Practical Asymmetric Synthesis of (S)-4-Ethyl-7,8-dihydro-4-hydroxy-1H-pyrano[3,4-f]indolizine- 3,6,10(4H)-trione, a Key Intermediate for the Synthesis of Irinotecan and Other Camptothecin Analogs
Henegar, Kevin E, Ashford, Scott W, Baughman, Ted A, Sih, John C, Gu, Rui-Lin
Published in Journal of organic chemistry (19.09.1997)
Published in Journal of organic chemistry (19.09.1997)
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Overcoming the Challenges of Making a Single Enantiomer N‑1 Substituted Tetrazole Prodrug Using a Tin-Mediated Alkylation and Enzymatic Resolution
Akin, Anne, Barilla, Mark T, Brandt, Thomas A, Brennan, John, Henegar, Kevin E, Hoagland, Steve, Kumar, Rajesh, Magano, Javier, McInturff, Emma L, Nematalla, Asaad, Piotrowski, David W, Van Haitsma, Jared, Wei, Liuqing, Xiao, Jun, Yu, Shu
Published in Organic process research & development (21.06.2019)
Published in Organic process research & development (21.06.2019)
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Maximizing Lipophilic Efficiency: The Use of Free-Wilson Analysis in the Design of Inhibitors of Acetyl-CoA Carboxylase
Freeman-Cook, Kevin D, Amor, Paul, Bader, Scott, Buzon, Leanne M, Coffey, Steven B, Corbett, Jeffrey W, Dirico, Kenneth J, Doran, Shawn D, Elliott, Richard L, Esler, William, Guzman-Perez, Angel, Henegar, Kevin E, Houser, Janet A, Jones, Christopher S, Limberakis, Chris, Loomis, Katherine, McPherson, Kirk, Murdande, Sharad, Nelson, Kendra L, Phillion, Dennis, Pierce, Betsy S, Song, Wei, Sugarman, Eliot, Tapley, Susan, Tu, Meihua, Zhao, Zhengrong
Published in Journal of medicinal chemistry (26.01.2012)
Published in Journal of medicinal chemistry (26.01.2012)
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Process Development and Scale-up for (±)-Reboxetine Mesylate
Henegar, Kevin E, Ball, Cynthia T, Horvath, Carolyn M, Maisto, Keith D, Mancini, Sarah E
Published in Organic process research & development (01.05.2007)
Published in Organic process research & development (01.05.2007)
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Inside-Outside Stereoisomerism. 6.+ Synthesis of trans-Bicyclo[4.4.1]undecan-11-one and the First Stereoselective Construction of the Tricyclic Nucleus of the Ring System of the Ingenane Diterpenes
Winkler, Jeffrey D, Henegar, Kevin E, Hong, Bor-Cherng, Williard, Paul G
Published in Journal of the American Chemical Society (01.05.1994)
Published in Journal of the American Chemical Society (01.05.1994)
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Bromine-Mediated Addition of Nucleophiles to the Electron-Rich Pyrimidine Subunit of Tirilazad
Cabaj, John E, Wuts, Peter G. M, Henegar, Kevin E
Published in Journal of organic chemistry (01.08.1994)
Published in Journal of organic chemistry (01.08.1994)
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A Practical Synthesis of Cabergoline
Ashford, Scott W, Henegar, Kevin E, Anderson, Andrew M, Wuts, Peter G. M
Published in Journal of organic chemistry (04.10.2002)
Published in Journal of organic chemistry (04.10.2002)
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Total synthesis of (.+-.)-kempene 2
Dauben, William G, Farkas, Imre, Bridon, Dominique P, Chuang, Che Ping, Henegar, Kevin E
Published in Journal of the American Chemical Society (01.07.1991)
Published in Journal of the American Chemical Society (01.07.1991)
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Inside-outside stereoisomerism. II. Synthesis of the carbocyclic ring system of the ingenane diterpenes via the intramolecular dioxolenone photocycloaddition
Winkler, Jeffrey D, Henegar, Kevin E, Williard, Paul G
Published in Journal of the American Chemical Society (01.04.1987)
Published in Journal of the American Chemical Society (01.04.1987)
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Practical Asymmetric Synthesis of ( S )-4-Ethyl-7,8-dihydro-4-hydroxy-1 H -pyrano[3,4-f]indolizine- 3,6,10(4 H )-trione, a Key Intermediate for the Synthesis of Irinotecan and Other Camptothecin Analogs
Henegar, Kevin E., Ashford, Scott W., Baughman, Ted A., Sih, John C., Gu, Rui-Lin
Published in Journal of organic chemistry (01.09.1997)
Published in Journal of organic chemistry (01.09.1997)
Get full text
Journal Article