RP-3500: A Novel, Potent, and Selective ATR Inhibitor that is Effective in Preclinical Models as a Monotherapy and in Combination with PARP Inhibitors
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A novel high throughput screening assay for HCV NS3 helicase activity
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Published in Antiviral research (01.06.2000)
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Black, W. Cameron, Abdoli, Abbas, An, Xiuli, Auger, Anick, Beaulieu, Patrick, Bernatchez, Michel, Caron, Cathy, Chefson, Amandine, Crane, Sheldon, Diallo, Mohamed, Dorich, Stéphane, Fader, Lee D., Ferraro, Gino B., Fournier, Sara, Gao, Qi, Ginzburg, Yelena, Hamel, Martine, Han, Yongshuai, Jones, Paul, Lanoix, Stéphanie, Lacbay, Cyrus M., Leclaire, Marie-Eve, Levy, Maayan, Mamane, Yael, Mulani, Amina, Papp, Robert, Pellerin, Charles, Picard, Audrey, Skeldon, Alexander, Skorey, Kathryn, Stocco, Rino, St.-Onge, Miguel, Truchon, Jean-François, Truong, Vouy Linh, Zimmermann, Michal, Zinda, Michael, Roulston, Anne
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The R1 Subunit of Herpes Simplex Virus Ribonucleotide Reductase Is a Good Substrate for Host Cell Protein Kinases but Is Not Itself a Protein Kinase
Langelier, Yves, Champoux, Louise, Hamel, Martine, Guilbault, Claire, Lamarche, Nathalie, Gaudreau, Pierrette, Massie, Bernard
Published in The Journal of biological chemistry (16.01.1998)
Published in The Journal of biological chemistry (16.01.1998)
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Abstract P054: RP-3500: A novel, potent and selective ATR inhibitor that is effective in pre-clinical models as a monotherapy and in combination with PARP inhibitors
Roulston, Anne, Zimmerman, Michal, Papp, Robert, Skeldon, Alex, Pellerin, Charles, Dumas-Bérube, Émilie, Dumais, Valerie, Dorich, Stephane, Fournier, Sara, Li, Li, Leclaire, Marie-Ève, Yin, Shou Yun, Chefson, Amandine, Alam, Hunain, Yang, William, Fugère-Desjardins, Chloe, Hammond, Sabrina, Skorey, Kathryn, Mulani, Amina, Rimkunas, Victoria, Veloso, Artur, Hamel, Martine, Stocco, Rino, Mamane, Yael, Li, Zuomei, Young, Jordan, Zinda, Mike, Black, Cameron
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Published in Molecular cancer therapeutics (01.12.2021)
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identification of 4,7-disubstituted naphthoic acid derivatives as UDP-competitive antagonists of P2Y
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Published in Bioorganic & medicinal chemistry letters (15.05.2011)
Published in Bioorganic & medicinal chemistry letters (15.05.2011)
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Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCV NS5B polymerase and HCV subgenomic RNA replication. Part 2: Tertiary amides
Chan, Laval, Pereira, Oswy, Reddy, T.Jagadeeswar, Das, Sanjoy K., Poisson, Carl, Courchesne, Marc, Proulx, Mélanie, Siddiqui, Arshad, Yannopoulos, Constantin G., Nguyen-Ba, Nghe, Roy, Caroline, Nasturica, Daniel, Moinet, Christophe, Bethell, Richard, Hamel, Martine, L'Heureux, Lucille, David, Maud, Nicolas, Olivier, Courtemanche-Asselin, Philippe, Brunette, Stéphanie, Bilimoria, Darius, Bédard, Jean
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Guay, Daniel, Beaulieu, Christian, Belley, Michel, Crane, Sheldon N, DeLuca, Jeancarlo, Gareau, Yves, Hamel, Martine, Henault, Martin, Hyjazie, Huda, Kargman, Stacia, Chan, Chi Chung, Xu, Lijing, Gordon, Robert, Li, Lianhai, Mamane, Yael, Morin, Nicolas, Mancini, Joseph, Thérien, Michel, Tranmer, Geoffrey, Truong, Vouy Linh, Wang, Zhaoyin, Black, W. Cameron
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Published in Bioorganic & medicinal chemistry letters (15.01.2011)
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New indole amide derivatives as potent CRTH2 receptor antagonists
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Hamel, Martine, Henault, Martin, Hyjazie, Huda, Morin, Nicolas, Bayly, Christopher, Skorey, Kathryn, Therien, Alex G, Mancini, Joseph, Brideau, Christine, Kargman, Stacia
Published in Journal of biomolecular screening (01.10.2011)
Published in Journal of biomolecular screening (01.10.2011)
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Discovery of thiophene-2-carboxylic acids as potent inhibitors of HCV NS5B polymerase and HCV subgenomic RNA replication. Part 1: Sulfonamides
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