2'-deoxyguanosine analogs related to 9-[(1,3-dihydroxy-2-propoxy)methyl]guanine
Martin, John C, McGee, Danny P. C, Jeffrey, Gary A, Hobbs, Doug W, Smee, Donald F, Matthews, Thomas R, Verheyden, Julian P. H
Published in Journal of medicinal chemistry (01.08.1986)
Published in Journal of medicinal chemistry (01.08.1986)
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Development of Orally Active Oxytocin Antagonists: Studies on 1-(1-{4-[1-(2-Methyl-1-oxidopyridin-3-ylmethyl)piperidin-4-yloxy]-2- methoxybenzoyl}piperidin-4-yl)-1,4-dihydrobenz[d][1,3]oxazin-2-one (L-372,662) and Related Pyridines
Bell, Ian M, Erb, Jill M, Freidinger, Roger M, Gallicchio, Steven N, Guare, James P, Guidotti, Maribeth T, Halpin, Rita A, Hobbs, Doug W, Homnick, Carl F, Kuo, Michelle S, Lis, Edward V, Mathre, David J, Michelson, Stuart R, Pawluczyk, Joseph M, Pettibone, Douglas J, Reiss, Duane R, Vickers, Stanley, Williams, Peter D, Woyden, Carla J
Published in Journal of medicinal chemistry (04.06.1998)
Published in Journal of medicinal chemistry (04.06.1998)
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Orally active, nonpeptide oxytocin antagonists
Evans, Ben E, Leighton, James L, Rittle, Kenneth E, Gilbert, Kevin F, Lundell, George F, Gould, Norman P, Hobbs, Doug W, DiPardo, Robert M, Veber, Daniel F, Pettibone, Douglas J, Clineschmidt, Bradley V, Anderson, Paul S, Freidinger, Roger M
Published in Journal of medicinal chemistry (01.10.1992)
Published in Journal of medicinal chemistry (01.10.1992)
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Recommendations for rescue of a submerged unresponsive compressed-gas diver
Mitchell, S J, Bennett, M H, Bird, N, Doolette, D J, Hobbs, G W, Kay, E, Moon, R E, Neuman, T S, Vann, R D, Walker, R, Wyatt, H A
Published in Undersea & hyperbaric medicine (01.11.2012)
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Published in Undersea & hyperbaric medicine (01.11.2012)
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Erratum to “Rational design of novel, potent piperazinone and imidazolidinone BACE1 inhibitors” [Bioorg. Med. Chem. Lett. 18 (2008) 3236–3241]
Cumming, J.N., Le, T.X., Babu, S., Carroll, C., Chen, X., Favreau, L., Gaspari, P., Guo, T., Hobbs, D.W., Huang, Y., Iserloh, U., Kennedy, M.E., Kuvelkar, R., Li, G., Lowrie, J., McHugh, N.A., Ozgur, L., Pan, J., Parker, E.M., Saionz, K., Stamford, A.W., Strickland, C., Tadesse, D., Voigt, J., Wang, L., Wu, Y., Zhang, L., Zhang, Q.
Published in Bioorganic & medicinal chemistry letters (01.08.2008)
Published in Bioorganic & medicinal chemistry letters (01.08.2008)
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