Identification of a series of oxadiazole-substituted α-isopropoxy phenylpropanoic acids with activity on PPARα, PPARγ, and PPARδ
Liu, Kevin G, Smith, Jennifer S, Ayscue, Andrea H, Henke, Brad R, Lambert, Millard H, Leesnitzer, Lisa M, Plunket, Kelli D, Willson, Timothy M, Sternbach, Daniel D
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
Published in Bioorganic & medicinal chemistry letters (03.09.2001)
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Synthesis and biological activity of l-tyrosine-based PPARγ agonists with reduced molecular weight
Liu, Kevin G., Lambert, Millard H., Ayscue, Andrea H., Henke, Brad R., Leesnitzer, Lisa M., Oliver, Jr, William R., Plunket, Kelli D., Xu, H.Eric, Sternbach, Daniel D., Willson, Timothy M.
Published in Bioorganic & medicinal chemistry letters (17.12.2001)
Published in Bioorganic & medicinal chemistry letters (17.12.2001)
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2-Amino-4,6-diarylpyridines as novel ligands for the estrogen receptor
HENKE, Brad R, DREWRY, David H, JONES, Stacey A, STEWART, Eugene L, WEAVER, Susan L, WIETHE, Robert W
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
Published in Bioorganic & medicinal chemistry letters (23.07.2001)
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3-[4-(1,2-Diphenylbut-1-enyl)phenyl]acrylic Acid: A Non-Steroidal Estrogen with Functional Selectivity for Bone over Uterus in Rats
Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Charifson, Paul S, Batchelor, Kenneth W, Lubahn, Dennis B, Moore, Linda B, Oliver, Beverly B, Sauls, Howard R, Triantafillou, James A, Wolfe, Steven G, Baer, Philip G
Published in Journal of medicinal chemistry (01.05.1994)
Published in Journal of medicinal chemistry (01.05.1994)
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HST5040: An investigational oral small molecule therapy entering phase 2 clinical development for methylmalonic (MMA) and propionic (PA) acidemias
Cox, Gerald, Armstrong, Allison, Waller, Mavis, Hayes, Mark, Collado, Maria Sol, Henke, Brad, Summar, Marshall, Wamhoff, Brian, Reardon, John, Figler, Robert, Johns, Brian, Chapman, Kimberly
Published in Molecular genetics and metabolism (01.04.2021)
Published in Molecular genetics and metabolism (01.04.2021)
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eP256 - HST5040: An investigational oral small molecule therapy entering phase 2 clinical development for methylmalonic (MMA) and propionic (PA) acidemias
Cox, Gerald, Armstrong, Allison, Waller, Mavis, Hayes, Mark, Collado, Maria Sol, Henke, Brad, Summar, Marshall, Wamhoff, Brian, Reardon, John, Figler, Robert, Johns, Brian, Chapman, Kimberly
Published in Molecular genetics and metabolism (01.04.2021)
Published in Molecular genetics and metabolism (01.04.2021)
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3-(1H-Indazol-3-ylmethyl)-1,5-benzodiazepines: CCK-A Agonists That Demonstrate Oral Activity as Satiety Agents
Henke, Brad R, Willson, Timothy M, Sugg, Elizabeth E, Croom, Dallas K, Dougherty, Robert W, Queen, Kennedy L, Birkemo, Larry S, Ervin, Gregory N, Grizzle, Mary K, Johnson, Michael F, James, Michael K
Published in Journal of medicinal chemistry (05.07.1996)
Published in Journal of medicinal chemistry (05.07.1996)
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3-[2-(N-Phenylacetamide)]-1,5-benzodiazepines: Orally Active, Binding Selective CCK-A Agonists
Willson, Timothy M, Henke, Brad R, Momtahen, Tanya M, Myers, Peter L, Sugg, Elizabeth E, Unwalla, Rayomand J, Croom, Dallas K, Dougherty, Robert W, Grizzle, Mary K, Johnson, Michael F, Queen, Kennedy L, Rimele, Thomas J, Yingling, Jeffrey D, James, Michael K
Published in Journal of medicinal chemistry (19.07.1996)
Published in Journal of medicinal chemistry (19.07.1996)
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Recent advances in estrogen receptor modulators
Henke, Brad R, Heyer, Dennis
Published in Current opinion in drug discovery & development (01.07.2005)
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Published in Current opinion in drug discovery & development (01.07.2005)
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CD38 CD38 INHIBITORS AND METHODS OF TREATMENT
HENKE BRAD RICHARD, BECHERER J. DAVID, CADILLA RODOLFO, HAFFNER CURT, DEATON DAVID NORMAN, SCHULTE CHRISTIE, PREUGSCHAT FRANK
Year of Publication 07.08.2017
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Year of Publication 07.08.2017
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