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Brain Penetrable Inhibitors of Ceramide Galactosyltransferase for the Treatment of Lysosomal Storage Disorders
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Implications of Promiscuous Pim-1 Kinase Fragment Inhibitor Hydrophobic Interactions for Fragment-Based Drug Design
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Trypanocidal Activity of 8-Methyl-5′-{[(Z)-4-Aminobut-2-enyl]-(Methylamino)}Adenosine (Genz-644131), an Adenosylmethionine Decarboxylase Inhibitor
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Novel S-Adenosylmethionine Decarboxylase Inhibitors for the Treatment of Human African Trypanosomiasis
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Published in Bioorganic & medicinal chemistry letters (15.04.2005)
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Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 1. N-Cyanoguanidine Bioisosteres Possessing in Vivo Bladder Selectivity
Butera, John A, Antane, Madelene M, Antane, Schuyler A, Argentieri, Thomas M, Freeden, Chris, Graceffa, Russell F, Hirth, Bradford H, Jenkins, Douglas, Lennox, Joseph R, Matelan, Edward, Norton, N. Wesley, Quagliato, Dominick, Sheldon, Jeffrey H, Spinelli, Walter, Warga, Dawn, Wojdan, Alexandra, Woods, Morgan
Published in Journal of medicinal chemistry (23.03.2000)
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Design and SAR of Novel Potassium Channel Openers Targeted for Urge Urinary Incontinence. 2. Selective and Potent Benzylamino Cyclobutenediones
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Published in Journal of medicinal chemistry (23.03.2000)
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Synthesis and potassium channel opening activity of substituted 10H-Benzofuro[3,2-b]indole- and 5,10-Dihydro-indeno[1,2-b]indole-1-carboxylic acids
Butera, John A., Antane, Schuyler A., Hirth, Bradford, Lennox, Joseph R., Sheldon, Jeffrey H., Norton, N.Wesley, Warga, Dawn, Argentieri, Thomas M.
Published in Bioorganic & medicinal chemistry letters (01.08.2001)
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Year of Publication 30.05.2024
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Year of Publication 30.05.2024
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Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Published in Bioorganic & medicinal chemistry letters (01.08.2010)
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Restricted Nitrogen Inversion in 9,10- Diazatetracyclo[6.3.0.0.4,110.5,9]undecanes. Dynamic NMR Studies
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Published in Journal of organic chemistry (29.05.1998)
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Discovery of novel sphingosine kinase 1 inhibitors
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Published in Bioorganic & medicinal chemistry letters (01.11.2009)
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Hirth, Bradford, Barker, Robert H., Celatka, Cassandra A., Klinger, Jeffrey D., Liu, Hanlan, Nare, Bakela, Nijjar, Amarjit, Phillips, Margaret A., Sybertz, Edmund, Willert, Erin K., Xiang, Yibin
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Discovery of novel sphingosine kinase-t inhibitors. Part 2
YIBIN XIANG, HIRTH, Bradford, KANE, John L, JUNKAI LIAO, NOSON, Kevin D, YEE, Christopher, ASMUSSEN, Gary, FITZGERALD, Maria, KLAUS, Christine, BOOKER, Michael
Published in Bioorganic & medicinal chemistry letters (2010)
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ZHAO ZHONG, GOOD ANDREW, SKERLJ RENATO, XIANG YIBIN, CHENG SENG, METZ MARKUS, SCHEULE RONALD, CELATKA CASSANDRA, JANCISICS KATHERINE, MARSHALL JOHN, CABRERA SALAZAR MARIO, HIRTH BRADFORD, BOURQUE ELYSE
Year of Publication 23.07.2014
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Year of Publication 23.07.2014
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