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Published in Bioorganic & medicinal chemistry letters (01.08.2009)
Published in Bioorganic & medicinal chemistry letters (01.08.2009)
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Rhodium-Catalyzed Silylcarbocyclization (SiCaC) and Carbonylative Silylcarbocyclization (CO−SiCaC) Reactions of Enynes
Ojima, Iwao, Vu, An T, Lee, Seung-Yub, McCullagh, James V, Moralee, Andrew C, Fujiwara, Masaki, Hoang, Tram H
Published in Journal of the American Chemical Society (07.08.2002)
Published in Journal of the American Chemical Society (07.08.2002)
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Discovery of GSK2798745: A Clinical Candidate for Inhibition of Transient Receptor Potential Vanilloid 4 (TRPV4)
Brooks, Carl A, Barton, Linda S, Behm, David J, Eidam, Hilary S, Fox, Ryan M, Hammond, Marlys, Hoang, Tram H, Holt, Dennis A, Hilfiker, Mark A, Lawhorn, Brian G, Patterson, Jaclyn R, Stoy, Patrick, Roethke, Theresa J, Ye, Guosen, Zhao, Steve, Thorneloe, Kevin S, Goodman, Krista B, Cheung, Mui
Published in ACS medicinal chemistry letters (08.08.2019)
Published in ACS medicinal chemistry letters (08.08.2019)
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Optimization of a Novel Series of TRPV4 Antagonists with In Vivo Activity in a Model of Pulmonary Edema
Hilfiker, Mark A, Hoang, Tram H, Cornil, Johan, Eidam, Hilary S, Matasic, Daniel S, Roethke, Theresa J, Klein, Michael, Thorneloe, Kevin S, Cheung, Mui
Published in ACS medicinal chemistry letters (14.02.2013)
Published in ACS medicinal chemistry letters (14.02.2013)
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Synthesis and SAR of potent LXR agonists containing an indole pharmacophore
Washburn, David G., Hoang, Tram H., Campobasso, Nino, Smallwood, Angela, Parks, Derek J., Webb, Christine L., Frank, Kelly A., Nord, Melanie, Duraiswami, Chaya, Evans, Christopher, Jaye, Michael, Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
Published in Bioorganic & medicinal chemistry letters (15.02.2009)
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Rational design of orally-active, pyrrolidine-based progesterone receptor partial agonists
Thompson, Scott K., Washburn, David G., Frazee, James S., Madauss, Kevin P., Hoang, Tram H., Lapinski, Leahann, Grygielko, Eugene T., Glace, Lindsay E., Trizna, Walter, Williams, Shawn P., Duraiswami, Chaya, Bray, Jeffrey D., Laping, Nicholas J.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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Synthesis and SAR of amino acid-derived heterocyclic progesterone receptor full and partial agonists
Hammond, Marlys, Patterson, Jaclyn R., Manns, Sharada, Hoang, Tram H., Washburn, David G., Trizna, Walter, Glace, Lindsay, Grygielko, Eugene T., Nagilla, Rakesh, Nord, Melanie, Fries, Harvey E., Minick, Douglas J., Laping, Nicholas J., Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
Published in Bioorganic & medicinal chemistry letters (15.05.2009)
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Journal Article
Improving the developability profile of pyrrolidine progesterone receptor partial agonists
Kallander, Lara S., Washburn, David G., Hoang, Tram H., Frazee, James S., Stoy, Patrick, Johnson, Latisha, Lu, Qing, Hammond, Marlys, Barton, Linda S., Patterson, Jaclyn R., Azzarano, Leonard M., Nagilla, Rakesh, Madauss, Kevin P., Williams, Shawn P., Stewart, Eugene L., Duraiswami, Chaya, Grygielko, Eugene T., Xu, Xiaoping, Laping, Nicholas J., Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
Published in Bioorganic & medicinal chemistry letters (01.01.2010)
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Discovery of orally active, pyrrolidinone-based progesterone receptor partial agonists
Washburn, David G., Hoang, Tram H., Frazee, James S., Johnson, Latisha, Hammond, Marlys, Manns, Sharada, Madauss, Kevin P., Williams, Shawn P., Duraiswami, Chaya, Tran, Thuy B., Stewart, Eugene L., Grygielko, Eugene T., Glace, Lindsay E., Trizna, Walter, Nagilla, Rakesh, Bray, Jeffrey D., Thompson, Scott K.
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
Published in Bioorganic & medicinal chemistry letters (15.08.2009)
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NAV1.8 억제제로서의 2,3-디히드로퀴나졸린 화합물
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Year of Publication 10.03.2022
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Year of Publication 10.03.2022
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HYDROXY FORMAMIDE DERIVATIVES AND THEIR USE
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Year of Publication 12.09.2016
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Year of Publication 12.09.2016
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TRPV4 ANTAGONISTS
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Year of Publication 04.04.2014
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Year of Publication 04.04.2014
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Nitrogen Containing 2,3-Dihydroquinazolinone Compounds as Nav1.8 Inhibitors
ELBAN, Mark Andrew, DONG, Xiaoyang, HOANG, Tram H, GUANG, Jie, HO, Ming-Hsun, ROMANO, Joseph J, WASHBURN, David Glenn
Year of Publication 14.03.2024
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Year of Publication 14.03.2024
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2,3-dihydroquinazolin compounds as NAV1.8 inhibitors
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Year of Publication 14.12.2023
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Year of Publication 14.12.2023
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NITROGEN CONTAINING 2,3-DIHYDROQUINAZOLINONE COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN, Mark Andrew, DONG, Xiaoyang, HOANG, Tram H, GUANG, Jie, HO, Ming-Hsun, ROMANO, Joseph J, WASHBURN, David Glenn
Year of Publication 25.10.2023
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Year of Publication 25.10.2023
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Compuestos 2,3-dihidroquinazolin como inhibidores nav1 .8
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Year of Publication 21.04.2023
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Year of Publication 21.04.2023
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN, Mark, HOANG, Tram H, MILLER, William H, VIMAL, Mythily, WASHBURN, David G, GUANG, Jie, YING, Maben, DAVIS, Roderick S, HO, Ming-Hsun, ROMANO, Joseph J
Year of Publication 06.04.2023
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Year of Publication 06.04.2023
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NITROGEN CONTAINING 2,3-DIHYDROQUINAZOLINONE COMPOUNDS AS NAV1.8 INHIBITORS
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Year of Publication 23.06.2022
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Year of Publication 23.06.2022
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NITROGEN CONTAINING 2,3-DIHYDROQUINAZOLINONE COMPOUNDS AS NAV1.8 INHIBITORS
ELBAN, Mark Andrew, DONG, Xiaoyang, HOANG, Tram H, GUANG, Jie, HO, Ming-Hsun, ROMANO, Joseph J, WASHBURN, David Glenn
Year of Publication 23.06.2022
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Year of Publication 23.06.2022
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2,3-DIHYDROQUINAZOLIN COMPOUNDS AS NAV1.8 INHIBITORS
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Year of Publication 04.05.2022
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Year of Publication 04.05.2022
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