Development of isoform selective PI3-kinase inhibitors as pharmacological tools for elucidating the PI3K pathway
Bruce, Ian, Akhlaq, Mohammed, Bloomfield, Graham C., Budd, Emma, Cox, Brian, Cuenoud, Bernard, Finan, Peter, Gedeck, Peter, Hatto, Julia, Hayler, Judy F., Head, Denise, Keller, Thomas, Kirman, Louise, Leblanc, Catherine, Grand, Darren Le, McCarthy, Clive, O’Connor, Desmond, Owen, Charles, Oza, Mrinalini S., Pilgrim, Gaynor, Press, Nicola E., Sviridenko, Lilya, Whitehead, Lewis
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
Published in Bioorganic & medicinal chemistry letters (01.09.2012)
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Design and Synthesis of Thrombin Inhibitors: Analogues of MD-805 with Reduced Stereogenicity and Improved Potency
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Published in Journal of medicinal chemistry (04.11.1999)
Published in Journal of medicinal chemistry (04.11.1999)
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Amidine protection for solution phase library synthesis
Bailey, Christine, Baker, Emma, Hayler, Judy, Kane, Peter
Published in Tetrahedron letters (25.06.1999)
Published in Tetrahedron letters (25.06.1999)
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PYRAZOLO [3,4-D] PYRIMIDINE DERIVATIVES USEFUL TO TREAT RESPIRATORY DISORDERS
Howsham, Catherine, Bloomfield, Graham Charles, Hayler, Judy Fox, Cox, Brian, Edwards, Lee, Bruce, Ian
Year of Publication 10.05.2018
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Year of Publication 10.05.2018
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the design and synthesis of thrombin inhibitors: the introduction of in vivo efficacy and oral bioavailability into benzthiazolylalanine inhibitors
Hayler, Judy, Kane, Peter D, LeGrand, Darren, Lugrin, Florence, Menear, Keith, Price, Richard, Allen, Mark, Cockcroft, Xiaoling, Ambler, John, Butler, Keith, Dunnet, Karren, Mitchelson, Andrew, Talbot, Mark, Tweed, Morris, Wills, Nicholas
Published in Bioorganic & medicinal chemistry letters (17.07.2000)
Published in Bioorganic & medicinal chemistry letters (17.07.2000)
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PYRAZOLO [3,4-D] PYRIMIDINE DERIVATIVES USEFUL TO TREAT RESPIRATORY DISORDERS
Cox Brian, Bruce Ian, Bloomfield Graham Charles, Edwards Lee, Hayler Judy Fox, Howsham Catherine
Year of Publication 20.10.2016
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Year of Publication 20.10.2016
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Optimisation of the P2 pharmacophore in a series of thrombin inhibitors: Ion-dipole interactions with lysine 60G
Ambler, John, Brown, Lyndon, Cockcroft, Xiao-Ling, Grütter, Markus, Hayler, Judy, Janus, Diana, Jones, Darryl, Kane, Peter, Menear, Keith, Priestle, John, Smith, Garrick, Talbot, Mark, Walker, Clive V, Wathey, Bernard
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
Published in Bioorganic & medicinal chemistry letters (03.05.1999)
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Studies towards the identification of potent, selective and bioavailable thrombin inhibitors
Ambler, John, Baker, Emma, Bentley, Dave, Brown, Lyndon, Butler, Keith, Butler, Paul, Farr, Dave, Dunnet, Karen, Grand, Darren Le, Hayler, Judy, Janus, Diana, Jones, Darryl, Menear, Keith, Mercer, Mark, Smith, Garrick, Talbot, Mark, Tweed, Morris
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
Published in Bioorganic & medicinal chemistry letters (08.03.1999)
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Pyrazolo [3,4-D] pyrimidine derivatives useful to treat respiratory disorders
EDWARDS LEE, HAYLER JUDY FOX, BRUCE IAN, COX BRIAN, BLOOMFIELD GRAHAM CHARLES, HOWSHAM CATHERINE
Year of Publication 02.12.2014
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Year of Publication 02.12.2014
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PYRAZOLO [3,4-D] PYRIMIDINE DERIVATIVES USEFUL TO TREAT RESPIRATORY DISORDERS
EDWARDS LEE, HAYLER JUDY FOX, BRUCE IAN, COX BRIAN, BLOOMFIELD GRAHAM CHARLES, HOWSHAM CATHERINE
Year of Publication 21.08.2014
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Year of Publication 21.08.2014
Patent
Pyrazolo [3,4-D] Pyrimidine Derivatives Useful to Treat Respiratory Disorders
EDWARDS LEE, HAYLER JUDY FOX, BRUCE IAN, COX BRIAN, BLOOMFIELD GRAHAM CHARLES, HOWSHAM CATHERINE
Year of Publication 20.02.2014
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Year of Publication 20.02.2014
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5-PHENYLTHIAZOLE DERIVATIVES AND USE AS P13 KINASE INHIBITORS
LOUISE KIRMAN, MRINALINI SACHIN OZA, IAN BRUCE, LEWIS WHITEHEAD, CATHERINE LEBLANC, JUDY HAYLER, PETER FINAN, LENA SHUKLA, NICOLA ELAINE BLAIR, CLIVE MCCARTHY, GRAHAM CHARLES BLOOMFIELD
Year of Publication 26.02.2016
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Year of Publication 26.02.2016
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Inhibitors of phosphatidylinositol 3-kinase
BRUCE, IAN, PILGRIM, GAYNOR ELIZABETH, PRESS, NICOLA, LE GRAND, DARREN MARK, RITCHIE, CATHY, VALADE, BARBARA, HAYLER, JUDY, KELLER, THOMAS HUGO, BUDD, EMMA, CUENOUD, BERNARD
Year of Publication 10.06.2015
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Year of Publication 10.06.2015
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5-phenylthiazole derivatives and their use as Pi3 kinase inhibitors
OZA MRINALINI SACHIN, WHITEHEAD LEWIS, SHUKLA LENA, BRUCE IAN, BLOOMFIELD GRAHAM CHARLES, MCCARTHY CLIVE, FINAN PETER, PRESS NICOLA ELAINE, HAYLER JUDY, LEBLANC CATHERINE, KIRMAN LOUISE
Year of Publication 30.04.2015
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Year of Publication 30.04.2015
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Thiazol-2-yl organic compounds
HAYLER, JUDY, FOX, HATTO, JULIA, DORIS, IDA, VALADE, BARBARA, BUDD, EMMA, LEGRAND, DARREN, MARK
Year of Publication 17.08.2011
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Year of Publication 17.08.2011
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5-phenyl-thiazol-2-yl-urea derivatives and use as PI3 kinase inhibitors
HAYLER JUDY FOX, LEGRAND DARREN MARK, BUDD EMMA, BRUCE IAN, COX BRIAN
Year of Publication 16.08.2011
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Year of Publication 16.08.2011
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5-phenyl-thiazol-2-yl-urea derivatives and use as PI3 kinase inhibitors
Budd, Emma, Hayler, Judy Fox, Bruce, Ian, Legrand, Darren Mark, Cox, Brian
Year of Publication 16.08.2011
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Year of Publication 16.08.2011
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