Mitochondrial complex I inhibition triggers a mitophagy-dependent ROS increase leading to necroptosis and ferroptosis in melanoma cells
Basit, Farhan, van Oppen, Lisanne Mpe, Schöckel, Laura, Bossenbroek, Hasse M, van Emst-de Vries, Sjenet E, Hermeling, Johannes Cw, Grefte, Sander, Kopitz, Charlotte, Heroult, Melanie, Hgm Willems, Peter, Koopman, Werner Jh
Published in Cell death & disease (30.03.2017)
Published in Cell death & disease (30.03.2017)
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The Wnt signaling regulator R-spondin 3 promotes angioblast and vascular development
Kazanskaya, Olga, Ohkawara, Bisei, Heroult, Melanie, Wu, Wei, Maltry, Nicole, Augustin, Hellmut G, Niehrs, Christof
Published in Development (Cambridge) (15.11.2008)
Published in Development (Cambridge) (15.11.2008)
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Discovery of VIP236, an αvβ3-Targeted Small-Molecule–Drug Conjugate with Neutrophil Elastase-Mediated Activation of 7-Ethyl Camptothecin Payload for Treatment of Solid Tumors
Lerchen, Hans-Georg, Stelte-Ludwig, Beatrix, Heroult, Melanie, Zubov, Dmitry, Gericke, Kersten Matthias, Wong, Harvey, Frigault, Melanie M, Johnson, Amy J, Izumi, Raquel, Hamdy, Ahmed
Published in Cancers (01.09.2023)
Published in Cancers (01.09.2023)
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A Small Molecule–Drug Conjugate (SMDC) Consisting of a Modified Camptothecin Payload Linked to an αVß3 Binder for the Treatment of Multiple Cancer Types
Lerchen, Hans-Georg, Stelte-Ludwig, Beatrix, Kopitz, Charlotte, Heroult, Melanie, Zubov, Dmitry, Willuda, Joerg, Schlange, Thomas, Kahnert, Antje, Wong, Harvey, Izumi, Raquel, Hamdy, Ahmed
Published in Cancers (13.01.2022)
Published in Cancers (13.01.2022)
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Journal Article
Differential Endothelial Transcriptomics Identifies Semaphorin 3G as a Vascular Class 3 Semaphorin
Kutschera, Simone, Weber, Holger, Weick, Anja, De Smet, Frederik, Genove, Guillem, Takemoto, Minoru, Prahst, Claudia, Riedel, Maria, Mikelis, Constantinos, Baulande, Sylvain, Champseix, Catherine, Kummerer, Petra, Conseiller, Emmanuel, Multon, Marie-Christine, Heroult, Melanie, Bicknell, Roy, Carmeliet, Peter, Betsholtz, Christer, Augustin, Hellmut G
Published in Arteriosclerosis, thrombosis, and vascular biology (01.01.2011)
Published in Arteriosclerosis, thrombosis, and vascular biology (01.01.2011)
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Inhibition of the mitogenic, angiogenic and tumorigenic activities of pleiotrophin by a synthetic peptide corresponding to its C-thrombospondin repeat-I domain
Hamma-Kourbali, Yamina, Bernard-Pierrot, Isabelle, Heroult, Mélanie, Dalle, Sophie, Caruelle, Danièle, Milhiet, Pierre Emmanuel, Fernig, David G., Delbé, Jean, Courty, José
Published in Journal of cellular physiology (01.01.2008)
Published in Journal of cellular physiology (01.01.2008)
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Collagen Triple Helix Repeat Containing 1, a Novel Secreted Protein in Injured and Diseased Arteries, Inhibits Collagen Expression and Promotes Cell Migration
Pyagay, Peter, Heroult, Mélanie, Wang, Qiaozeng, Lehnert, Wolfgang, Belden, John, Liaw, Lucy, Friesel, Robert E, Lindner, Volkhard
Published in Circulation research (04.02.2005)
Published in Circulation research (04.02.2005)
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Abstract 1314: A novel small molecule drug conjugate -avb3 integrin antagonist linked to a cytotoxic camptothecin derivative- for the treatment of multiple cancer types
Lerchen, Hans-Georg, Stelte-Ludwig, Beatrix, Kopitz, Charlotte, Heroult, Melanie, Zubov, Dmitry, Willuda, Joerg, Schlange, Thomas, Kahnert, Antje, Izumi, Raquel, Hamdy, Ahmed
Published in Cancer research (Chicago, Ill.) (01.07.2021)
Published in Cancer research (Chicago, Ill.) (01.07.2021)
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Journal Article
A Small Molecule-Drug Conjugate (SMDC) Consisting of a Modified Camptothecin Payload Linked to an α V ß 3 Binder for the Treatment of Multiple Cancer Types
Lerchen, Hans-Georg, Stelte-Ludwig, Beatrix, Kopitz, Charlotte, Heroult, Melanie, Zubov, Dmitry, Willuda, Joerg, Schlange, Thomas, Kahnert, Antje, Wong, Harvey, Izumi, Raquel, Hamdy, Ahmed
Published in Cancers (13.01.2022)
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Published in Cancers (13.01.2022)
Journal Article
Rogaratinib: A potent and selective pan‐FGFR inhibitor with broad antitumor activity in FGFR‐overexpressing preclinical cancer models
Grünewald, Sylvia, Politz, Oliver, Bender, Sebastian, Héroult, Mélanie, Lustig, Klemens, Thuss, Uwe, Kneip, Christoph, Kopitz, Charlotte, Zopf, Dieter, Collin, Marie‐Pierre, Boemer, Ulf, Ince, Stuart, Ellinghaus, Peter, Mumberg, Dominik, Hess‐Stumpp, Holger, Ziegelbauer, Karl
Published in International journal of cancer (01.09.2019)
Published in International journal of cancer (01.09.2019)
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Abstract 4703: The BET inhibitor BAY 1238097 shows efficacy in BRAF wild-type and mutant melanoma models
Haendler, Bernard, Gelato, Kathy A., Schöckel, Laura, Sugawara, Tatsuo, Lejeune, Pascale, Ellinger-Ziegelbauer, Heidrun, Fernandez-Montalvan, Amaury E., Holton, Simon, Siegel, Stephan, Heroult, Melanie, Walter, Annette, Ince, Stuart, Ocker, Matthias
Published in Cancer research (Chicago, Ill.) (15.07.2016)
Published in Cancer research (Chicago, Ill.) (15.07.2016)
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A CD44v6 peptide reveals a role of CD44 in VEGFR-2 signaling and angiogenesis
Tremmel, Martina, Matzke, Alexandra, Albrecht, Imke, Laib, Anna M., Olaku, Vivienne, Ballmer-Hofer, Kurt, Christofori, Gerhard, Héroult, Mélanie, Augustin, Hellmut G., Ponta, Helmut, Orian-Rousseau, Véronique
Published in Blood (10.12.2009)
Published in Blood (10.12.2009)
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Targeting mitochondrial complex I using BAY 87-2243 reduces melanoma tumor growth
Schöckel, Laura, Glasauer, Andrea, Basit, Farhan, Bitschar, Katharina, Truong, Hoa, Erdmann, Gerrit, Algire, Carolyn, Hägebarth, Andrea, Willems, Peter Hgm, Kopitz, Charlotte, Koopman, Werner Jh, Héroult, Mélanie
Published in Cancer & metabolism (20.10.2015)
Published in Cancer & metabolism (20.10.2015)
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Journal Article
Neuropilin-1-VEGFR-2 Complexing Requires the PDZ-binding Domain of Neuropilin-1
Prahst, Claudia, Héroult, Mélanie, Lanahan, Anthony A., Uziel, Noa, Kessler, Ofra, Shraga-Heled, Niva, Simons, Michael, Neufeld, Gera, Augustin, Hellmut G.
Published in The Journal of biological chemistry (12.09.2008)
Published in The Journal of biological chemistry (12.09.2008)
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Abstract 1739: Preclinical profile of BAY 1163877 - a selective pan-FGFR inhibitor in phase 1 clinical trial
Heroult, Melanie, Ellinghaus, Peter, Sieg, Christian, Brohm, Dirk, Gruenewald, Sylvia, Collin, Marie-Pierre, Boemer, Ulf, Lobell, Mario, Huebsch, Walter, Ocker, Matthias, Ince, Stuart, Haegebarth, Andrea, Jautelat, Rolf, Hess-Stumpp, Holger, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Abstract 1442: Effects of selective and broad glucose transporter (GLUT) inhibition on glucose distribution in tumor bearing mice
Heroult, Melanie, Steinke, Wolfram, Frisk, Anna-Lena, Borkowski, Sandra, Meyer, Kirstin, Petrul, Heike, Heisler, Iring, Quanz, Maria, Neuhaus, Roland, Buchmann, Bernd, Mueller, Thomas, Bauser, Marcus, Haegebarth, Andrea, Brands, Michael, Ziegelbauer, Karl
Published in Cancer research (Chicago, Ill.) (01.10.2014)
Published in Cancer research (Chicago, Ill.) (01.10.2014)
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Neuropilin-1 mediates vascular permeability independently of vascular endothelial growth factor receptor-2 activation
Roth, Lise, Prahst, Claudia, Ruckdeschel, Tina, Savant, Soniya, Weström, Simone, Fantin, Alessandro, Riedel, Maria, Héroult, Mélanie, Ruhrberg, Christiana, Augustin, Hellmut G
Published in Science signaling (26.04.2016)
Published in Science signaling (26.04.2016)
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Expression of the growth factor pleiotrophin and its receptor protein tyrosine phosphatase beta/zeta in the serum, cartilage and subchondral bone of patients with osteoarthritis
Kaspiris, Angelos, Mikelis, Constantinos, Heroult, Melanie, Khaldi, Lubna, Grivas, Theodoros B, Kouvaras, Ioannis, Dangas, Spyridon, Vasiliadis, Elias, Lioté, Frédéric, Courty, José, Papadimitriou, Evangelia
Published in Joint, bone, spine : revue du rhumatisme (01.07.2013)
Published in Joint, bone, spine : revue du rhumatisme (01.07.2013)
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Journal Article
Discovery of Rogaratinib (BAY 1163877): a pan‐FGFR Inhibitor
Collin, Marie‐Pierre, Lobell, Mario, Hübsch, Walter, Brohm, Dirk, Schirok, Hartmut, Jautelat, Rolf, Lustig, Klemens, Bömer, Ulf, Vöhringer, Verena, Héroult, Mélanie, Grünewald, Sylvia, Hess‐Stumpp, Holger
Published in ChemMedChem (06.03.2018)
Published in ChemMedChem (06.03.2018)
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