Absorption, distribution, metabolism, and excretion of ticagrelor in healthy subjects
Teng, Renli, Oliver, Stuart, Hayes, Martin A, Butler, Kathleen
Published in Drug metabolism and disposition (01.09.2010)
Published in Drug metabolism and disposition (01.09.2010)
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Journal Article
Enzymatic Late‐Stage Modifications: Better Late Than Never
Romero, Elvira, Jones, Bethan S., Hogg, Bethany N., Rué Casamajo, Arnau, Hayes, Martin A., Flitsch, Sabine L., Turner, Nicholas J., Schnepel, Christian
Published in Angewandte Chemie International Edition (26.07.2021)
Published in Angewandte Chemie International Edition (26.07.2021)
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Journal Article
Phytochemicals in Drug Discovery—A Confluence of Tradition and Innovation
Chihomvu, Patience, Ganesan, A, Gibbons, Simon, Woollard, Kevin, Hayes, Martin A
Published in International journal of molecular sciences (13.08.2024)
Published in International journal of molecular sciences (13.08.2024)
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Journal Article
Late‐Stage Functionalization of Histidine in Unprotected Peptides
Noisier, Anaïs F. M., Johansson, Magnus J., Knerr, Laurent, Hayes, Martin A., Drury, William J., Valeur, Eric, Malins, Lara R., Gopalakrishnan, Ranganath
Published in Angewandte Chemie International Edition (19.12.2019)
Published in Angewandte Chemie International Edition (19.12.2019)
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Journal Article
The Impact of Metagenomics on Biocatalysis
Hogg, Bethany N., Schnepel, Christian, Finnigan, James D., Charnock, Simon J., Hayes, Martin A., Turner, Nicholas J.
Published in Angewandte Chemie International Edition (21.05.2024)
Published in Angewandte Chemie International Edition (21.05.2024)
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Journal Article
Biocatalytic Monoacylation of Symmetrical Diamines and Its Application to the Synthesis of Pharmaceutically Relevant Amides
Lubberink, Max, Schnepel, Christian, Citoler, Joan, Derrington, Sasha R, Finnigan, William, Hayes, Martin A, Turner, Nicholas J, Flitsch, Sabine L
Published in ACS catalysis (04.09.2020)
Published in ACS catalysis (04.09.2020)
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Journal Article
Regiodivergent Radical Termination for Intermolecular Biocatalytic C–C Bond Formation
Petchey, Mark R., Ye, Yuxuan, Spelling, Victor, Finnigan, James D., Gittings, Samantha, Johansson, Magnus J., Hayes, Martin A., Hyster, Todd K.
Published in Journal of the American Chemical Society (21.02.2024)
Published in Journal of the American Chemical Society (21.02.2024)
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Journal Article
A Universal, Continuous Assay for SAM‐dependent Methyltransferases
Menke, Marian J., Schneider, Pascal, Badenhorst, Christoffel P. S., Kunzendorf, Andreas, Heinz, Florian, Dörr, Mark, Hayes, Martin A., Bornscheuer, Uwe T.
Published in Angewandte Chemie International Edition (18.12.2023)
Published in Angewandte Chemie International Edition (18.12.2023)
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Journal Article
The evolution of cytochrome P450 enzymes as biocatalysts in drug discovery and development
Gillam, Elizabeth M J, Hayes, Martin A
Published in Current topics in medicinal chemistry (01.09.2013)
Published in Current topics in medicinal chemistry (01.09.2013)
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Journal Article
The Role of Cytochrome P450 AbyV in the Final Stages of Abyssomicin C Biosynthesis
Devine, Andrew J., Parnell, Alice E., Back, Catherine R., Lees, Nicholas R., Johns, Samuel T., Zulkepli, Ainul Z., Barringer, Rob, Zorn, Katja, Stach, James E. M., Crump, Matthew P., Hayes, Martin A., Kamp, Marc W., Race, Paul R., Willis, Christine L.
Published in Angewandte Chemie International Edition (16.01.2023)
Published in Angewandte Chemie International Edition (16.01.2023)
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Journal Article
Engineering Biocatalysts for the C−H Activation of Fatty Acids by Ancestral Sequence Reconstruction
Jones, Bethan S., Ross, Connie M., Foley, Gabriel, Pozhydaieva, Nadiia, Sharratt, Joseph W., Kress, Nico, Seibt, Lisa S., Thomson, Raine E. S., Gumulya, Yosephine, Hayes, Martin A., Gillam, Elizabeth M. J., Flitsch, Sabine L.
Published in Angewandte Chemie International Edition (24.04.2024)
Published in Angewandte Chemie International Edition (24.04.2024)
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Journal Article
Biocatalysis in Drug Design: Engineered Reductive Aminases (RedAms) Are Used to Access Chiral Building Blocks with Multiple Stereocenters
Casamajo, Arnau Rué, Yu, Yuqi, Schnepel, Christian, Morrill, Charlotte, Barker, Rhys, Levy, Colin W., Finnigan, James, Spelling, Victor, Westerlund, Kristina, Petchey, Mark, Sheppard, Robert J., Lewis, Richard J., Falcioni, Francesco, Hayes, Martin A., Turner, Nicholas J.
Published in Journal of the American Chemical Society (11.10.2023)
Published in Journal of the American Chemical Society (11.10.2023)
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Journal Article
Design and Development of Glucocorticoid Receptor Modulators as Immunology Antibody–Drug Conjugate Payloads
Hobson, Adrian D, McPherson, Michael J, Waegell, Wendy, Goess, Christian A, Stoffel, Robert H, Li, Xiang, Zhou, Jian, Wang, Zhongyuan, Yu, Yajie, Hernandez, Axel, Bryant, Shaughn H, Mathieu, Suzanne L, Bischoff, Agnieszka K, Fitzgibbons, Julia, Pawlikowska, Martyna, Puthenveetil, Sujiet, Santora, Ling C, Wang, Lu, Wang, Lu, Marvin, Christopher C, Hayes, Martin E, Shrestha, Anurupa, Sarris, Kathy A, Li, Biqin
Published in Journal of medicinal chemistry (24.03.2022)
Published in Journal of medicinal chemistry (24.03.2022)
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Journal Article
Biocatalysis using Thermostable Cytochrome P450 Enzymes in Bacterial Membranes - Comparison of Metabolic Pathways with Human Liver Microsomes and Recombinant Human Enzymes
Jurva, Ulrik, Sandinge, Ann-Sofie, Baek, Jong Min, Avanthay, Mickaël, Thomson, Raine E S, D'Cunha, Stephlina A, Andersson, Shalini, Hayes, Martin A, Gillam, Elizabeth M J
Published in Drug metabolism and disposition (01.03.2024)
Published in Drug metabolism and disposition (01.03.2024)
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Journal Article
Self-Immolative Carbamate Linkers for CD19-Budesonide Antibody–Drug Conjugates
Marvin, Christopher C., Hobson, Adrian D., McPherson, Michael, Dunstan, Theresa A., Vargo, Thomas R., Hayes, Martin E., Fettis, Margaret M., Bischoff, Agnieszka, Wang, Lu, Wang, Lu, Hernandez, Axel, Jia, Ying, Oh, Jason Z., Tian, Yu
Published in Bioconjugate chemistry (18.10.2023)
Published in Bioconjugate chemistry (18.10.2023)
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Journal Article
Discovery and Early Clinical Development of an Inhibitor of 5‑Lipoxygenase Activating Protein (AZD5718) for Treatment of Coronary Artery Disease
Pettersen, Daniel, Broddefalk, Johan, Emtenäs, Hans, Hayes, Martin A, Lemurell, Malin, Swanson, Marianne, Ulander, Johan, Whatling, Carl, Amilon, Carl, Ericsson, Hans, Westin Eriksson, Annika, Granberg, Kenneth, Plowright, Alleyn T, Shamovsky, Igor, Dellsèn, Anita, Sundqvist, Monica, Någård, Mats, Lindstedt, Eva-Lotte
Published in Journal of medicinal chemistry (09.05.2019)
Published in Journal of medicinal chemistry (09.05.2019)
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