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Site-directed mutagenesis of the putative human muscarinic M2 receptor binding site
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Acute, chronic and conditioned effects of intranasal oxytocin in the mu-opioid receptor knockout mouse model of autism: Social context matters
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Cyclo-release synthesis of cyclic disulfides on solid phase
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Published in Tetrahedron letters (16.12.2000)
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Fluorogenic Squaraine Dimers with Polarity-Sensitive Folding As Bright Far-Red Probes for Background-Free Bioimaging
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LIT-001, the First Nonpeptide Oxytocin Receptor Agonist that Improves Social Interaction in a Mouse Model of Autism
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Discovery of a Locally and Orally Active CXCL12 Neutraligand (LIT-927) with Anti-inflammatory Effect in a Murine Model of Allergic Airway Hypereosinophilia
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Published in Journal of medicinal chemistry (13.09.2018)
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Published in Journal of organic chemistry (2017)
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Published in Journal of medicinal chemistry (01.06.1988)
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Comparative Study of the Synthesis and Structural and Physicochemical Properties of Diketopiperazines vs Aza-diketopiperazines
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Published in Journal of organic chemistry (17.03.2017)
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A step-economical multicomponent synthesis of 3D-shaped aza-diketopiperazines and their drug-like chemical space analysisElectronic supplementary information (ESI) available: Detailed experimental procedures and analytical data for all the compounds. See DOI: 10.1039/c6ob01434h
Regenass, Pierre, Riché, Stéphanie, Péron, Florent, Rognan, Didier, Hibert, Marcel, Girard, Nicolas, Bonnet, Dominique
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An Antedrug of the CXCL12 Neutraligand Blocks Experimental Allergic Asthma without Systemic Effect in Mice
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Published in The Journal of biological chemistry (26.04.2013)
Published in The Journal of biological chemistry (26.04.2013)
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Selective Fluorescent Nonpeptidic Antagonists For Vasopressin V2 GPCR: Application To Ligand Screening and Oligomerization Assays
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Convenient Method To Access New 4,4-Dialkoxy- and 4,4-Diaryloxy-diaza-s-indacene Dyes: Synthesis and Spectroscopic Evaluation
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Published in Journal of organic chemistry (05.01.2007)
Published in Journal of organic chemistry (05.01.2007)
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