Discovery of an Oral Potent Selective Inhibitor of Hematopoietic Prostaglandin D Synthase (HPGDS)
Carron, Chris P, Trujillo, John I, Olson, Kirk L, Huang, Wei, Hamper, Bruce C, Dice, Tom, Neal, Bradley E, Pelc, Matthew J, Day, Jacqueline E, Rohrer, Douglas C, Kiefer, James R, Moon, Joseph B, Schweitzer, Barbara A, Blake, Tanisha D, Turner, Steve R, Woerndle, Rhonda, Case, Brenda L, Bono, Christine P, Dilworth, Vickie M, Funckes-Shippy, Christie L, Hood, Becky L, Jerome, Gina M, Kornmeier, Christine M, Radabaugh, Melissa R, Williams, Melanie L, Davies, Michael S, Wegner, Craig D, Welsch, Dean J, Abraham, William M, Warren, Chad J, Dowty, Martin E, Hua, Fengmei, Zutshi, Anup, Yang, Jerry Z, Thorarensen, Atli
Published in ACS medicinal chemistry letters (13.05.2010)
Published in ACS medicinal chemistry letters (13.05.2010)
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Journal Article
Support of academic synthetic chemistry using separation technologies from the pharmaceutical industry
Regalado, Erik L, Kozlowski, Marisa C, Curto, John M, Ritter, Tobias, Campbell, Michael G, Mazzotti, Anthony R, Hamper, Bruce C, Spilling, Christopher D, Mannino, Michael P, Wan, Li, Yu, Jin-Quan, Liu, Jinchu, Welch, Christopher J
Published in Organic & biomolecular chemistry (14.04.2014)
Published in Organic & biomolecular chemistry (14.04.2014)
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Journal Article
Discovery of N‑(4-Fluoro-3-methoxybenzyl)-6-(2-(((2S,5R)‑5-(hydroxymethyl)-1,4-dioxan-2-yl)methyl)‑2H‑tetrazol-5-yl)-2-methylpyrimidine-4-carboxamide. A Highly Selective and Orally Bioavailable Matrix Metalloproteinase-13 Inhibitor for the Potential Treatment of Osteoarthritis
Ruminski, Peter G, Massa, Mark, Strohbach, Joseph, Hanau, Cathleen E, Schmidt, Michelle, Scholten, Jeffrey A, Fletcher, Theresa R, Hamper, Bruce C, Carroll, Jeffery N, Shieh, Huey S, Caspers, Nicole, Collins, Brandon, Grapperhaus, Margaret, Palmquist, Katherine E, Collins, Joe, Baldus, John E, Hitchcock, Jeffrey, Kleine, H. Peter, Rogers, Michael D, McDonald, Joseph, Munie, Grace E, Messing, Dean M, Portolan, Silvia, Whiteley, Laurence O, Sunyer, Teresa, Schnute, Mark E
Published in Journal of medicinal chemistry (14.01.2016)
Published in Journal of medicinal chemistry (14.01.2016)
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Journal Article
Enantioseparation of α-Hydroxyallylphosphonates and Phosphonoallylic Carbonate Derivatives on Chiral Stationary Phases Using Sequential UV, Polarimetric, and Refractive Index Detection
Hamper, Bruce C., Mannino, Michael P., Mueller, Melissa E., Harrison, Liam T., Spilling, Christopher D.
Published in Chirality (New York, N.Y.) (01.09.2016)
Published in Chirality (New York, N.Y.) (01.09.2016)
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Journal Article
Discovery of (pyridin-4-yl)-2H-tetrazole as a novel scaffold to identify highly selective matrix metalloproteinase-13 inhibitors for the treatment of osteoarthritis
SCHNUTE, Mark E, O'BRIEN, Patrick M, CARROLL, Jeffery N, PATT, William C, SHIEH, Huey S, COLLINS, Brandon, PAVLOVSKY, Alexander G, PALMQUIST, Katherine E, ASTON, Karl W, HITCHCOCK, Jeffrey, ROGERS, Michael D, MCDONALD, Joseph, NAHRA, Joe, JOHNSON, Adam R, MUNIE, Grace E, WITTWER, Arthur J, MAN, Chiu-Fai, SETTLE, Steven L, NEMIROVSKIY, Olga, VICKERY, Lillian E, AGAWAL, Arun, DYER, Richard D, SUNYER, Teresa, MORRIS, Mark, HOWARD ROARK, W, HANAU, Cathleen E, RUMINSKI, Peter G, SCHOLTEN, Jeffrey A, FLETCHER, Theresa R, HAMPER, Bruce C
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
Published in Bioorganic & medicinal chemistry letters (15.01.2010)
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Journal Article
Structure-based parallel medicinal chemistry approach to improve metabolic stability of benzopyran COX-2 inhibitors
Xing, Li, Hamper, Bruce C., Fletcher, Theresa R., Wendling, Jay M., Carter, Jeffery, Gierse, James K., Liao, Subo
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
Published in Bioorganic & medicinal chemistry letters (01.02.2011)
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Journal Article
Synthesis of highly substituted 5-(trifluoromethyl)ketoimidazoles using a mixed-solid/solution phase motif
Hamper, Bruce C., Jerome, Kevin D., Yalamanchili, Gopi, Walker, Daniel M., Chott, Robert C., Mischke, Deborah A.
Published in Biotechnology and bioengineering (2000)
Published in Biotechnology and bioengineering (2000)
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Journal Article
Solid Phase Synthesis of β-Peptoids: N-Substituted β-Aminopropionic Acid Oligomers
Hamper, Bruce C, Kolodziej, Stephen A, Scates, Angela M, Smith, Ronald G, Cortez, Enriqueta
Published in Journal of organic chemistry (06.02.1998)
Published in Journal of organic chemistry (06.02.1998)
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Journal Article
Corroboration of techniques for assigning absolute configuration: lacinilene C methyl ether as an exemplary study
Stipanovic, Robert D, McCormick, John P, Schlemper, Elmer O, Hamper, Bruce C, Shinmyozu, Teruo, Pirkle, William H
Published in Journal of organic chemistry (01.06.1986)
Published in Journal of organic chemistry (01.06.1986)
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Journal Article
A Practical Gram-Scale Synthesis of Acrylohydroxamic Acid
Hamper, Bruce C., Sullivan, Brendan T., Rath, Nigam P., Spilling, Christopher D.
Published in Synthesis (Stuttgart) (18.12.2017)
Published in Synthesis (Stuttgart) (18.12.2017)
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Journal Article
Enantioseparation of [alpha]-Hydroxyallylphosphonates and Phosphonoallylic Carbonate Derivatives on Chiral Stationary Phases Using Sequential UV, Polarimetric, and Refractive Index Detection
Hamper, Bruce C, Mannino, Michael P, Mueller, Melissa E, Harrison, Liam T, Spilling, Christopher D
Published in Chirality (New York, N.Y.) (01.09.2016)
Published in Chirality (New York, N.Y.) (01.09.2016)
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Journal Article
Synthesis and Herbicidal Activity of 3-Aryl-5-(haloalkyl)-4-isoxazolecarboxamides and Their Derivatives
Hamper, Bruce C, Leschinsky, Kindrick L, Massey, Steven S, Bell, Crystal L, Brannigan, Lawrence H, Prosch, S. Douglas
Published in Journal of agricultural and food chemistry (01.01.1995)
Published in Journal of agricultural and food chemistry (01.01.1995)
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