2‑Aryl-5-carboxytetrazole as a New Photoaffinity Label for Drug Target Identification
Herner, András, Marjanovic, Jasmina, Lewandowski, Tracey M, Marin, Violeta, Patterson, Melanie, Miesbauer, Laura, Ready, Damien, Williams, Jon, Vasudevan, Anil, Lin, Qing
Published in Journal of the American Chemical Society (09.11.2016)
Published in Journal of the American Chemical Society (09.11.2016)
Get full text
Journal Article
A new family of bioorthogonally applicable fluorogenic labels
Herner, Andras, Nikic, Ivana, Kallay, Mihaly, Lemke, Edward A., Kele, Peter
Published in Organic & biomolecular chemistry (28.05.2013)
Published in Organic & biomolecular chemistry (28.05.2013)
Get full text
Journal Article
Bioorthogonal fluorescent labels: a review on combined forces
Cserép, Gergely B, Herner, András, Kele, Péter
Published in Methods and applications in fluorescence (08.09.2015)
Published in Methods and applications in fluorescence (08.09.2015)
Get full text
Journal Article
Clickable fluorophores for biological labeling-with or without copper
Kele, Peter, Li, Xiaohua, Link, Martin, Nagy, Krisztina, Herner, Andras, Lorincz, Krisztian, Beni, Szabolcs, Wolfbeis, Otto S.
Published in Organic & biomolecular chemistry (01.01.2009)
Published in Organic & biomolecular chemistry (01.01.2009)
Get full text
Journal Article
Tyrosine specific sequential labeling of proteins
Cserép, Gergely B., Herner, András, Wolfbeis, Otto S., Kele, Péter
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
Get full text
Journal Article
선택적 BCL-XL PROTAC 화합물 및 사용 방법
NAKAJIMA KATSUMASA, NOVAK TIBOR, STARCK JEROME BENOIT, LIU GANG, COLLAND FREDERIC, MARKACZ PIROSKA, KUN VILIBALD, D'ALESSIO JOSEPH ANTHONY, HERNER ANDRAS, THOMAS RANNY MATTHEW, PACZAL ATTILA, SZOKOL BIANKA, FRANZETTI GEORGES ALAIN, ZHAO LIANG, BURGER MATTHEW T, SEISS KATHERINE ELIZABETH, TIMARI MATYAS PAL, DESOS PATRICE
Year of Publication 19.12.2023
Get full text
Year of Publication 19.12.2023
Patent
암을 치료하기 위한 BCL-XL 단백질 억제제 및 아폽토시스 촉진성 제제로서의 6,7-디하이드로-5H-피리도[2,3-C]피리다진 유도체 및 관련 화합물
NOVAK TIBOR, STARCK JEROME BENOIT, COLLAND FREDERIC, HERNER ANDRAS, WEBB PAUL, KOTSCHY ANDRAS, PACZAL ATTILA, SANDERS EMMA, BEDFORD SIMON, DODSWORTH MARK PHILIP, TIMARI MATYAS PAL, CHANRION MAIEA, MARAGNO ANA LETICIA, MURRAY JAMES BROOKE, DAVIDSON JAMES EDWARD PAUL
Year of Publication 31.03.2022
Get full text
Year of Publication 31.03.2022
Patent
3,6-디아미노-피리다진-3-일 유도체, 이를 함유하는 약학적 조성물 및 아폽토시스 유발제로서의 용도
MADARASZ ZOLTAN, NYERGES MIKLOS, NOVAK TIBOR, COLLAND FREDERIC, HERNER ANDRAS, STROFEK AGNES, WEBB PAUL, KOTSCHY ANDRAS, DUNKEL PETRA, PACZAL ATTILA, STARCK JEROMEBENOIT, BEDFORD SIMON, RUDASOVA MONIKA, PARSONS RACHEL JANE, SZIGETI MARIANNA, DODSWORTH MARK PHILIP, TIMARI MATYAS PAL, CHANRION MAIEA, MARAGNO ANA LETICIA, DESOS PATRICE, MURRAY JAMES BROOKE, MOLNAR MARK, DAVIDSON JAMES EDWARD PAUL
Year of Publication 04.04.2022
Get full text
Year of Publication 04.04.2022
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, COLLAND, Frederic, NOVAK, Tibor, KOTSCHY, Andras, DAVIDSON, James Edward Paul, DODSWORTH, Mark Philip, BEDFORD, Simon, HERNER, Andras, CHANRION, Maîa, TIMARI, Matyas Pal, Murray, James Brooke, PACZAL, Attila, STARCK, Jerôme-Benoit, WEBB, Paul
Year of Publication 28.06.2024
Get full text
Year of Publication 28.06.2024
Patent
6,7-DIHYDRO-5H-PYRIDO(2,3-C)PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MURRAY James Brooke, PACZAL Attila, KOTSCHY Andras, STARCK Jerome-Benoit, CHANRION Maia, DODSWORTH Mark Philip, COLLAND Frederic, DAVIDSON James Edward Paul, SANDERS Emma, TIMARI Matyas Pal, HERNER Andras, NOVAK Tibor, BEDFORD Simon, MARAGNO Ana Leticia, WEBB Paul
Year of Publication 30.04.2024
Get full text
Year of Publication 30.04.2024
Patent
A new family of bioorthogonally applicable fluorogenic labelsThis work is dedicated to Roger M. Leblanc on the occasion of his birthday.Electronic supplementary information (ESI) available: 1H- and 13C-NMR spectra for small molecules and fluorescence spectra for 1a-c and 9a-c, further images of live cell labeling experiments and optimized geometries are provided. See DOI: 10.1039/c3ob40296g
Herner, András, Niki, Ivana, Kállay, Mihály, Lemke, Edward A, Kele, Péter
Year of Publication 28.05.2013
Year of Publication 28.05.2013
Get full text
Journal Article
SELECTIVE BCL-XL PROTAC COMPOUNDS AND METHODS OF USE
D'ALESSIO, JOSEPH ANTHONY, MARKACZ, PIROSKA, TIMARI, MATYAS PAL, THOMAS, RANNY MATTHEW, NOVAK, TIBOR, HERNER, ANDRAS, ZHAO, LIANG, COLLAND, FREDERIC, LIU, GANG, PACZAL, ATTILA, SEISS, KATHERINE ELIZABETH, NAKAJIMA, KATSUMASA, BURGER, MATTHEW T, KUN, VILIBALD, SZOKOL, BIANKA, FRANZETTI, GEORGES-ALAIN, STARCK, JEROME-BENOIT, DESOS, PATRICE
Year of Publication 11.08.2022
Get full text
Year of Publication 11.08.2022
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MURRAY, JAMES BROOKE, MARAGNO, ANA LETICIA, TIMARI, MATYAS PAL, NOVAK, TIBOR, HERNER, ANDRAS, DODSWORTH, MARK PHILIP, WEBB, PAUL, SANDERS, EMMA, COLLAND, FREDERIC, BEDFORD, SIMON, PACZAL, ATTILA, CHANRION, MAIA, DAVIDSON, JAMES EDWARD PAUL, STARCK, JEROME-BENOIT, KOTSCHY, ANDRAS
Year of Publication 04.02.2021
Get full text
Year of Publication 04.02.2021
Patent
3,6-DIAMINO-PYRIDAZIN-3-YL DERIVATIVES, PHARMACEUTICAL COMPOSITIONS CONTAINING THEM AND THEIR USES AS PRO-APOPTOTIC AGENTS
PARSONS, RACHEL JANE, MURRAY, JAMES BROOKE, DUNKEL, PETRA, RUDASOVA, MONIKA, MARAGNO, ANA LETICIA, NYERGES, MIKLOS, TIMARI, MATYAS PAL, NOVAK, TIBOR, HERNER, ANDRAS, MADARASZ, ZOLTAN, DODSWORTH, MARK PHILIP, SZIGETI, MARIANNA, WEBB, PAUL, COLLAND, FREDERIC, BEDFORD, SIMON, PACZAL, ATTILA, STROFEK, AGNES, CHANRION, MAIA, DAVIDSON, JAMES EDWARD PAUL, MOLNAR, MARK, STARCK, JEROME-BENOIT, DESOS, PATRICE, KOTSCHY, ANDRAS
Year of Publication 04.02.2021
Get full text
Year of Publication 04.02.2021
Patent
6,7-dihydro-5H-pyrido[2,3-c]pyridazine derivatives and related compounds as Bcl-xL protein inhibitors and pro-apoptotic agents for treating cancer
MURRAY James Brooke, PACZAL Attila, KOTSCHY Andras, STARCK Jerome-Benoit, CHANRION Maia, DODSWORTH Mark Philip, COLLAND Frederic, DAVIDSON James Edward Paul, SANDERS Emma, TIMARI Matyas Pal, HERNER Andras, NOVAK Tibor, BEDFORD Simon, MARAGNO Ana Leticia, WEBB Paul
Year of Publication 30.06.2024
Get full text
Year of Publication 30.06.2024
Patent
DERIVADOS DE 6,7-DIHIDRO-5H-PIRIDO[2,3-C]PIRIDAZIN Y COMPUESTOS RELACIONADOS COMO INHIBIDORES DE PROTEINA BCL-XL Y AGENTES PROAPOPTOTICOS PARA EL TRATAMIENTO DEL CANCER
CHANRION, Maia, MARAGNO, Ana Leticia, SANDERS, Emma, MURRAY, James Brooke, COLLAND, Frederic, NOVAK, Tibor, KOTSCHY, Andras, DAVIDSON, James Edward Paul, DODSWORTH, Mark Philip, BEDFORD, Simon, HERNER, Andras, TIMARI, Matyas Pal, PACZAL, Attila, STARCK, Jerôme-Benoit, WEBB, Paul
Year of Publication 04.05.2022
Get full text
Year of Publication 04.05.2022
Patent