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Published in PloS one (22.06.2015)
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Thalji, Reema K., McAtee, Jeff J., Belyanskaya, Svetlana, Brandt, Martin, Brown, Gregory D., Costell, Melissa H., Ding, Yun, Dodson, Jason W., Eisennagel, Steve H., Fries, Rusty E., Gross, Jeffrey W., Harpel, Mark R., Holt, Dennis A., Israel, David I., Jolivette, Larry J., Krosky, Daniel, Li, Hu, Lu, Quinn, Mandichak, Tracy, Roethke, Theresa, Schnackenberg, Christine G., Schwartz, Benjamin, Shewchuk, Lisa M., Xie, Wensheng, Behm, David J., Douglas, Stephen A., Shaw, Ami L., Marino, Joseph P.
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In vitro, antithrombotic and bleeding time studies of BMS-654457, a small-molecule, reversible and direct inhibitor of factor XIa
Wong, Pancras C., Quan, Mimi L., Watson, Carol A., Crain, Earl J., Harpel, Mark R., Rendina, Alan R., Luettgen, Joseph M., Wexler, Ruth R., Schumacher, William A., Seiffert, Dietmar A.
Published in Journal of thrombosis and thrombolysis (01.11.2015)
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Albiglutide, a long lasting glucagon-like peptide-1 analog, protects the rat heart against ischemia/reperfusion injury: evidence for improving cardiac metabolic efficiency
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Published in PloS one (26.08.2011)
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Discovery of potent, selective sulfonylfuran urea endothelial lipase inhibitors
Goodman, Krista B., Bury, Michael J., Cheung, Mui, Cichy-Knight, Maria A., Dowdell, Sarah E., Dunn, Allison K., Lee, Dennis, Lieby, Jeffrey A., Moore, Michael L., Scherzer, Daryl A., Sha, Deyou, Suarez, Dominic P., Murphy, Dennis J., Harpel, Mark R., Manas, Eric S., McNulty, Dean E., Annan, Roland S., Matico, Rosalie E., Schwartz, Benjamin K., Trill, John J., Sweitzer, Thomas D., Wang, Da-yuan, Keller, Paul M., Krawiec, John A., Jaye, Michael C.
Published in Bioorganic & medicinal chemistry letters (2009)
Published in Bioorganic & medicinal chemistry letters (2009)
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Tetrahydroquinoline Derivatives as Potent and Selective Factor XIa Inhibitors
Quan, Mimi L, Wong, Pancras C, Wang, Cailan, Woerner, Francis, Smallheer, Joanne M, Barbera, Frank A, Bozarth, Jeffrey M, Brown, Randi L, Harpel, Mark R, Luettgen, Joseph M, Morin, Paul E, Peterson, Tara, Ramamurthy, Vidhyashankar, Rendina, Alan R, Rossi, Karen A, Watson, Carol A, Wei, Anzhi, Zhang, Ge, Seiffert, Dietmar, Wexler, Ruth R
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In Vivo Half-Life Extension of BMP1/TLL Metalloproteinase Inhibitors Using Small-Molecule Human Serum Albumin Binders
Vantourout, Julien C, Mason, Andrew M, Yuen, Josephine, Simpson, Graham L, Evindar, Ghotas, Kuai, Letian, Hobbs, Michael, Edgar, Emma, Needle, Saul, Bai, Xiaopeng, Wilson, Steve, Scott-Stevens, Paul, Traylen, William, Lambert, Kim, Young, Neil, Bunally, Shenaz, Summerfield, Scott G, Snell, Richard, Lad, Rakesh, Shi, Eric, Skinner, Steven, Shewchuk, Lisa, Watson, Allan J.B, Chung, Chun-wa, Pal, Sandeep, Holt, Dennis A, Kallander, Lara S, Prendergast, Joanne, Rivera, Katrina, Washburn, David G, Harpel, Mark R, Arico-Muendel, Christopher, Isidro-Llobet, Albert
Published in Bioconjugate chemistry (17.02.2021)
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Copeland, Robert A, Harpel, Mark R, Tummino, Peter J
Published in Expert opinion on therapeutic targets (01.07.2007)
Published in Expert opinion on therapeutic targets (01.07.2007)
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NADPH oxidase-dependent and -independent mechanisms of reported inhibitors of reactive oxygen generation
Gatto, Gregory J., Ao, Zhaohui, Kearse, Michael G., Zhou, Mei, Morales, Cyndi R., Daniels, Erin, Bradley, Benjamin T., Goserud, Matthew T., Goodman, Krista B., Douglas, Stephen A., Harpel, Mark R., Johns, Douglas G.
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Lawhorn, Brian G., Tran, Tritin, Hong, Victor S., Morgan, Lisa A., Le, BaoChau T., Harpel, Mark R., Jolivette, Larry, Diaz, Elsie, Schwartz, Benjamin, Gross, Jeffrey W., Tomaszek, Thaddeus, Semus, Simon, Concha, Nestor, Smallwood, Angela, Holt, Dennis A., Kallander, Lara S.
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Yue, Tian-Li, Willette, Robert N., Hong, Victor S., Wu, Charlene W., Cui, Jianqi, Krosky, Daniel J., Costell, Melissa H., Schnackenberg, Christine G., Harpel, Mark R.
Published in BioMed research international (01.01.2013)
Published in BioMed research international (01.01.2013)
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Mutagenesis and Mechanism-Based Inhibition of Streptococcus pyogenes Glu-tRNAGln Amidotransferase Implicate a Serine-Based Glutaminase Site
Harpel, Mark R, Horiuchi, Kurumi Y, Luo, Ying, Shen, Li, Jiang, Wenjun, Nelson, David J, Rogers, Kelley C, Decicco, Carl P, Copeland, Robert A
Published in Biochemistry (Easton) (21.05.2002)
Published in Biochemistry (Easton) (21.05.2002)
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Year of Publication 02.05.2023
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Year of Publication 02.05.2023
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Mechanistic Studies of Reaction Coupling in Glu-tRNAGln Amidotransferase
Horiuchi, Kurumi Y, Harpel, Mark R, Shen, Li, Luo, Ying, Rogers, Kelley C, Copeland, Robert A
Published in Biochemistry (Easton) (29.05.2001)
Published in Biochemistry (Easton) (29.05.2001)
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Expression, purification, and characterization of human and rat acetyl coenzyme A carboxylase (ACC) isozymes
Cheng, Dong, Chu, Ching-Hsuen, Chen, Luping, Feder, John N, Mintier, Gabe A, Wu, Yuli, Cook, Joseph W, Harpel, Mark R, Locke, Gregory A, An, Yongmi, Tamura, James K
Published in Protein expression and purification (01.01.2007)
Published in Protein expression and purification (01.01.2007)
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Expression, purification, and characterization of human and rat acetyl cfenzyme A carboxylase (ACC) isozymes
Cheng, Dong, Chu, Ching-Hsuen, Chen, Luping, Feder, John N., Mintier, Gabe A., Wu, Yuli, Cook, Joseph W., Harpel, Mark R., Locke, Gregory A., An, Yongmi, Tamura, James K.
Published in Protein expression and purification (2007)
Published in Protein expression and purification (2007)
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Mutagenesis and Mechanism-Based Inhibition of Streptococcus pyogenes Glu−tRNAGln Amidotransferase Implicate a Serine-Based Glutaminase Site
Harpel, Mark R, Horiuchi, Kurumi Y, Luo, Ying, Shen, Li, Jiang, Wenjun, Nelson, David J, Rogers, Kelley C, Decicco, Carl P, Copeland, Robert A
Published in Biochemistry (Easton) (24.09.2002)
Published in Biochemistry (Easton) (24.09.2002)
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