The Reaction of Grignard Reagents with Bunte Salts: A Thiol-Free Synthesis of Sulfides
Reeves, Jonathan T, Camara, Kaddy, Han, Zhengxu S, Xu, Yibo, Lee, Heewon, Busacca, Carl A, Senanayake, Chris H
Published in Organic letters (21.02.2014)
Published in Organic letters (21.02.2014)
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General and Stereoselective Method for the Synthesis of Sterically Congested and Structurally Diverse P‑Stereogenic Secondary Phosphine Oxides
Han, Zhengxu S, Wu, Hao, Xu, Yibo, Zhang, Yongda, Qu, Bo, Li, Zhibin, Caldwell, Donald R, Fandrick, Keith R, Zhang, Li, Roschangar, Frank, Song, Jinhua J, Senanayake, Chris H
Published in Organic letters (07.04.2017)
Published in Organic letters (07.04.2017)
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Efficient Asymmetric Synthesis of P‑Chiral Phosphine Oxides via Properly Designed and Activated Benzoxazaphosphinine-2-oxide Agents
Han, Zhengxu S, Goyal, Navneet, Herbage, Melissa A, Sieber, Joshua D, Qu, Bo, Xu, Yibo, Li, Zhibin, Reeves, Jonathan T, Desrosiers, Jean-Nicolas, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Mangunuru, Hari P. R, Zhang, Yongda, Krishnamurthy, Dhileep, Lu, Bruce Z, Song, Jinhua J, Wang, Guijun, Senanayake, Chris H
Published in Journal of the American Chemical Society (20.02.2013)
Published in Journal of the American Chemical Society (20.02.2013)
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Copper Catalyzed Regioselective and Stereospecific Aziridine Opening with Pyridyl Grignard Nucleophiles
Lee, Jaehee, Ju, Xuan, Lee, Miseon, Jiang, Qi, Jang, Hwanjong, Kim, Wan Shin, Wu, Linglin, Williams, Suja, Wang, Xiao-Jun, Zeng, Xingzhong, Payne, Jenna, Han, Zhengxu S
Published in Organic letters (15.04.2022)
Published in Organic letters (15.04.2022)
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A Practical Procedure for Reduction of Primary, Secondary and Tertiary Amides to Amines
Reeves, Jonathan T., Tan, Zhulin, Marsini, Maurice A., Han, Zhengxu S., Xu, Yibo, Reeves, Diana C., Lee, Heewon, Lu, Bruce Z., Senanayake, Chris H.
Published in Advanced synthesis & catalysis (14.01.2013)
Published in Advanced synthesis & catalysis (14.01.2013)
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Efficient Asymmetric Synthesis of Structurally Diverse P-Stereogenic Phosphinamides for Catalyst Design
Han, Zhengxu S., Zhang, Li, Xu, Yibo, Sieber, Joshua D., Marsini, Maurice A., Li, Zhibin, Reeves, Jonathan T., Fandrick, Keith R., Patel, Nitinchandra D., Desrosiers, Jean-Nicolas, Qu, Bo, Chen, Anji, Rudzinski, DiAndra M., Samankumara, Lalith P., Ma, Shengli, Grinberg, Nelu, Roschangar, Frank, Yee, Nathan K., Wang, Guijun, Song, Jinhua J., Senanayake, Chris H.
Published in Angewandte Chemie (International ed.) (27.04.2015)
Published in Angewandte Chemie (International ed.) (27.04.2015)
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Rhodium‐Catalyzed Addition of Aryl Boronic Acids to 2,2‐Disubstituted Malononitriles
Malapit, Christian A., Caldwell, Donald R., Luvaga, Irungu K., Reeves, Jonathan T., Volchkov, Ivan, Gonnella, Nina C., Han, Zhengxu S., Busacca, Carl A., Howell, Amy R., Senanayake, Chris H.
Published in Angewandte Chemie International Edition (06.06.2017)
Published in Angewandte Chemie International Edition (06.06.2017)
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P‐Stereogenic Chiral Phosphine−Palladium Complex Catalyzed Enantioselective Synthesis of Phosphoryl‐Substituted Atropisomeric Vinylarenes
Wu, Hao, Han, Zhengxu S., Qu, Bo, Wang, Dan, Zhang, Yongda, Xu, Yibo, Grinberg, Nelu, Lee, Heewon, Song, Jinhua J., Roschangar, Frank, Wang, Guijun, Senanayake, Chris H.
Published in Advanced synthesis & catalysis (23.11.2017)
Published in Advanced synthesis & catalysis (23.11.2017)
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A Mild Dihydrobenzooxaphosphole Oxazoline/Iridium Catalytic System for Asymmetric Hydrogenation of Unfunctionalized Dialins
Qu, Bo, Samankumara, Lalith P., Ma, Shengli, Fandrick, Keith R., Desrosiers, Jean-Nicolas, Rodriguez, Sonia, Li, Zhibin, Haddad, Nizar, Han, Zhengxu S., McKellop, Keith, Pennino, Scott, Grinberg, Nelu, Gonnella, Nina C., Song, Jinhua J., Senanayake, Chris H.
Published in Angewandte Chemie (International ed.) (22.12.2014)
Published in Angewandte Chemie (International ed.) (22.12.2014)
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Amine-Tunable Ruthenium Catalysts for Asymmetric Reduction of Ketones
Rodríguez, Sonia, Qu, Bo, Fandrick, Keith R., Buono, Frederic, Haddad, Nizar, Xu, Yibo, Herbage, Melissa A., Zeng, Xingzhong, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Han, Zhengxu S., Yee, Nathan K., Senanayake, Chris H.
Published in Advanced synthesis & catalysis (10.02.2014)
Published in Advanced synthesis & catalysis (10.02.2014)
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Journal Article
Development of a Large-Scale Asymmetric Process for tert-Butanesulfinamide
DeCroos, Philomen, Han, Zhengxu S, Sidhu, Kanwar, Lorenz, Jon, Nummy, Larry, Byrne, Denis, Qu, Bo, Xu, Yibo, Wu, Ling, Lee, Heewon, Roschangar, Frank, Song, Jinhua J, Senanayake, Chris H
Published in Organic process research & development (15.02.2019)
Published in Organic process research & development (15.02.2019)
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Journal Article
Carbamoyl Anion Addition to N‑Sulfinyl Imines: Highly Diastereoselective Synthesis of α‑Amino Amides
Reeves, Jonathan T, Tan, Zhulin, Herbage, Melissa A, Han, Zhengxu S, Marsini, Maurice A, Li, Zhibin, Li, Guisheng, Xu, Yibo, Fandrick, Keith R, Gonnella, Nina C, Campbell, Scot, Ma, Shengli, Grinberg, Nelu, Lee, Heewon, Lu, Bruce Z, Senanayake, Chris H
Published in Journal of the American Chemical Society (17.04.2013)
Published in Journal of the American Chemical Society (17.04.2013)
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Green Chemistry Articles of Interest to the Pharmaceutical Industry
Bryan, Marian C, Dalton, Charlotte, Díaz-Rodríguez, Alba, Doerfler, Jaika, Engl, Oliver D, Ferguson, Paul, Molina, Alejandro Gimenez, Han, Zhengxu S, Hosford, Joseph, Howell, Gareth P, Hutchby, Marc, Li, Wei, Munday, Rachel H, Navarro, Antonio, Parmentier, Michael, Pawlas, Jan, Richardson, Paul F, Smith, William J, Steven, Alan, Takale, Balaram S, Terrett, Jack A, Treitler, Daniel S, Zeng, Mingshuo
Published in Organic process research & development (18.02.2022)
Published in Organic process research & development (18.02.2022)
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Rational Design of New Dihydrobenzooxophosphole-Based Lewis Base Organocatalysts
Qu, Bo, Samankumara, Lalith P., Saha, Anjan, Schumer, Mac G., Han, Zhengxu S., Haddad, Nizar, Busacca, Carl A., Yee, Nathan K., Kozlowski, Marisa C., Song, Jinghua J., Senanayake, Chris H.
Published in Synlett (01.04.2020)
Published in Synlett (01.04.2020)
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Development of New P‑Chiral P,π-Dihydrobenzooxaphosphole Hybrid Ligands for Asymmetric Catalysis
Sieber, Joshua D, Chennamadhavuni, Divya, Fandrick, Keith R, Qu, Bo, Han, Zhengxu S, Savoie, Jolaine, Ma, Shengli, Samankumara, Lalith P, Grinberg, Nelu, Lee, Heewon, Song, Jinhua J, Senanayake, Chris H
Published in Organic letters (17.10.2014)
Published in Organic letters (17.10.2014)
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Development of a Scalable, Chromatography-Free Synthesis of t‑Bu-SMS-Phos and Application to the Synthesis of an Important Chiral CF3‑Alcohol Derivative with High Enantioselectivity Using Rh-Catalyzed Asymmetric Hydrogenation
Sieber, Joshua D, Rodriguez, Sonia, Frutos, Rogelio, Buono, Frederic, Zhang, Yongda, Li, Ning, Qu, Bo, Premasiri, Ajith, Li, Zhibin, Han, Zhengxu S, Xu, Yibo, Byrne, Denis, Haddad, Nizar, Lorenz, Jon, Grinberg, Nelu, Kurouski, Dmitry, Lee, Heewon, Narayanan, Bikshandarkoil, Nummy, Laurence, Mulder, Jason, Brown, Jack D, Granger, Alice, Gao, Joe, Krawiec, Mariusz, Williams, Zeena, Pennino, Scott, Song, Jinhua J, Hossain, Azad, Yee, Nathan K, Busacca, Carl, Roschangar, Frank, Xin, Yanchao, Mao, Zhantong, Zhang, Xinzhu, Hong, Yaping, Senanayake, Chris H
Published in Journal of organic chemistry (02.02.2018)
Published in Journal of organic chemistry (02.02.2018)
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Journal Article
Metal-Free Cycloetherification by in Situ Generated P‑Stereogenic α‑Diazanium Intermediates: A Convergent Synthesis of Enantiomerically Pure Dihydrobenzooxaphospholes
Li, Shi-Guang, Han, Zhengxu S, Viereck, Peter, Lee, Heewon, Kurouski, Dmitry, Senanayake, Chris H, Tsantrizos, Youla S
Published in Organic letters (17.02.2017)
Published in Organic letters (17.02.2017)
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Green Chemistry Articles of Interest to the Pharmaceutical Industry
Dalton, Charlotte, Diorazio, Louis J, Doerfler, Jaika, Engl, Oliver D, Han, Zhengxu S, Howell, Gareth P, Latham, Jonathan, Li, Wei, McLaws, Mark, Munday, Rachel H, Navarro, Antonio, Parmentier, Michael, Pawlas, Jan, Richardson, Paul, Roiban, Gheorghe-Doru, Steven, Alan, Terrett, Jack A, Treitler, Daniel S, Zeng, Mingshuo
Published in Organic process research & development (16.04.2021)
Published in Organic process research & development (16.04.2021)
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Journal Article
Modular Dihydrobenzoazaphosphole Ligands for Suzuki-Miyaura Cross-Coupling
Zhang, Yongda, Lao, Kendricks S., Sieber, Joshua D., Xu, Yibo, Wu, Linglin, Wang, Xiao-Jun, Desrosiers, Jean-Nicolas, Lee, Heewon, Haddad, Nizar, Han, Zhengxu S., Yee, Nathan K., Song, Jinhua J., Howell, Amy R., Senanayake, Chris H.
Published in Synthesis (Stuttgart) (01.11.2018)
Published in Synthesis (Stuttgart) (01.11.2018)
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