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Published in Science (American Association for the Advancement of Science) (13.07.2012)
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Published in Journal of medicinal chemistry (14.07.2016)
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Jespers, Willem, Heitman, Laura H, IJzerman, Adriaan P, Sotelo, Eddy, van Westen, Gerard J P, Åqvist, Johan, Gutiérrez-de-Terán, Hugo
Published in PLoS computational biology (01.11.2021)
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Schuetz, Doris A., de Witte, Wilhelmus Egbertus Arnout, Wong, Yin Cheong, Knasmueller, Bernhard, Richter, Lars, Kokh, Daria B., Sadiq, S. Kashif, Bosma, Reggie, Nederpelt, Indira, Heitman, Laura H., Segala, Elena, Amaral, Marta, Guo, Dong, Andres, Dorothee, Georgi, Victoria, Stoddart, Leigh A., Hill, Steve, Cooke, Robert M., De Graaf, Chris, Leurs, Rob, Frech, Matthias, Wade, Rebecca C., de Lange, Elizabeth Cunera Maria, IJzerman, Adriaan P., Müller-Fahrnow, Anke, Ecker, Gerhard F.
Published in Drug discovery today (01.06.2017)
Published in Drug discovery today (01.06.2017)
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Molecular Basis of Ligand Dissociation from the Adenosine A2A Receptor
Guo, Dong, Pan, Albert C, Dror, Ron O, Mocking, Tamara, Liu, Rongfang, Heitman, Laura H, Shaw, David E, IJzerman, Adriaan P
Published in Molecular pharmacology (01.05.2016)
Published in Molecular pharmacology (01.05.2016)
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Indanes-Properties, Preparation, and Presence in Ligands for G Protein Coupled Receptors
Vilums, Maris, Heuberger, Jules, Heitman, Laura H., IJzerman, Adriaan P.
Published in Medicinal research reviews (01.11.2015)
Published in Medicinal research reviews (01.11.2015)
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Li, Xiaoting, Chang, Hao, Bouma, Jara, de Paus, Laura V., Mukhopadhyay, Partha, Paloczi, Janos, Mustafa, Mohammed, van der Horst, Cas, Kumar, Sanjay Sunil, Wu, Lijie, Yu, Yanan, van den Berg, Richard J. B. H. N., Janssen, Antonius P. A., Lichtman, Aron, Liu, Zhi-Jie, Pacher, Pal, van der Stelt, Mario, Heitman, Laura H., Hua, Tian
Published in Nature communications (15.03.2023)
Published in Nature communications (15.03.2023)
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The Role of a Sodium Ion Binding Site in the Allosteric Modulation of the A2A Adenosine G Protein-Coupled Receptor
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Published in Structure (London) (03.12.2013)
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Ortiz Zacarías, Natalia V, Röth, Sascha, Broekhuis, Jeremy D, van der Es, Daan, Moreau, Kevin, Heitman, Laura H
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Gorostiola González, Marina, Rakers, Pepijn R J, Jespers, Willem, IJzerman, Adriaan P, Heitman, Laura H, van Westen, Gerard J P
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Published in Scientific reports (08.07.2021)
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Published in Frontiers in pharmacology (10.08.2021)
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Lemmerhirt, Jan Phillip, Isaak, Andreas, Liu, Rongfang, Kock, Max, Daniliuc, Constantin G., Jacobson, Kenneth A., Heitman, Laura H., Junker, Anna
Published in Molecules (Basel, Switzerland) (31.03.2022)
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Mocking, Tamara A M, Sijben, Hubert J, Vermeulen, Yimé W, IJzerman, Adriaan P, Heitman, Laura H
Published in International journal of molecular sciences (21.01.2022)
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Label-free high-throughput screening assay for the identification of norepinephrine transporter (NET/SLC6A2) inhibitors
Sijben, Hubert J., van Oostveen, Wieke M., Hartog, Peter B. R., Stucchi, Laura, Rossignoli, Andrea, Maresca, Giovanna, Scarabottolo, Lia, IJzerman, Adriaan P., Heitman, Laura H.
Published in Scientific reports (10.06.2021)
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Cancer-Related Somatic Mutations in Transmembrane Helices Alter Adenosine A1 Receptor Pharmacology
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Published in Molecules (Basel, Switzerland) (10.06.2022)
Published in Molecules (Basel, Switzerland) (10.06.2022)
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