A novel small molecule chaperone of rod opsin and its potential therapy for retinal degeneration
Chen, Yuanyuan, Chen, Yu, Jastrzebska, Beata, Golczak, Marcin, Gulati, Sahil, Tang, Hong, Seibel, William, Li, Xiaoyu, Jin, Hui, Han, Yong, Gao, Songqi, Zhang, Jianye, Liu, Xujie, Heidari-Torkabadi, Hossein, Stewart, Phoebe L, Harte, William E, Tochtrop, Gregory P, Palczewski, Krzysztof
Published in Nature communications (17.05.2018)
Published in Nature communications (17.05.2018)
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Primary amines protect against retinal degeneration in mouse models of retinopathies
Maeda, Akiko, Golczak, Marcin, Chen, Yu, Okano, Kiichiro, Kohno, Hideo, Shiose, Satomi, Ishikawa, Kaede, Harte, William, Palczewska, Grazyna, Maeda, Tadao, Palczewski, Krzysztof
Published in Nature chemical biology (25.12.2011)
Published in Nature chemical biology (25.12.2011)
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Potent competitive inhibition of human ribonucleotide reductase by a nonnucleoside small molecule
Ahmad, Md. Faiz, Alam, Intekhab, Huff, Sarah E., Pink, John, Flanagan, Sheryl A., Shewach, Donna, Misko, Tessianna A., Oleinick, Nancy L., Harte, William E., Viswanathan, Rajesh, Harris, Michael E., Dealwis, Chris Godfrey
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (01.08.2017)
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A small molecule mitigates hearing loss in a mouse model of Usher syndrome III
Alagramam, Kumar N, Gopal, Suhasini R, Geng, Ruishuang, Chen, Daniel H-C, Nemet, Ina, Lee, Richard, Tian, Guilian, Miyagi, Masaru, Malagu, Karine F, Lock, Christopher J, Esmieu, William R K, Owens, Andrew P, Lindsay, Nicola A, Ouwehand, Krista, Albertus, Faywell, Fischer, David F, Bürli, Roland W, MacLeod, Angus M, Harte, William E, Palczewski, Krzysztof, Imanishi, Yoshikazu
Published in Nature chemical biology (01.06.2016)
Published in Nature chemical biology (01.06.2016)
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4-Thiazolidinones: Novel inhibitors of the bacterial enzyme MurB
ANDRES, C. J, BRONSON, A. J. J, STOCK, D, YAXIONG SUN, WALSH, A. W, D'ANDREA, A. S. V, DESHPANDE, A. M. S, FALK, P. J, GRANT-YOUNG, K. A, HARTE, W. E, HO, H.-T, MISCO, P. F, ROBERTSON, J. G
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
Published in Bioorganic & medicinal chemistry letters (17.04.2000)
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Small-molecule AgrA inhibitors F12 and F19 act as antivirulence agents against Gram-positive pathogens
Greenberg, Michael, Kuo, David, Jankowsky, Eckhard, Long, Lisa, Hager, Chris, Bandi, Kiran, Ma, Danyang, Manoharan, Divya, Shoham, Yaron, Harte, William, Ghannoum, Mahmoud A, Shoham, Menachem
Published in Scientific reports (01.10.2018)
Published in Scientific reports (01.10.2018)
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pH-Dependent Changes in Photoaffinity Labeling Patterns of the H1 Influenza Virus Hemagglutinin by Using an Inhibitor of Viral Fusion
Cianci, C, Yu, K L, Dischino, D D, Harte, W, Deshpande, M, Luo, G, Colonno, R J, Meanwell, N A, Krystal, M
Published in Journal of Virology (01.03.1999)
Published in Journal of Virology (01.03.1999)
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Journal Article
CD62/P-Selectin Binding Sites for Myeloid Cells and Sulfatides Are Overlapping
Bajorath, Juergen, Hollenbaugh, Diane, King, Gordon, Harte, William, Eustice, David C, Darveau, Richard P, Aruffo, Alejandro
Published in Biochemistry (Easton) (15.02.1994)
Published in Biochemistry (Easton) (15.02.1994)
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Molecular dynamics of HIV-1 protease
Harte, Jr, W E, Swaminathan, S, Beveridge, D L
Published in Proteins, structure, function, and bioinformatics (01.07.1992)
Published in Proteins, structure, function, and bioinformatics (01.07.1992)
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Synergism of Calcium and Carbohydrate Binding to Mammalian Lectin
Harte, William E, Bajorath, Jurgen
Published in Journal of the American Chemical Society (01.11.1994)
Published in Journal of the American Chemical Society (01.11.1994)
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Journal Article
Sulfated Galactocerebrosides as Potential Antiinflammatory Agents
Marinier, Anne, Martel, Alain, Banville, Jacques, Bachand, Carol, Remillard, Roger, Lapointe, Philippe, Turmel, Brigitte, Menard, Marcel, Harte, William E, Wright, J. J. Kim, Todderud, Gordon, Tramposch, Kenneth M, Bajorath, Jürgen, Hollenbaugh, Diane, Aruffo, Alejandro
Published in Journal of medicinal chemistry (26.09.1997)
Published in Journal of medicinal chemistry (26.09.1997)
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Journal Article
Potent competitive inhibition of human ribonucleotide reductase by a nonnucleoside small molecule
Ahmad, Md. Faiz, Alam, Intekhab, Huff, Sarah E., Pink, John, Flanagan, Sheryl A., Shewach, Donna, Misko, Tessianna A., Oleinick, Nancy L., Harte, William E., Viswanathan, Rajesh, Harris, Michael E., Dealwis, Chris Godfrey
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2017)
Published in Proceedings of the National Academy of Sciences - PNAS (17.07.2017)
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ADAAPT: Amgen's data access, analysis, and prediction tools
Cho, Sung Jin, Sun, Yaxiong, Harte, William
Published in Journal of computer-aided molecular design (01.04.2006)
Published in Journal of computer-aided molecular design (01.04.2006)
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Syntheses, Conformations, and Basicities of Bicyclic Triamines
Bell, Thomas W, Choi, Heung-Jin, Harte, William, Drew, Michael G. B
Published in Journal of the American Chemical Society (08.10.2003)
Published in Journal of the American Chemical Society (08.10.2003)
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