2‑Aryl-5-carboxytetrazole as a New Photoaffinity Label for Drug Target Identification
Herner, András, Marjanovic, Jasmina, Lewandowski, Tracey M, Marin, Violeta, Patterson, Melanie, Miesbauer, Laura, Ready, Damien, Williams, Jon, Vasudevan, Anil, Lin, Qing
Published in Journal of the American Chemical Society (09.11.2016)
Published in Journal of the American Chemical Society (09.11.2016)
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Journal Article
A new family of bioorthogonally applicable fluorogenic labels
Herner, Andras, Nikic, Ivana, Kallay, Mihaly, Lemke, Edward A., Kele, Peter
Published in Organic & biomolecular chemistry (28.05.2013)
Published in Organic & biomolecular chemistry (28.05.2013)
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Journal Article
Bioorthogonal fluorescent labels: a review on combined forces
Cserép, Gergely B, Herner, András, Kele, Péter
Published in Methods and applications in fluorescence (08.09.2015)
Published in Methods and applications in fluorescence (08.09.2015)
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Journal Article
Clickable fluorophores for biological labeling-with or without copper
Kele, Peter, Li, Xiaohua, Link, Martin, Nagy, Krisztina, Herner, Andras, Lorincz, Krisztian, Beni, Szabolcs, Wolfbeis, Otto S.
Published in Organic & biomolecular chemistry (01.01.2009)
Published in Organic & biomolecular chemistry (01.01.2009)
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Journal Article
Tyrosine specific sequential labeling of proteins
Cserép, Gergely B., Herner, András, Wolfbeis, Otto S., Kele, Péter
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
Published in Bioorganic & medicinal chemistry letters (01.11.2013)
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Journal Article
A new family of bioorthogonally applicable fluorogenic labelsThis work is dedicated to Roger M. Leblanc on the occasion of his birthday.Electronic supplementary information (ESI) available: 1H- and 13C-NMR spectra for small molecules and fluorescence spectra for 1a-c and 9a-c, further images of live cell labeling experiments and optimized geometries are provided. See DOI: 10.1039/c3ob40296g
Herner, András, Niki, Ivana, Kállay, Mihály, Lemke, Edward A, Kele, Péter
Year of Publication 28.05.2013
Year of Publication 28.05.2013
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Journal Article
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, PACZAL, Attila, KOTSCHY, András, WEBB, Paul
Year of Publication 28.08.2024
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Year of Publication 28.08.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
Sanders, Emma, Novak, Tibor, Paczal, Attila, Colland, Frédéric, Davidson, James Edward Paul, Kotschy, András, Timári, Mátyás Pál, Chanrion, Maïa, Dodsworth, Mark Philip, Starck, Jérôme-Benoît, Bedford, Simon, Murray, James, Webb, Paul, Herner, András, Maragno, Ana Leticia
Year of Publication 07.06.2024
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Year of Publication 07.06.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
TIMÁRI, MÁTYÁS PÁL, STARCK, JÉRÔME-BENOIT, MURRAY, JAMES BROOKE, HERNER, ANDRÁS, MARAGNO, ANA LETICIA, COLLAND, FRÉDÉRIC, NOVAK, TIBOR, DODSWORTH, MARK PHILIP, WEBB, PAUL, SANDERS, EMMA, BEDFORD, SIMON, PACZAL, ATTILA, CHANRION, MAÏA, KOTSCHY, ANDRÁS, DAVIDSON, JAMES EDWARD PAUL
Year of Publication 29.04.2024
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Year of Publication 29.04.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MURRAY, JAMES, BROOKE, STARCK, JÉRÔME-BENOIT, HERNER, ANDRÁS, COLLAND, FRÉDÉRIC, NOVAK, TIBOR, WEBB, PAUL, SANDERS, EMMA, DAVIDSON, JAMES, EDWARD, PAUL, BEDFORD, SIMON, PACZAL, ATTILA, TIMÁRI, MÁTYÁS, PÁL, CHANRION, MAÏA, KOTSCHY, ANDRÁS, DODSWORTH, MARK, PHILIP, MARAGNO, ANA, LETICIA
Year of Publication 29.03.2024
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Year of Publication 29.03.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZIN-DERIVATER OG RELATEREDE FORBINDELSER SOM BCL-XL PROTEININHIBITORER OG PRO-APOPTOTISKE STOFFER TIL BEHANDLING AF CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, KOTSCHY, András, PACZAL, Attila, WEBB, Paul
Year of Publication 25.03.2024
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Year of Publication 25.03.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, PACZAL, Attila, KOTSCHY, András, WEBB, Paul
Year of Publication 21.03.2024
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Year of Publication 21.03.2024
Patent
Dérivés 6,7-dihydro-5h-pyrido[2,3-c]pyridazine et composés similaires en tant qu'inhibiteurs de la protéine bcl-xl et agents pro-apoptotiques pour le traitement du cancer
MARAGNO, Ana Leticia, TIMÁRI, Mátyás Pál, SANDERS, Emma, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, COLLAND, Frédéric, DAVIDSON, James Edward Paul, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, KOTSCHY, András, PACZAL, Attila, WEBB, Paul
Year of Publication 29.02.2024
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Year of Publication 29.02.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, PACZAL, Attila, KOTSCHY, András, WEBB, Paul
Year of Publication 12.02.2024
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Year of Publication 12.02.2024
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, NOVAK, Tibor, CHANRION, Maïa, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, STARCK, Jérôme-Benoit, PACZAL, Attila, KOTSCHY, András, WEBB, Paul
Year of Publication 27.12.2023
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Year of Publication 27.12.2023
Patent
6,7-DIHYDRO-5H-PYRIDO[2,3-C]PYRIDAZINE DERIVATIVES AND RELATED COMPOUNDS AS BCL-XL PROTEIN INHIBITORS AND PRO-APOPTOTIC AGENTS FOR TREATING CANCER
MARAGNO, Ana Leticia, SANDERS, Emma, TIMÁRI, Mátyás Pál, MURRAY, James Brooke, CHANRION, Maïa, STARCK, Jerome-Benoit, DAVIDSON, James Edward Paul, COLLAND, Frédéric, HERNER, András, DODSWORTH, Mark Philip, BEDFORD, Simon, NOVÁK, Tibor, PACZAL, Attila, KOTSCHY, András, WEBB, Paul
Year of Publication 25.12.2023
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Year of Publication 25.12.2023
Patent