Bioactive sulfoximines: Syntheses and properties of Vioxx® analogs
Park, Seong Jun, Buschmann, Helmut, Bolm, Carsten
Published in Bioorganic & medicinal chemistry letters (15.08.2011)
Published in Bioorganic & medicinal chemistry letters (15.08.2011)
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Journal Article
Synthesis and Biological Evaluation of the 1‑Arylpyrazole Class of σ1 Receptor Antagonists: Identification of 4‑{2-[5-Methyl-1-(naphthalen-2-yl)‑1H‑pyrazol-3-yloxy]ethyl}morpholine (S1RA, E‑52862)
Díaz, José Luis, Cuberes, Rosa, Berrocal, Joana, Contijoch, Montserrat, Christmann, Ute, Fernández, Ariadna, Port, Adriana, Holenz, Jörg, Buschmann, Helmut, Laggner, Christian, Serafini, Maria Teresa, Burgueño, Javier, Zamanillo, Daniel, Merlos, Manuel, Vela, José Miguel, Almansa, Carmen
Published in Journal of medicinal chemistry (11.10.2012)
Published in Journal of medicinal chemistry (11.10.2012)
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Journal Article
N-Cyano Sulfoximines: COX Inhibition, Anticancer Activity, Cellular Toxicity, and Mutagenicity
Park, Seong Jun, Baars, Hannah, Mersmann, Stefanie, Buschmann, Helmut, Baron, Jens Malte, Amann, Philipp M., Czaja, Katharina, Hollert, Henner, Bluhm, Kerstin, Redelstein, Regine, Bolm, Carsten
Published in ChemMedChem (01.02.2013)
Published in ChemMedChem (01.02.2013)
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Journal Article
Syntheses and biological activities of sulfoximine-based acyclic triaryl olefins
Chen, Xiao Yun, Park, Seong Jun, Buschmann, Helmut, De Rosa, Maria, Bolm, Carsten
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
Published in Bioorganic & medicinal chemistry letters (01.07.2012)
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Journal Article
5-HT7 receptor activation inhibits mechanical hypersensitivity secondary to capsaicin sensitization in mice
BRENCHAT, Alex, ROMERO, Luz, MIGUEL VELA, José, GARCIA, Monica, PUJOL, Marta, BURGUENO, Javier, TORRENS, Antoni, HAMON, Michel, BAEYENS, José Manuel, BUSCHMANN, Helmut, ZAMANILLO, Daniel
Published in Pain (Amsterdam) (01.02.2009)
Published in Pain (Amsterdam) (01.02.2009)
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Journal Article
Mechanistic and functional differentiation of tapentadol and tramadol
Raffa, Robert B, Buschmann, Helmut, Christoph, Thomas, Eichenbaum, Gary, Englberger, Werner, Flores, Christopher M, Hertrampf, Torsten, Kögel, Babette, Schiene, Klaus, Straßburger, Wolfgang, Terlinden, Rolf, Tzschentke, Thomas M
Published in Expert opinion on pharmacotherapy (01.07.2012)
Published in Expert opinion on pharmacotherapy (01.07.2012)
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Journal Article
Sigma-1 receptor antagonism as opioid adjuvant strategy: Enhancement of opioid antinociception without increasing adverse effects
Vidal-Torres, Alba, de la Puente, Beatriz, Rocasalbas, Maria, Touriño, Clara, Andreea Bura, Simona, Fernández-Pastor, Begoña, Romero, Luz, Codony, Xavier, Zamanillo, Daniel, Buschmann, Helmut, Merlos, Manuel, Manuel Baeyens, José, Maldonado, Rafael, Vela, José Miguel
Published in European journal of pharmacology (05.07.2013)
Published in European journal of pharmacology (05.07.2013)
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Journal Article
New Developments in the Origins of the Homochirality of Biologically Relevant Molecules
Buschmann, Helmut, Thede, Richard, Heller, Detlef
Published in Angewandte Chemie International Edition (17.11.2000)
Published in Angewandte Chemie International Edition (17.11.2000)
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Journal Article
Differential anti-neuropathic pain effects of tetrodotoxin in sciatic nerve- versus infraorbital nerve-ligated rats – Behavioral, pharmacological and immunohistochemical investigations
Kayser, Valérie, Viguier, Florent, Ioannidi, Myrto, Bernard, Jean-François, Latrémolière, Alban, Michot, Benoît, Vela, José-Miguel, Buschmann, Helmut, Hamon, Michel, Bourgoin, Sylvie
Published in Neuropharmacology (01.02.2010)
Published in Neuropharmacology (01.02.2010)
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Journal Article
Functional and Molecular Characterization of Voltage-Gated Sodium Channels in Uteri from Nonpregnant Rats
SEDA, Marian, PINTO, Francisco M, WRAY, Susan, CINTADO, Cristina G, NOHEDA, Pedro, BUSCHMANN, Helmut, CANDENAS, Luz
Published in Biology of reproduction (01.11.2007)
Published in Biology of reproduction (01.11.2007)
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Journal Article
The quality of drugs and drug products - Always guaranteed?
Buschmann, Helmut, Handler, Norbert, Holzgrabe, Ulrike
Published in Journal of pharmaceutical and biomedical analysis (15.02.2024)
Published in Journal of pharmaceutical and biomedical analysis (15.02.2024)
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Journal Article
Epigenetic Drug Discovery
Sippl, Wolfgang, Jung, Manfred, Mannhold, Raimund, Buschmann, Helmut, Holenz, Jörg
Year of Publication 2019
Year of Publication 2019
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Functional and Molecular Characterization of Voltage-Gated Sodium Channels in Uteri from Nonpregnant Rats1
Seda, Marian, Pinto, Francisco M, Wray, Susan, Cintado, Cristina G, Noheda, Pedro, Buschmann, Helmut, Candenas, Luz
Published in Biology of reproduction (01.11.2007)
Published in Biology of reproduction (01.11.2007)
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Journal Article
Stereoselective and efficient synthesis of ( S)-pregabalin from d-mannitol
Izquierdo, Sandra, Aguilera, Jordi, Buschmann, Helmut H., García, Mónica, Torrens, Antoni, Ortuño, Rosa M.
Published in Tetrahedron: asymmetry (03.04.2008)
Published in Tetrahedron: asymmetry (03.04.2008)
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Journal Article
Application of advanced high resolution mass spectrometric techniques for the analysis of losartan potassium regarding known and unknown impurities
Backer, Laura, Buschmann, Helmut, Kinzig, Martina, Sörgel, Fritz, Scherf-Clavel, Oliver, Holzgrabe, Ulrike
Published in Journal of pharmaceutical and biomedical analysis (15.03.2024)
Published in Journal of pharmaceutical and biomedical analysis (15.03.2024)
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Journal Article
Prediction of Degradation Profiles for Various Sartans under Solvent-Free Mechanochemical Conditions
Amer, Mostafa M., Backer, Laura, Buschmann, Helmut, Handler, Norbert, Scherf-Clavel, Oliver, Holzgrabe, Ulrike, Bolm, Carsten
Published in Analytical chemistry (Washington) (13.08.2024)
Published in Analytical chemistry (Washington) (13.08.2024)
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Journal Article
Strategy to Assess and Control Nitrosamine Formation in API during Storage: A Sitagliptin Case Study
Badia, Laura, Camps, Helena, Lloveras, Isabel, Handler, Norbert, Buschmann, Helmut, Valls, Jordi, Poznik, Michal
Published in Organic process research & development (16.08.2024)
Published in Organic process research & development (16.08.2024)
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Journal Article
Discovery, Chemistry, and Preclinical Development of Pritelivir, a Novel Treatment Option for Acyclovir-Resistant Herpes Simplex Virus Infections
Birkmann, Alexander, Bonsmann, Susanne, Kropeit, Dirk, Pfaff, Tamara, Rangaraju, Manickam, Sumner, Melanie, Timmler, Burkhard, Zimmermann, Holger, Buschmann, Helmut, Ruebsamen-Schaeff, Helga
Published in Journal of medicinal chemistry (27.10.2022)
Published in Journal of medicinal chemistry (27.10.2022)
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Journal Article