Synthesis and structure-activity relationships of a novel series of 2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide K-ATP channel openers: Discovery of (-)-(9S)-9-(3-bromo-4-fluorophenyl)-2,3,5,6,7,9-hexahydrothieno[3,2-b]quinolin-8(4H)-one 1,1-dioxide (A-278637), a potent K-ATP opener that selectively inhibits spontaneous bladder contractions
Carroll, WA, Altenbach, RJ, Bai, H, Brioni, JD, Brune, ME, Buckner, SA, Cassidy, C, Chen, YY, Coghlan, MJ, Daza, AV, Drizin, Fey, TA, Fitzgerald, M, Gopalakrishnan, M, Gregg, RJ, Henry, RF, Holladay, MW, King, LL, Kort, ME, Kym, PR, Milicic, Tang, R, Turner, SC, Whiteaker, KL, Yi, L, Zhang, H, Sullivan, JP
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Published in Journal of medicinal chemistry (03.06.2004)
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A Scaleable Synthesis of Fiduxosin
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Published in Organic process research & development (01.11.2004)
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Synthesis and structure-activity relationships of a novel series of tricyclic dihydropyridine-based K-ATP openers that potently inhibit bladder contractions in vitro
Carroll, WA, Agrios, KA, Altenbach, RJ, Buckner, SA, Chen, YY, Coghlan, MJ, Daza, AV, Drizin, Gopalakrishnan, M, Henry, RF, Kort, ME, Kym, PR, Milicic, Smith, JC, Tang, R, Turner, SC, Whiteaker, KL, Zhang, H, Sullivan, JP
Published in Journal of medicinal chemistry (03.06.2004)
Published in Journal of medicinal chemistry (03.06.2004)
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Structure-activity studies for a novel series of tricyclic dihydropyridopyrazolones and dihydropyridoisoxazolones as KATP channel openers
DRIZIN, Irene, ALTENBACH, Robert J, CARROLL, William A, BUCKNER, Steven A, WHITEAKER, Kristi L, SCOTT, Victoria E, DARBYSHIRE, John F, JAYANTI, Venkata, HENRY, Rodger F, COGHLAN, Michael J, GOPALAKRISHNAN, Murali
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Synthesis of a novel farnesyl transferase inhibitor, ABT-100; selective preparation of a stereogenic tertiary carbinol
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Rao, S. T., Zurbenko, I. G., Neagu, R., Porter, P. S., Ku, J. Y., Henry, R. F.
Published in Bulletin of the American Meteorological Society (01.10.1997)
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An Assessment of the Sensitivity and Reliability of the Relative Reduction Factor Approach in the Development of 8-hr Ozone Attainment Plans
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Cherniawsky, J Y, eman, M G G, Crawford, W R, Henry, R F
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An Operational Assessment of the Application of the Relative Reduction Factors in the Demonstration of Attainment of the 8-Hr Ozone National Ambient Air Quality Standard
Sistla, G., Hogrefe, C., Hao, W., Ku, J.-Y., Zalewsky, E., Henry, R.F., Civerolo, K.
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Synthesis of Novel GABA Uptake Inhibitors. 3. Diaryloxime and Diarylvinyl Ether Derivatives of Nipecotic Acid and Guvacine as Anticonvulsant Agents
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Synthesis of 1H-pyridin-2-one derivatives as potent and selective farnesyltransferase inhibitors
LE WANG, LIN, Nan-Horng, SHAM, Hing L, QUN LI, HENRY, Rodger F, HAIYING ZHANG, COHEN, Jerome, GU, Wen-Zhen, MARSH, Kennan C, BAUCH, Joy L, ROSENBERG, Saul H
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An Unusual Intramolecular Hetero-Diels−Alder Cycloaddition
Stoner, Eric J, Allen, Michael S, Christesen, Alan C, Henry, Rodger F, Hollis, L. Steven, Keyes, Robert, Marsden, Ian, Rehm, Tamara C, Shiroor, Sandeep G, Soni, Niru B, Stewart, Kent D
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STEREOCONTROLLED SYNTHESIS OF C-2-SYMMETRICAL AND PSEUDO-C-2-SYMMETRICAL DIAMINO ALCOHOLS AND DIOLS FOR USE IN HIV PROTEASE INHIBITORS
KEMPF, DJ, SOWIN, TJ, DOHERTY, EM, HANNICK, SM, CODAVOCI, L, HENRY, RF, GREEN, BE, SPANTON, SG, NORBECK, DW
Published in Journal of organic chemistry (09.10.1992)
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Synthesis and structural elucidation of novel uranyl-crown ether compounds isolated from nitric, hydrochloric, sulfuric, and acetic acids
Rogers, Robin D, Bond, Andrew H, Hipple, William G, Rollins, Andrew N, Henry, Rodger F
Published in Inorganic chemistry (01.06.1991)
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Anhydrolide Macrolides. 1. Synthesis and Antibacterial Activity of 2,3-Anhydro-6-O-methyl 11,12-Carbamate Erythromycin A Analogues
Elliott, Richard L, Pireh, Daisy, Griesgraber, George, Nilius, Angela M, Ewing, Patty J, Bui, Mai Ha, Raney, Patti M, Flamm, Robert K, Kim, Ki, Henry, Rodger F, Chu, Daniel T. W, Plattner, Jacob J, Or, Yat Sun
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Effects of changes in data reporting practices on trend assessments
Henry, Robert F, Trivikrama Rao, S, Zurbenko, Igor G, Steven Porter, P
Published in Atmospheric environment (1994) (2000)
Published in Atmospheric environment (1994) (2000)
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Short period (1-4 h) sea level fluctuations on the Canterbury coast, New Zealand
Goring, Derek G., Henry, R. Falconer
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A Novel 13-Membered Erythromycin Analog via DAST-Induced Ring Contraction
Burnell-Curty, Cynthia, Faghih, Ramin, Pagano, Thomas, Henry, Rodger F, Lartey, Paul A
Published in Journal of organic chemistry (26.07.1996)
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3-Keto-11, 12-carbazate Derivatives of 6-O-Methylerythromycin A Synthesis and In Vitro Activity
GRIESGRABER, GEORGE, OR, YAT SUN, CHU, DANIEL T. W., NILIUS, ANGELA M., JOHNSON, PAULINE M., FLAMM, ROBERT K., HENRY, RODGER F., PLATTNER, JACOB J.
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