Identification of a nonkinase target mediating cytotoxicity of novel kinase inhibitors
Ross-Macdonald, Petra, de Silva, Heshani, Guo, Qi, Xiao, Hong, Hung, Chen-Yi, Penhallow, Becky, Markwalder, Jay, He, Liqi, Attar, Ricardo M, Lin, Tai-an, Seitz, Steven, Tilford, Charles, Wardwell-Swanson, Judith, Jackson, Donald
Published in Molecular cancer therapeutics (01.11.2008)
Published in Molecular cancer therapeutics (01.11.2008)
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Synthesis and Structure−Activity Relationships of 8-(Pyrid-3-yl)pyrazolo[1,5-a]-1,3,5-triazines: Potent, Orally Bioavailable Corticotropin Releasing Factor Receptor-1 (CRF1) Antagonists
Gilligan, Paul J, Clarke, Todd, He, Liqi, Lelas, Snjezana, Li, Yu-Wen, Heman, Karen, Fitzgerald, Lawrence, Miller, Keith, Zhang, Ge, Marshall, Anne, Krause, Carol, McElroy, John F, Ward, Kathyrn, Zeller, Kim, Wong, Harvey, Bai, Steven, Saye, Joanne, Grossman, Scott, Zaczek, Robert, Arneric, Stephen P, Hartig, Paul, Robertson, David, Trainor, George
Published in Journal of medicinal chemistry (14.05.2009)
Published in Journal of medicinal chemistry (14.05.2009)
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Modulation of cofilin phosphorylation by inhibition of the Lim family kinases
He, Liqi, Seitz, Steven P., Trainor, George L., Tortolani, David, Vaccaro, Wayne, Poss, Michael, Tarby, Christine M., Tokarski, John S., Penhallow, Becky, Hung, Chen-Yi, Attar, Ricardo, Lin, Tai-An
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
Published in Bioorganic & medicinal chemistry letters (15.09.2012)
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8-(4-Methoxyphenyl)pyrazolo[1,5-a]-1,3,5-triazines: Selective and Centrally Active Corticotropin-Releasing Factor Receptor-1 (CRF1) Antagonists
Gilligan, Paul J, He, Liqi, Clarke, Todd, Tivitmahaisoon, Parcharee, Lelas, Snjezana, Li, Yu-Wen, Heman, Karen, Fitzgerald, Lawrence, Miller, Keith, Zhang, Ge, Marshall, Anne, Krause, Carol, McElroy, John, Ward, Kathyrn, Shen, Helen, Wong, Harvey, Grossman, Scott, Nemeth, Gregory, Zaczek, Robert, Arneric, Stephen P, Hartig, Paul, Robertson, David W, Trainor, George
Published in Journal of medicinal chemistry (14.05.2009)
Published in Journal of medicinal chemistry (14.05.2009)
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SAR of PXR transactivation in benzimidazole-based IGF-1R kinase inhibitors
Zimmermann, Kurt, Wittman, Mark D., Saulnier, Mark G., Velaparthi, Upender, Sang, Xiaopeng, Frennesson, David B., Struzynski, Charles, Seitz, Steven P., He, Liqi, Carboni, Joan M., Li, Aixin, Greer, Ann F., Gottardis, Marco, Attar, Ricardo M., Yang, Zheng, Balimane, Praveen, Discenza, Lorell N., Lee, Francis Y., Sinz, Michael, Kim, Sean, Vyas, Dolatrai
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
Published in Bioorganic & medicinal chemistry letters (01.03.2010)
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Effects of a Non-peptide CRF Antagonist (DMP696) on the Behavioral and Endocrine Sequelae of Maternal Separation
Maciag, Carla M, Dent, Gersham, Gilligan, Paul, He, Liqi, Dowling, Krista, Ko, Tracey, Levine, Seymour, Smith, Mark A
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2002)
Published in Neuropsychopharmacology (New York, N.Y.) (01.05.2002)
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The CRF1 receptor antagonist DMP696 produces anxiolytic effects and inhibits the stress-induced hypothalamic-pituitary-adrenal axis activation without sedation or ataxia in rats
MCELROY, John F, WARD, Kathryn A, ZELLER, Kim L, JONES, Keith W, GILLIGAN, Paul J, LIQI HE, LELAS, Sniezana
Published in Psychopharmacologia (01.12.2002)
Published in Psychopharmacologia (01.12.2002)
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Non-Peptide Corticotropin-Releasing Hormone Antagonists: Syntheses and Structure−Activity Relationships of 2-Anilinopyrimidines and -triazines
Arvanitis, Argyrios G, Gilligan, Paul J, Chorvat, Robert J, Cheeseman, Robert S, Christos, Thomas E, Bakthavatchalam, Rajagopal, Beck, James P, Cocuzza, Anthony J, Hobbs, Frank W, Wilde, Richard G, Arnold, Charles, Chidester, Dennis, Curry, Matthew, He, Liqi, Hollis, Andrea, Klaczkiewicz, John, Krenitsky, Paul J, Rescinito, Joseph P, Scholfield, Everett, Culp, Steven, De Souza, Errol B, Fitzgerald, Lawrence, Grigoriadis, Dimitri, Tam, S. William, Wong, Y. Nancy, Huang, Shiew-Mei, Shen, Helen L
Published in Journal of medicinal chemistry (11.03.1999)
Published in Journal of medicinal chemistry (11.03.1999)
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4-(1,3-Dimethoxyprop-2-ylamino)-2,7-dimethyl-8-(2,4-dichlorophenyl)pyrazolo[1,5-a]-1,3,5-triazine: A Potent, Orally Bioavailable CRF1 Receptor Antagonist
He, Liqi, Gilligan, Paul J, Zaczek, Robert, Fitzgerald, Lawrence W, McElroy, John, Shen, H-S. L, Saye, Jo Anne, Kalin, Ned H, Shelton, Steven, Christ, David, Trainor, George, Hartig, Paul
Published in Journal of medicinal chemistry (10.02.2000)
Published in Journal of medicinal chemistry (10.02.2000)
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Discovery of Novel TLR7 Agonists as Systemic Agent for Combination With aPD1 for Use in Immuno-oncology
Poudel, Yam B., He, Liqi, Cox, Matthew, Zhang, Qian, Johnson, Walter L., Cong, Qiang, Cheng, Heng, Chowdari, Naidu S., Tarby, Christine, Donnell, Andrew F., Broekema, Matthais, O’Malley, Daniel P., Zhang, Yong, A. M. Subbaiah, Murugaiah, Kumar, Boda Vijay, Subramani, Lakshumanan, Wang, Bei, Li, Yi-Xin, Sivaprakasam, Prasanna, Critton, David, Mulligan, Dawn, Sandhu, Bhupindar, Xie, Chunshan, Ramakrishnan, Radha, Nagar, Jignesh, Dudhgaonkar, Shailesh, Oderinde, Martins S., Murtaza, Anwar, Schieven, Gary L., Mathur, Arvind, Gavai, Ashvinikumar V., Vite, Gregory, Gangwar, Sanjeev
Published in ACS medicinal chemistry letters (08.02.2024)
Published in ACS medicinal chemistry letters (08.02.2024)
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Journal Article
Identification and Optimization of Small Molecule Pyrazolopyrimidine TLR7 Agonists for Applications in Immuno-oncology
He, Liqi, Zhang, Meng Yao, Cox, Matthew, Zhang, Qian, Donnell, Andrew F., Zhang, Yong, Tarby, Christine, Gill, Patrice, Subbaiah, Murugaiah A. M., Ramar, Thangeswaran, Reddy, Maheswara, Puttapaka, Vijaya, Li, Yi-Xin, Sivaprakasam, Prasanna, Critton, David, Mulligan, Dawn, Xie, Chunshan, Ramakrishnan, Radha, Nagar, Jignesh, Dudhgaonkar, Shailesh, Murtaza, Anwar, Oderinde, Martins S., Schieven, Gary L., Mathur, Arvind, Gavai, Ashvinikumar V., Vite, Gregory, Gangwar, Sanjeev, Poudel, Yam B.
Published in ACS medicinal chemistry letters (08.02.2024)
Published in ACS medicinal chemistry letters (08.02.2024)
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Abstract 5417: The identification of BMS-595, an orally active imidazo[1,2-b]pyridazine CK2 inhibitor with in vivo anti-tumor activity
Tarby, Christine M., He, Liqi, Fink, Brian E., Nation, Andrew, Zhao, Yufen, Kim, Soong-Hoon, Chen, Libing, Tokarski, John S., Yu, Chiang, Pabalan, Jonathan G., Roongta, Urvashi V., Lippy, Jonathan, Obermeier, Mary, Elzinga, Paul A., Fura, Aberra, Henley, Benjamin, Fargnoli, Joseph J., Foster, William R., Gavai, Ashvinikumar V., Wong, Tai W., Hunt, John T., Vite, Gregory D., Purandare, Ashok V., Rupnow, Brent A.
Published in Cancer research (Chicago, Ill.) (01.08.2015)
Published in Cancer research (Chicago, Ill.) (01.08.2015)
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The CRF 1 receptor antagonist DMP696 produces anxiolytic effects and inhibits the stress-induced hypothalamic-pituitary-adrenal axis activation without sedation or ataxia in rats
McElroy, John, Ward, Kathryn, Zeller, Kim, Jones, Keith, Gilligan, Paul, He, Liqi, Lelas, Snjezana
Published in Psychopharmacology (01.12.2002)
Published in Psychopharmacology (01.12.2002)
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