A Nonpeptide Oxytocin Receptor Agonist for a Durable Relief of Inflammatory Pain
Hilfiger, Louis, Zhao, Qian, Kerspern, Damien, Inquimbert, Perrine, Andry, Virginie, Goumon, Yannick, Darbon, Pascal, Hibert, Marcel, Charlet, Alexandre
Published in Scientific reports (20.02.2020)
Published in Scientific reports (20.02.2020)
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Neutralization of CXCL12 attenuates established pulmonary hypertension in rats
Bordenave, Jennifer, Thuillet, Raphaël, Tu, Ly, Phan, Carole, Cumont, Amélie, Marsol, Claire, Huertas, Alice, Savale, Laurent, Hibert, Marcel, Galzi, Jean-Luc, Bonnet, Dominique, Humbert, Marc, Frossard, Nelly, Guignabert, Christophe
Published in Cardiovascular research (01.03.2020)
Published in Cardiovascular research (01.03.2020)
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Journal Article
Development of original metabolically stable apelin-17 analogs with diuretic and cardiovascular effects
Gerbier, Romain, Alvear-Perez, Rodrigo, Margathe, Jean-Francois, Flahault, Adrien, Couvineau, Pierre, Gao, Ji, De Mota, Nadia, Dabire, Hubert, Li, Bo, Ceraudo, Emilie, Hus-Citharel, Annette, Esteoulle, Lucie, Bisoo, Cynthia, Hibert, Marcel, Berdeaux, Alain, Iturrioz, Xavier, Bonnet, Dominique, Llorens-Cortes, Catherine
Published in The FASEB journal (01.02.2017)
Published in The FASEB journal (01.02.2017)
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Journal Article
Effects of oxytocin receptor agonism on acquisition and expression of pair bonding in male prairie voles
Johnson, Michael C, Zweig, Jonathan A, Zhang, Yangmiao, Nunez, Louis, Ryabinina, Olga P, Hibert, Marcel, Ryabinin, Andrey E
Published in Translational psychiatry (15.07.2024)
Published in Translational psychiatry (15.07.2024)
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Journal Article
Protein-based virtual screening of chemical databases. II. Are homology models of g-protein coupled receptors suitable targets?
Bissantz, Caterina, Bernard, Philippe, Hibert, Marcel, Rognan, Didier
Published in Proteins, structure, function, and bioinformatics (01.01.2003)
Published in Proteins, structure, function, and bioinformatics (01.01.2003)
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Journal Article
Red Fluorescent Turn-On Ligands for Imaging and Quantifying G Protein-Coupled Receptors in Living Cells
Karpenko, Iuliia A., Kreder, Rémy, Valencia, Christel, Villa, Pascal, Mendre, Christiane, Mouillac, Bernard, Mély, Yves, Hibert, Marcel, Bonnet, Dominique, Klymchenko, Andrey S.
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
Published in Chembiochem : a European journal of chemical biology (10.02.2014)
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Journal Article
Biased Agonist Pharmacochaperones of the AVP V2 Receptor May Treat Congenital Nephrogenic Diabetes Insipidus
JEAN-ALPHONSE, Frédéric, PERKOVSKA, Sanja, MENDRE, Christiane, FRANTZ, Marie-Céline, DURROUX, Thierry, MEJEAN, Catherine, MORIN, Denis, LOISON, Stéphanie, BONNET, Dominique, HIBERT, Marcel, MOUILLAC, Bernard
Published in Journal of the American Society of Nephrology (01.10.2009)
Published in Journal of the American Society of Nephrology (01.10.2009)
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Chemical Library Screening and Structure-Function Relationship Studies Identify Bisacodyl as a Potent and Selective Cytotoxic Agent Towards Quiescent Human Glioblastoma Tumor Stem-Like Cells
Zeniou, Maria, Fève, Marie, Mameri, Samir, Dong, Jihu, Salomé, Christophe, Chen, Wanyin, El-Habr, Elias A, Bousson, Fanny, Sy, Mohamadou, Obszynski, Julie, Boh, Alexandre, Villa, Pascal, Assad Kahn, Suzana, Didier, Bruno, Bagnard, Dominique, Junier, Marie-Pierre, Chneiweiss, Hervé, Haiech, Jacques, Hibert, Marcel, Kilhoffer, Marie-Claude
Published in PloS one (13.08.2015)
Published in PloS one (13.08.2015)
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Journal Article
Quantitative Structure–Property Relationship Modeling: A Valuable Support in High-Throughput Screening Quality Control
Ruggiu, Fiorella, Gizzi, Patrick, Galzi, Jean-Luc, Hibert, Marcel, Haiech, Jacques, Baskin, Igor, Horvath, Dragos, Marcou, Gilles, Varnek, Alexandre
Published in Analytical chemistry (Washington) (04.03.2014)
Published in Analytical chemistry (Washington) (04.03.2014)
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Journal Article
Fluorescent Derivatives of AC-42 To Probe Bitopic Orthosteric/Allosteric Binding Mechanisms on Muscarinic M1 Receptors
Daval, Sandrine B, Valant, Céline, Bonnet, Dominique, Kellenberger, Esther, Hibert, Marcel, Galzi, Jean-Luc, Ilien, Brigitte
Published in Journal of medicinal chemistry (08.03.2012)
Published in Journal of medicinal chemistry (08.03.2012)
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Journal Article
Small Neutralizing Molecules to Inhibit Actions of the Chemokine CXCL12
Hachet-Haas, Muriel, Balabanian, Karl, Rohmer, François, Pons, Françoise, Franchet, Christel, Lecat, Sandra, Chow, Ken Y.C., Dagher, Rania, Gizzi, Patrick, Didier, Bruno, Lagane, Bernard, Kellenberger, Esther, Bonnet, Dominique, Baleux, Françoise, Haiech, Jacques, Parmentier, Marc, Frossard, Nelly, Arenzana-Seisdedos, Fernando, Hibert, Marcel, Galzi, Jean-luc
Published in The Journal of biological chemistry (22.08.2008)
Published in The Journal of biological chemistry (22.08.2008)
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Identification by high throughput screening of small compounds inhibiting the nucleic acid destabilization activity of the HIV-1 nucleocapsid protein
Shvadchak, Volodymyr, Sanglier, Sarah, Rocle, Sandrine, Villa, Pascal, Haiech, Jacques, Hibert, Marcel, Van Dorsselaer, Alain, Mély, Yves, de Rocquigny, Hugues
Published in Biochimie (01.07.2009)
Published in Biochimie (01.07.2009)
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Journal Article
Versatile Synthetic Approach for Selective Diversification of Bicyclic Aza-Diketopiperazines
Péron, Florent, Riché, Stéphanie, Lesur, Brigitte, Hibert, Marcel, Breton, Philippe, Fourquez, Jean-Marie, Girard, Nicolas, Bonnet, Dominique
Published in ACS omega (30.11.2018)
Published in ACS omega (30.11.2018)
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Journal Article
Homodimerization of the death-associated protein kinase catalytic domain: development of a new small molecule fluorescent reporter
Zimmermann, Michael, Atmanene, Cédric, Xu, Qingyan, Fouillen, Laetitia, Van Dorsselaer, Alain, Bonnet, Dominique, Marsol, Claire, Hibert, Marcel, Sanglier-Cianferani, Sarah, Pigault, Claire, McNamara, Laurie K, Watterson, D Martin, Haiech, Jacques, Kilhoffer, Marie-Claude
Published in PloS one (30.11.2010)
Published in PloS one (30.11.2010)
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Identification of the Binding Sites of the SR49059 Nonpeptide Antagonist into the V1a Vasopressin Receptor Using Sulfydryl-reactive Ligands and Cysteine Mutants as Chemical Sensors
Tahtaoui, Chouaïb, Balestre, Marie-Noëlle, Klotz, Philippe, Rognan, Didier, Barberis, Claude, Mouillac, Bernard, Hibert, Marcel
Published in The Journal of biological chemistry (10.10.2003)
Published in The Journal of biological chemistry (10.10.2003)
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Journal Article
Fluorescence resonance energy transfer to probe human M1 muscarinic receptor structure and drug binding properties
Ilien, Brigitte, Franchet, Christelle, Bernard, Philippe, Morisset, Séverine, Odile Weill, Claire, Bourguignon, Jean‐Jacques, Hibert, Marcel, Galzi, Jean‐Luc
Published in Journal of neurochemistry (01.05.2003)
Published in Journal of neurochemistry (01.05.2003)
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Journal Article
Limitations in a frataxin knockdown cell model for Friedreich ataxia in a high-throughput drug screen
Calmels, Nadège, Seznec, Hervé, Villa, Pascal, Reutenauer, Laurence, Hibert, Marcel, Haiech, Jacques, Rustin, Pierre, Koenig, Michel, Puccio, Hélène
Published in BMC neurology (24.08.2009)
Published in BMC neurology (24.08.2009)
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