Search Results - "HAMELINK, Elizabeth" :: K.UTB vyhledávací portál | TBU Library Retrieval Portal

Biological and computational evaluation of resveratrol inhibitors against Alzheimer's disease

Biological and computational evaluation of resveratrol inhibitors against Alzheimer's disease

by Koukoulitsa, Catherine, Villalonga-Barber, Caroline, Csonka, Robert, Alexi, Xanthippi, Leonis, Georgios, Dellis, Dimitris, Hamelink, Elizabeth, Belda, Oscar, Steele, Barry R., Micha-Screttas, Maria, Alexis, Michael N., Papadopoulos, Manthos G., Mavromoustakos, Thomas
Published in Journal of enzyme inhibition and medicinal chemistry (02.01.2016)

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Structure–activity relationship study on a novel series of cyclopentane-containing macrocyclic inhibitors of the hepatitis C virus NS3/4A protease leading to the discovery of TMC435350

Structure–activity relationship study on a novel series of cyclopentane-containing macrocyclic inhibitors of the hepatitis C virus NS3/4A protease leading to the discovery of TMC435350

by Raboisson, Pierre, de Kock, Herman, Rosenquist, Åsa, Nilsson, Magnus, Salvador-Oden, Lourdes, Lin, Tse-I, Roue, Natalie, Ivanov, Vladimir, Wähling, Horst, Wickström, Kristina, Hamelink, Elizabeth, Edlund, Michael, Vrang, Lotta, Vendeville, Sandrine, Van de Vreken, Wim, McGowan, David, Tahri, Abdellah, Hu, Lili, Boutton, Carlo, Lenz, Oliver, Delouvroy, Frederic, Pille, Geert, Surleraux, Dominique, Wigerinck, Piet, Samuelsson, Bertil, Simmen, Kenneth
Published in Bioorganic & medicinal chemistry (01.09.2008)

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Synthesis and SAR of potent inhibitors of the Hepatitis C virus NS3/4A protease: Exploration of P2 quinazoline substituents

Synthesis and SAR of potent inhibitors of the Hepatitis C virus NS3/4A protease: Exploration of P2 quinazoline substituents

by Nilsson, Magnus, Belfrage, Anna Karin, Lindström, Stefan, Wähling, Horst, Lindquist, Charlotta, Ayesa, Susana, Kahnberg, Pia, Pelcman, Mikael, Benkestock, Kurt, Agback, Tatiana, Vrang, Lotta, Terelius, Ylva, Wikström, Kristina, Hamelink, Elizabeth, Rydergård, Christina, Edlund, Michael, Eneroth, Anders, Raboisson, Pierre, Lin, Tse-I, de Kock, Herman, Wigerinck, Piet, Simmen, Kenneth, Samuelsson, Bertil, Rosenquist, Åsa
Published in Bioorganic & medicinal chemistry letters (15.07.2010)

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Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II

Synthesis, biological evaluation, and modeling studies of inhibitors aimed at the malarial proteases plasmepsins I and II

by Muthas, Daniel, Nöteberg, Daniel, Sabnis, Yogesh A., Hamelink, Elizabeth, Vrang, Lotta, Samuelsson, Bertil, Karlén, Anders, Hallberg, Anders
Published in Bioorganic & medicinal chemistry (15.09.2005)

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Design and synthesis of potent macrocyclic renin inhibitors

Design and synthesis of potent macrocyclic renin inhibitors

by Sund, Christian, Belda, Oscar, Wiktelius, Daniel, Sahlberg, Christer, Vrang, Lotta, Sedig, Susanne, Hamelink, Elizabeth, Henderson, Ian, Agback, Tatiana, Jansson, Katarina, Borkakoti, Neera, Derbyshire, Dean, Eneroth, Anders, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry letters (01.01.2011)

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Potent Inhibitors of the Plasmodium falciparum Enzymes Plasmepsin I and II Devoid of Cathepsin D Inhibitory Activity

Potent Inhibitors of the Plasmodium falciparum Enzymes Plasmepsin I and II Devoid of Cathepsin D Inhibitory Activity

by ERSMARK, Karolina, FEIERBERG, Isabella, BJELIC, Sinisa, HAMELINK, Elizabeth, HACKETT, Fiona, BLACKMAN, Michael J., HULTéN, Johan, SAMUELSSON, Bertil, ÅQVIST, Johan, HALLBERG, Anders
Published in Journal of medicinal chemistry (01.01.2004)

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Design and synthesis of potent hydroxyethylamine (HEA) BACE-1 inhibitors carrying prime side 4,5,6,7-tetrahydrobenzazole and 4,5,6,7-tetrahydropyridinoazole templates

Design and synthesis of potent hydroxyethylamine (HEA) BACE-1 inhibitors carrying prime side 4,5,6,7-tetrahydrobenzazole and 4,5,6,7-tetrahydropyridinoazole templates

by Sund, Christian, Belda, Oscar, Borkakoti, Neera, Lindberg, Jimmy, Derbyshire, Dean, Vrang, Lotta, Hamelink, Elizabeth, Åhgren, Cathrine, Woestenenk, Esmeralda, Wikström, Kristina, Eneroth, Anders, Lindström, Erik, Kalayanov, Genadiy
Published in Bioorganic & medicinal chemistry letters (01.11.2012)

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Synthesis of Malarial Plasmepsin Inhibitors and Prediction of Binding Modes by Molecular Dynamics Simulations

Synthesis of Malarial Plasmepsin Inhibitors and Prediction of Binding Modes by Molecular Dynamics Simulations

by Ersmark, Karolina, Nervall, Martin, Hamelink, Elizabeth, Janka, Linda K, Clemente, Jose C, Dunn, Ben M, Blackman, Michael J, Samuelsson, Bertil, Åqvist, Johan, Hallberg, Anders
Published in Journal of medicinal chemistry (22.09.2005)

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Design and Synthesis of Plasmepsin I and Plasmepsin II Inhibitors with Activity in Plasmodium falciparum-Infected Cultured Human Erythrocytes

Design and Synthesis of Plasmepsin I and Plasmepsin II Inhibitors with Activity in Plasmodium falciparum-Infected Cultured Human Erythrocytes

by NöTEBERG, Daniel, HAMELINK, Elizabeth, HULTéN, Johan, WAHLGREN, Mats, VRANG, Lotta, SAMUELSSON, Bertil, HALLBERG, Anders
Published in Journal of medicinal chemistry (27.02.2003)

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Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs

Novel potent macrocyclic inhibitors of the hepatitis C virus NS3 protease: Use of cyclopentane and cyclopentene P2-motifs

by Bäck, Marcus, Johansson, Per-Ola, Wångsell, Fredrik, Thorstensson, Fredrik, Kvarnström, Ingemar, Ayesa, Susana, Wähling, Horst, Pelcman, Mikael, Jansson, Katarina, Lindström, Stefan, Wallberg, Hans, Classon, Björn, Rydergård, Christina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (15.11.2007)

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New potent C2-Symmetric malaria plasmepsin I and II inhibitors

New potent C2-Symmetric malaria plasmepsin I and II inhibitors

by OSCARSSON, Karin, OSCARSON, Stefan, VRANG, Lotta, HAMELINK, Elizabeth, HALLBERG, Anders, SAMUELSSON, Bertil
Published in Bioorganic & medicinal chemistry (03.04.2003)

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Potent inhibitors of the hepatitis C virus NS3 protease: Use of a novel P2 cyclopentane-derived template

Potent inhibitors of the hepatitis C virus NS3 protease: Use of a novel P2 cyclopentane-derived template

by Johansson, Per-Ola, Bäck, Marcus, Kvarnström, Ingemar, Jansson, Katarina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (01.08.2006)

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Design and Synthesis of Potent Inhibitors of the Malaria Aspartyl Proteases Plasmepsin I and II. Use of Solid-Phase Synthesis to Explore Novel Statine Motifs

Design and Synthesis of Potent Inhibitors of the Malaria Aspartyl Proteases Plasmepsin I and II. Use of Solid-Phase Synthesis to Explore Novel Statine Motifs

by Johansson, Per-Ola, Chen, Yantao, Belfrage, Anna Karin, Blackman, Michael J, Kvarnström, Ingemar, Jansson, Katarina, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Journal of medicinal chemistry (17.06.2004)

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Macrocyclic inhibitors of the malarial aspartic proteases plasmepsin I, II, and IV

Macrocyclic inhibitors of the malarial aspartic proteases plasmepsin I, II, and IV

by Ersmark, Karolina, Nervall, Martin, Gutiérrez-de-Terán, Hugo, Hamelink, Elizabeth, Janka, Linda K., Clemente, Jose C., Dunn, Ben M., Gogoll, Adolf, Samuelsson, Bertil, Åqvist, Johan, Hallberg, Anders
Published in Bioorganic & medicinal chemistry (01.04.2006)

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Design and Synthesis of Potent Inhibitors of Plasmepsin I and II: X-ray Crystal Structure of Inhibitor in Complex with Plasmepsin II

Design and Synthesis of Potent Inhibitors of Plasmepsin I and II: X-ray Crystal Structure of Inhibitor in Complex with Plasmepsin II

by Johansson, Per-Ola, Lindberg, Jimmy, Blackman, Michael J, Kvarnström, Ingemar, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Journal of medicinal chemistry (30.06.2005)

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New potent C 2 -Symmetric malaria plasmepsin I and II inhibitors

New potent C 2 -Symmetric malaria plasmepsin I and II inhibitors

by Oscarsson, Karin, Oscarson, Stefan, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (03.04.2003)

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Synthesis of novel potent hepatitis C virus NS3 protease inhibitors: Discovery of 4-hydroxy-cyclopent-2-ene-1,2-dicarboxylic acid as a N-acyl- l-hydroxyproline bioisostere

Synthesis of novel potent hepatitis C virus NS3 protease inhibitors: Discovery of 4-hydroxy-cyclopent-2-ene-1,2-dicarboxylic acid as a N-acyl- l-hydroxyproline bioisostere

by Thorstensson, Fredrik, Wångsell, Fredrik, Kvarnström, Ingemar, Vrang, Lotta, Hamelink, Elizabeth, Jansson, Katarina, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (2007)

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Solid-phase library synthesis of reversed-statine type inhibitors of the malarial aspartyl proteases plasmepsin I and II

Solid-phase library synthesis of reversed-statine type inhibitors of the malarial aspartyl proteases plasmepsin I and II

by Dahlgren, Anders, Kvarnström, Ingemar, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (20.03.2003)

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New inhibitors of the malaria aspartyl proteases plasmepsin I and II

New inhibitors of the malaria aspartyl proteases plasmepsin I and II

by Dahlgren, Anders, Kvarnström, Ingemar, Vrang, Lotta, Hamelink, Elizabeth, Hallberg, Anders, Rosenquist, Åsa, Samuelsson, Bertil
Published in Bioorganic & medicinal chemistry (05.08.2003)

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Design and Synthesis of Plasmepsin I and Plasmepsin II Inhibitors with Activity in Plasmodium f alciparum-Infected Cultured Human Erythrocytes

Design and Synthesis of Plasmepsin I and Plasmepsin II Inhibitors with Activity in Plasmodium f alciparum-Infected Cultured Human Erythrocytes

by Nöteberg, Daniel, Hamelink, Elizabeth, Hultén, Johan, Wahlgren, Mats, Vrang, Lotta, Samuelsson, Bertil, Hallberg, Anders
Published in Journal of medicinal chemistry (27.02.2003)

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