Structure of the Human Dopamine D3 Receptor in Complex with a D2/D3 Selective Antagonist
Chien, Ellen Y.T, Liu, Wei, Zhao, Qiang, Katritch, Vsevolod, Won Han, Gye, Hanson, Michael A, Shi, Lei, Newman, Amy Hauck, Javitch, Jonathan A, Cherezov, Vadim, Stevens, Raymond C
Published in Science (American Association for the Advancement of Science) (19.11.2010)
Published in Science (American Association for the Advancement of Science) (19.11.2010)
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Nanopharmacological Force Sensing to Reveal Allosteric Coupling in Transporter Binding Sites
Zhu, Rong, Sinwel, Doris, Hasenhuetl, Peter S., Saha, Kusumika, Kumar, Vivek, Zhang, Peng, Rankl, Christian, Holy, Marion, Sucic, Sonja, Kudlacek, Oliver, Karner, Andreas, Sandtner, Walter, Stockner, Thomas, Gruber, Hermann J., Freissmuth, Michael, Hauck Newman, Amy, Sitte, Harald H., Hinterdorfer, Peter
Published in Angewandte Chemie (International ed.) (26.01.2016)
Published in Angewandte Chemie (International ed.) (26.01.2016)
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Distinct effects of (R)‐modafinil and its (R)‐ and (S)‐fluoro‐analogs on mesolimbic extracellular dopamine assessed by voltammetry and microdialysis in rats
Keighron, Jacqueline D., Giancola, JoLynn B., Shaffer, Rachel J., DeMarco, Emily M., Coggiano, Mark A., Slack, Rachel D., Newman, Amy Hauck, Tanda, Gianluigi
Published in The European journal of neuroscience (01.08.2019)
Published in The European journal of neuroscience (01.08.2019)
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Yawning and hypothermia in rats : Effects of dopamine D3 and D2 agonists and antagonists
COLLINS, Gregory T, HAUCK NEWMAN, Amy, GRUNDT, Peter, RICE, Kenner C, HUSBANDS, Stephen M, CHAUVIGNAC, Cédric, JIANYONG CHEN, SHAOMENG WANG, WOODS, James H
Published in Psychopharmacologia (01.08.2007)
Published in Psychopharmacologia (01.08.2007)
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PG01037, a novel dopamine D3 receptor antagonist, inhibits the effects of methamphetamine in rats
Higley, Amanda E, Spiller, Krista, Grundt, Peter, Newman, Amy Hauck, Kiefer, Stephen W, Xi, Zheng-Xiong, Gardner, Eliot L
Published in Journal of psychopharmacology (Oxford) (01.02.2011)
Published in Journal of psychopharmacology (Oxford) (01.02.2011)
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Illuminating the monoamine transporters: Fluorescently labelled ligands to study dopamine, serotonin and norepinephrine transporters
Camacho-Hernandez, Gisela Andrea, Jahan, Khorshada, Newman, Amy Hauck
Published in Basic & clinical pharmacology & toxicology (01.11.2023)
Published in Basic & clinical pharmacology & toxicology (01.11.2023)
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Dopamine D3R antagonist VK4-116 attenuates oxycodone self-administration and reinstatement without compromising its antinociceptive effects
You, Zhi-Bing, Bi, Guo-Hua, Galaj, Ewa, Kumar, Vivek, Cao, Jianjing, Gadiano, Alexandra, Rais, Rana, Slusher, Barbara S., Gardner, Eliot L., Xi, Zheng-Xiong, Newman, Amy Hauck
Published in Neuropsychopharmacology (New York, N.Y.) (01.07.2019)
Published in Neuropsychopharmacology (New York, N.Y.) (01.07.2019)
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Are There Prevalent Sex Differences in Psychostimulant Use Disorder? A Focus on the Potential Therapeutic Efficacy of Atypical Dopamine Uptake Inhibitors
Hersey, Melinda, Bartole, Mattingly K, Jones, Claire S, Newman, Amy Hauck, Tanda, Gianluigi
Published in Molecules (Basel, Switzerland) (01.07.2023)
Published in Molecules (Basel, Switzerland) (01.07.2023)
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A bitopic agonist bound to the dopamine 3 receptor reveals a selectivity site
Arroyo-Urea, Sandra, Nazarova, Antonina L, Carrión-Antolí, Ángela, Bonifazi, Alessandro, Battiti, Francisco O, Lam, Jordy Homing, Newman, Amy Hauck, Katritch, Vsevolod, García-Nafría, Javier
Published in Nature communications (05.09.2024)
Published in Nature communications (05.09.2024)
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Dual DAT and sigma receptor inhibitors attenuate cocaine effects on nucleus accumbens dopamine dynamics in rats
Hersey, Melinda, Mereu, Maddalena, Jones, Claire S., Bartole, Mattingly K., Chen, Andy Y., Cao, Jianjing, Hiranita, Takato, Chun, Lauren E., Lopez, Jessica P., Katz, Jonathan L., Newman, Amy Hauck, Tanda, Gianluigi
Published in The European journal of neuroscience (01.05.2024)
Published in The European journal of neuroscience (01.05.2024)
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Journal Article
The binding sites for cocaine and dopamine in the dopamine transporter overlap
Javitch, Jonathan A, Loland, Claus J, Beuming, Thijs, Weinstein, Harel, Bergmann, Marianne L, Shi, Lei, Gether, Ulrik, Kniazeff, Julie, Raniszewska, Klaudia, Gracia, Luis, Newman, Amy Hauck
Published in Nature neuroscience (01.07.2008)
Published in Nature neuroscience (01.07.2008)
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R-Modafinil (Armodafinil): A Unique Dopamine Uptake Inhibitor and Potential Medication for Psychostimulant Abuse
Loland, Claus J, Mereu, Maddalena, Okunola, Oluyomi M, Cao, Jianjing, Prisinzano, Thomas E, Mazier, Sonia, Kopajtic, Theresa, Shi, Lei, Katz, Jonathan L, Tanda, Gianluigi, Newman, Amy Hauck
Published in Biological psychiatry (1969) (01.09.2012)
Published in Biological psychiatry (1969) (01.09.2012)
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Membrane potential shapes regulation of dopamine transporter trafficking at the plasma membrane
Richardson, Ben D, Saha, Kaustuv, Krout, Danielle, Cabrera, Elizabeth, Felts, Bruce, Henry, L Keith, Swant, Jarod, Zou, Mu-Fa, Newman, Amy Hauck, Khoshbouei, Habibeh
Published in Nature communications (25.01.2016)
Published in Nature communications (25.01.2016)
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Applicability of the Dopamine and Rate Hypotheses in Explaining the Differences in Behavioral Pharmacology of the Chloro-Benztropine Analogs: Studies Conducted Using Intracerebral Microdialysis and Population Pharmacodynamic Modeling
Othman, Ahmed A, Newman, Amy Hauck, Eddington, Natalie D
Published in The Journal of pharmacology and experimental therapeutics (01.08.2007)
Published in The Journal of pharmacology and experimental therapeutics (01.08.2007)
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Effects of the selective dopamine D3 receptor antagonist PG01037 on morphine-induced hyperactivity and antinociception in mice
Botz-Zapp, Christian A., Foster, Stephanie L., Pulley, Desta M., Hempel, Briana, Bi, Guo-Hua, Xi, Zheng-Xiong, Newman, Amy Hauck, Weinshenker, David, Manvich, Daniel F.
Published in Behavioural brain research (11.10.2021)
Published in Behavioural brain research (11.10.2021)
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Journal Article
Interactions of calmodulin kinase II with the dopamine transporter facilitate cocaine-induced enhancement of evoked dopamine release
Keighron, Jacqueline D, Bonaventura, Jordi, Li, Yang, Yang, Jae-Won, DeMarco, Emily M, Hersey, Melinda, Cao, Jianjing, Sandtner, Walter, Michaelides, Michael, Sitte, Harald H, Newman, Amy Hauck, Tanda, Gianluigi
Published in Translational psychiatry (13.06.2023)
Published in Translational psychiatry (13.06.2023)
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