Discovery of a Potent and Selective Tyrosine Kinase 2 Inhibitor: TAK-279
Leit, Silvana, Greenwood, Jeremy, Carriero, Samantha, Mondal, Sayan, Abel, Robert, Ashwell, Mark, Blanchette, Heather, Boyles, Nicholas A., Cartwright, Mark, Collis, Alan, Feng, Shulu, Ghanakota, Phani, Harriman, Geraldine C., Hosagrahara, Vinayak, Kaila, Neelu, Kapeller, Rosanna, Rafi, Salma B., Romero, Donna L., Tarantino, Paul M., Timaniya, Jignesh, Toms, Angela V., Wester, Ronald T., Westlin, William, Srivastava, Bhaskar, Miao, Wenyan, Tummino, Peter, McElwee, Joshua J., Edmondson, Scott D., Masse, Craig E.
Published in Journal of medicinal chemistry (10.08.2023)
Published in Journal of medicinal chemistry (10.08.2023)
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Design, Synthesis, and Evaluation of Naphthalene-Sulfonamide Antagonists of Human CCR8
Jenkins, Tracy J, Guan, Bing, Dai, Mingshi, Li, Gang, Lightburn, Thomas E, Huang, Shan, Freeze, B. Scott, Burdi, Douglas F, Jacutin-Porte, Swanee, Bennett, Robert, Chen, Weirong, Minor, Charles, Ghosh, Shomir, Blackburn, Christopher, Gigstad, Kenneth M, Jones, Matthew, Kolbeck, Roland, Yin, Wei, Smith, Sean, Cardillo, Daniel, Ocain, Timothy D, Harriman, Geraldine C
Published in Journal of medicinal chemistry (08.02.2007)
Published in Journal of medicinal chemistry (08.02.2007)
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Journal Article
Potent and selective TYK2-JH1 inhibitors highly efficacious in rodent model of psoriasis
Leit, Silvana, Greenwood, Jeremy R., Mondal, Sayan, Carriero, Samantha, Dahlgren, Markus, Harriman, Geraldine C., Kennedy-Smith, Joshua J., Kapeller, Rosana, Lawson, Jon P., Romero, Donna L., Toms, Angela V., Shelley, Mee, Wester, Ronald T., Westlin, William, McElwee, Joshua J., Miao, Wenyan, Edmondson, Scott D., Masse, Craig E.
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
Published in Bioorganic & medicinal chemistry letters (01.10.2022)
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Selective cell adhesion inhibitors: Barbituric acid based α4β7—MAdCAM inhibitors
Harriman, Geraldine C., Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R., Briskin, Michael J.
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
Published in Bioorganic & medicinal chemistry letters (01.04.2008)
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Journal Article
Selective cell adhesion inhibitors: Barbituric acid based alpha 4 beta 7 - MAdCAM inhibitors
Harriman, Geraldine C, Brewer, Matthias, Bennett, Robert, Kuhn, Cyrille, Bazin, Marc, Larosa, Greg, Skerker, Paul, Cochran, Nancy, Gallant, Debra, Baxter, Deborah, Picarella, Dominic, Jaffee, Bruce, Luly, Jay R, Briskin, Michael J
Published in Bioorganic & medicinal chemistry (01.04.2008)
Published in Bioorganic & medicinal chemistry (01.04.2008)
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ACC Solid forms of a thienopyrimidinedione ACC inhibitor and methods for production thereof
SCOTT MARK E, VARIA KUNAL ARVIND, CALIMSIZ SELCUK, HU SIJUN, HARRIMAN GERALDINE C, VARGHESE VIMAL, YANG XIAOWEI, AMEDIO JOHN C. JR, SABOURIN KYLE, MORRISON HENRY, ALEXANDER KATY, GEIER MICHAEL, WANG XIAOTIAN, LAWSON JON P
Year of Publication 30.08.2024
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Year of Publication 30.08.2024
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ACC Solid forms of a thienopyrimidinedione ACC inhibitor and methods for production thereof
SCOTT MARK E, VARIA KUNAL ARVIND, CALIMSIZ SELCUK, HU SIJUN, HARRIMAN GERALDINE C, VARGHESE VIMAL, YANG XIAOWEI, AMEDIO JOHN C. JR, SABOURIN KYLE, MORRISON HENRY, ALEXANDER KATY, GEIER MICHAEL, WANG XIAOTIAN, LAWSON JON P
Year of Publication 14.03.2023
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Year of Publication 14.03.2023
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ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BHAT SATHESH, HARRIMAN GERALDINE C, HARWOOD JAMES
Year of Publication 30.12.2019
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Year of Publication 30.12.2019
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ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BHAT SATHESH, HARRIMAN GERALDINE C, HARWOOD JAMES
Year of Publication 19.04.2019
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Year of Publication 19.04.2019
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The Chemistry of the Taxane Diterpene: Stereoselective Reductions of Taxanes
Georg, Gunda I, Harriman, Geraldine C. B, Datta, Apurba, Ali, Syed, Cheruvallath, Zacharia, Dutta, Dinah, Vander Velde, David G, Himes, Richard H
Published in Journal of organic chemistry (27.11.1998)
Published in Journal of organic chemistry (27.11.1998)
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피라졸 ACC 억제제 및 그의 용도
GREENWOOD JEREMY ROBERT, LEIT DE MORADEI SILVANA MARCEL, GHOSH SHOMIR, HARRIMAN GERALDINE C
Year of Publication 18.07.2018
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Year of Publication 18.07.2018
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GREENWOOD JEREMY ROBERT, LEIT DE MORADEI SILVANA MARCEL, GHOSH SHOMIR, HARRIMAN GERALDINE C
Year of Publication 18.07.2018
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Year of Publication 18.07.2018
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GREENWOOD JEREMY ROBERT, LEIT DE MORADEI SILVANA MARCEL, GHOSH SHOMIR, HARRIMAN GERALDINE C
Year of Publication 18.07.2018
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Year of Publication 18.07.2018
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ACC 억제제 및 그의 용도
LEIT DE MORADEI SILVANA MARCEL, GHOSH SHOMIR, HARRIMAN GERALDINE C, GREENWOOD JEREMY R
Year of Publication 20.06.2018
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Year of Publication 20.06.2018
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HARWOOD H. JAMES, KAPELLER LIBERMANN ROSANA, HARRIMAN GERALDINE C, WESTLIN WILLIAM F
Year of Publication 08.09.2017
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Year of Publication 08.09.2017
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GREENWOOD JEREMY ROBERT, MASSE CRAIG E, SHELLEY MEE, HARRIMAN GERALDINE C, ROMERO DONNA L, ROBINSON SHAUGHNESSY
Year of Publication 20.12.2016
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Year of Publication 20.12.2016
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LEIT DE MORADEI SILVANA MARCEL, SCHOSTAREZ HEINRICH J, POEL TONI JO, SLOMCZYNSKA URSZULA J, LEIGHTY MATTHEW W, GHOSH SHOMIR, HARRIMAN GERALDINE C, SIMONS LLOYD J, WALKER DANIEL P, MILLER WILLIAM H, LAWSON JON P
Year of Publication 06.11.2019
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Year of Publication 06.11.2019
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GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BORG GEORGE, HARRIMAN GERALDINE C
Year of Publication 20.01.2016
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Year of Publication 20.01.2016
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ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BORG GEORGE, HARRIMAN GERALDINE C
Year of Publication 19.01.2016
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Year of Publication 19.01.2016
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ACC INHIBITORS AND USES THEREOF
GREENWOOD JEREMY ROBERT, MASSE CRAIG E, BORG GEORGE, HARRIMAN GERALDINE C
Year of Publication 14.01.2016
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Year of Publication 14.01.2016
Patent